ARTICLE
|
doi:10.20944/preprints202404.1701.v1
Subject:
Computer Networks And Communications,
Computer Science And Mathematics
Keywords:
Cryptographic; Private Set Intersection; Cuckoo Filter; Cloud Assistance; Private Contact Discovery)
Online: 26 April 2024 (00:14:06 CEST)
REVIEW
|
doi:10.20944/preprints202404.1013.v3
Subject:
Pharmacy,
Medicine And Pharmacology
Keywords:
computational pharmaceutics; AI; multi-scale modeling; quantum computing; drug discovery; blockchain frameworks
Online: 22 April 2024 (18:38:54 CEST)
REVIEW
|
doi:10.20944/preprints202404.0437.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
neurodegenerative diseases; Parkinson’ s disease; Alzheimer’ s disease; drug discovery; disease-modifying drugs
Online: 5 April 2024 (12:39:57 CEST)
REVIEW
|
doi:10.20944/preprints202404.0055.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Lead optimization; drug discovery; artificial intelligence; machine learning; deep neural networks; cheminformatics; chemical modifications; drug development
Online: 1 April 2024 (13:35:22 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1775.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Hepatitis B virus; Antivirals; Flavonoid; Drug discovery; Pharmacophore; Quantitative structure-activity relationship
Online: 28 March 2024 (13:31:24 CET)
ARTICLE
|
doi:10.20944/preprints202210.0223.v3
Subject:
Biology And Life Sciences,
Virology
Keywords:
Drug discovery; Systems biology; SARS-CoV-2; Dengue; Influenza A; RSV; cell viability analysis; antivirals; in vitro validation; in vivo validation
Online: 22 March 2024 (16:46:59 CET)
ARTICLE
|
doi:10.20944/preprints202402.0943.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
degradation monitoring; health monitoring; causal discovery; jaccard distance, inter- 14 pretability; causal interpretability
Online: 19 February 2024 (10:09:53 CET)
ARTICLE
|
doi:10.20944/preprints202401.2140.v1
Subject:
Environmental And Earth Sciences,
Soil Science
Keywords:
causal machine learning; soil analysis; causal discovery; crop fertilization; flood; agriculture; deposition; climate change
Online: 31 January 2024 (02:55:42 CET)
REVIEW
|
doi:10.20944/preprints202401.1443.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
The Blood-Brain Barrier (BBB); CNS drug discovery; passive diffusion; active transport; Efflux transporters; Influx Transporters; P-glycoproteins (P-gp); breast cancer resistance protein (BCRP); in silico models
Online: 19 January 2024 (09:32:31 CET)
REVIEW
|
doi:10.20944/preprints202401.1357.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
HIV-1; AIDS; FDA; Combination antiretroviral therapy; latent reservoirs; apoptosis; drug resistance; anti-HIV-1 drug design and discovery
Online: 18 January 2024 (10:29:57 CET)
ARTICLE
|
doi:10.20944/preprints202401.0907.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
cancer; protein degradation; degraders; drug discovery; PROTAC; CDK9
Online: 11 January 2024 (10:20:13 CET)
ARTICLE
|
doi:10.20944/preprints202312.2030.v1
Subject:
Biology And Life Sciences,
Aquatic Science
Keywords:
Myzostomida; symbiotic polychaetes; crinoids; Hainan Island; marine biodiversity; echinoderm symbionts; SCUBA; Sanya; new species discovery
Online: 27 December 2023 (10:08:27 CET)
REVIEW
|
doi:10.20944/preprints202312.1443.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
marine Streptomyces; alkaloid; secondary metabolite; discovery; development
Online: 19 December 2023 (16:05:45 CET)
REVIEW
|
doi:10.20944/preprints202312.1256.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Biobanking; human biospecimens; drug discovery; health research
Online: 18 December 2023 (10:33:49 CET)
REVIEW
|
doi:10.20944/preprints202312.0982.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
HER2; HER2 discovery; HER2 role in cancers; HER 2 low; HER2DX; prognostic; predictive; biomarker; anti-HER therapies; HER2 landmark trials
Online: 13 December 2023 (11:35:40 CET)
REVIEW
|
doi:10.20944/preprints202312.0548.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
brain cancers; gangliosides; mass spectrometry; biomarker discovery; screening; structural analysis
Online: 7 December 2023 (19:55:09 CET)
ARTICLE
|
doi:10.20944/preprints202311.1523.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Biomarker discovery; disease pathogenesis; autoimmunity; antigenic mimicry; machine learning
Online: 23 November 2023 (11:10:59 CET)
ARTICLE
|
doi:10.20944/preprints202311.1460.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Onchocerciasis; drug discovery; anthelmintics; O. gutturosa; motility and MTT inhibition; FDA approved drugs
Online: 23 November 2023 (09:31:11 CET)
REVIEW
|
doi:10.20944/preprints202311.1221.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
oxidative stress; atrial fibrillation; mitochondrial dysfunction; inflammation; antioxidant drug discovery
Online: 20 November 2023 (05:08:48 CET)
REVIEW
|
doi:10.20944/preprints202311.1051.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Toxoplasma gondii; proteomics; host-parasite interactions; PTMs; drug discovery
Online: 16 November 2023 (07:46:09 CET)
REVIEW
|
doi:10.20944/preprints202311.0852.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Computer-Aided Drug Design (CADD); Machine Learning and Artificial Intelligence (AI); Drug discovery; Chemoinformatics; Molecular modeling; Molecular Docking; Target identification
Online: 14 November 2023 (16:54:42 CET)
ARTICLE
|
doi:10.20944/preprints202311.0766.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 13 November 2023 (08:41:42 CET)
REVIEW
|
doi:10.20944/preprints202311.0529.v1
Subject:
Public Health And Healthcare,
Primary Health Care
Keywords:
SARS-CoV-2; Papain-like protease; COVID-19; Molecular modelling; Molecular dynamics simulations; Drug discovery; Antiviral drugs; Inhibitors; Therapeutic agents; therapeutic targets; Irreversible inhibitors; Repurposing drugs
Online: 8 November 2023 (16:11:55 CET)
ARTICLE
|
doi:10.20944/preprints202310.1816.v1
Subject:
Computer Science And Mathematics,
Probability And Statistics
Keywords:
causal discovery; independence tests; functional data analysis; kernel methods
Online: 30 October 2023 (04:50:39 CET)
REVIEW
|
doi:10.20944/preprints202310.1465.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
drug discovery; target identification; target validation; lead identification; bioinformatics
Online: 24 October 2023 (04:09:01 CEST)
REVIEW
|
doi:10.20944/preprints202208.0213.v2
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
GIBAC; Biophysics; Structural Biology; Drug discovery \& design; Artificial intelligence-integrated drug discovery
Online: 19 October 2023 (13:38:05 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202310.1222.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Supercomputers; Pandemic; Drug Discovery; Public Health Preparedness
Online: 19 October 2023 (05:19:13 CEST)
REVIEW
|
doi:10.20944/preprints202310.0771.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 12 October 2023 (04:19:37 CEST)
ARTICLE
|
doi:10.20944/preprints202310.0425.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
hepatitis B; antiviral; drug discovery; HBc protein; pharmacophore-based screening; drug repurposing
Online: 8 October 2023 (05:11:37 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1350.v1
Subject:
Computer Science And Mathematics,
Computer Networks And Communications
Keywords:
echo chamber; filter bubble; digital social networks; social network analysis; polarization; diversity; community discovery
Online: 20 September 2023 (04:51:16 CEST)
REVIEW
|
doi:10.20944/preprints202309.0943.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
arbovirus; monoclonal antibody; flavivirus; alphavirus; neutralizing antibody; antibody discovery
Online: 14 September 2023 (03:51:07 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0699.v1
Subject:
Computer Science And Mathematics,
Computer Networks And Communications
Keywords:
wireless sensor networks; energy harvesting; neighbor discovery; data fusion
Online: 12 September 2023 (04:10:25 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2113.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
herbs; spices; flavonoids; antioxidants; diabetes; volatile compounds; drug discovery; phytochemicals; human health
Online: 31 August 2023 (10:12:18 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2118.v1
Subject:
Engineering,
Other
Keywords:
Behaviour analysis; domestic environments; activities of daily living; knowledge discovery in databases
Online: 31 August 2023 (09:30:42 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1966.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Drug discovery; computational chemistry; conceptual DFT; marine cyclopeptides; chemical reactivity properties; bioavailability scores
Online: 29 August 2023 (09:36:49 CEST)
REVIEW
|
doi:10.20944/preprints202308.1518.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
SARS-CoV-2; main protease; inhibitors; molecular modeling; molecular dynamics simulations; binding energy calculation; ADME properties; potential therapeutics; drug discovery
Online: 22 August 2023 (07:19:37 CEST)
REVIEW
|
doi:10.20944/preprints202308.0887.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Drug Discovery; Drug Repurposing; SARS-CoV-2; COVID; Molecular Docking; QSAR; Molecular Dynamic; Virtual Screening; Drug Design
Online: 11 August 2023 (09:03:55 CEST)
REVIEW
|
doi:10.20944/preprints202308.0434.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
In silico studies; drug discovery; SARS-CoV-2; molecular docking; virtual screening; molecular dynamics simulations; drug candidates; antiviral activity; receptor-ligand complex; drug design
Online: 4 August 2023 (11:11:21 CEST)
ARTICLE
|
doi:10.20944/preprints202307.2034.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bcl-2; Anti-apoptotic protein; Indole; Cancer drug discovery
Online: 28 July 2023 (14:36:37 CEST)
REVIEW
|
doi:10.20944/preprints202307.0757.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Lippia javanica; Pharmacological; metabolites; ethnobotanical; drug discovery
Online: 12 July 2023 (05:42:56 CEST)
ARTICLE
|
doi:10.20944/preprints202306.2033.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Process Mining; Process Model Discovery; Mining action+state evolution
Online: 28 June 2023 (16:19:00 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1818.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Alternative Splicing; two-colour (GFP/RFP) Fluorescent Reporter; MAPT; Exon-Skipping; FTDP-17; High Content Screening; siRNA; Nucleic Acids Therapeutics; Drug discovery
Online: 26 June 2023 (13:55:26 CEST)
REVIEW
|
doi:10.20944/preprints202306.0609.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Kinases; human diseases; macrocyclic inhibitors; drug discovery
Online: 8 June 2023 (08:54:08 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0109.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
triple negative breast cancer; MCAK/KIF2C; aneuploidy; chromosomal instability; drug discovery
Online: 1 June 2023 (15:47:29 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1006.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Melanoma; drug discovery; spliceosomal inhibition; BRAF; cell line xenograft; organ histopathology
Online: 15 May 2023 (09:19:54 CEST)
REVIEW
|
doi:10.20944/preprints202305.0945.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Systems Pharmacology; Polypharmacology; Adverse Events; Drug Discovery; Functional genomics; Disease Modeling; Network analysis; Innovation
Online: 12 May 2023 (12:18:59 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0908.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Deep Learning; Topic Discovery; Latent Dirichlet Allocation; Latent Semantic Analysis; Probabilistic Latent Semantic Analysis
Online: 12 May 2023 (08:52:57 CEST)
Subject:
Environmental And Earth Sciences,
Paleontology
Keywords:
Pyrenees; paleoecology; hypothesis testing; discovery; serendipity; Quaternary; Lateglacial; Holocene; last millennia
Online: 10 May 2023 (08:24:15 CEST)
REVIEW
|
doi:10.20944/preprints202305.0473.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Drug Discovery; Drug Design; Drug Development, Quantum Computing, Quantum Machine Learning
Online: 8 May 2023 (08:37:23 CEST)
REVIEW
|
doi:10.20944/preprints202304.0209.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Gut microbiome; Machine learning; Deep learning; Metagenomics; Autoimmune diseases; Biomarkers discovery; Diagnostic models
Online: 23 April 2023 (02:59:58 CEST)
REVIEW
|
doi:10.20944/preprints202304.0677.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Metabolomics; Simultaneous Quantitation and Discovery (SQUAD); Targeted Metabolomics; Untargeted Metabolomics
Online: 21 April 2023 (07:29:13 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0322.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Hemolytic peptide; Network science; Half-Space Proximal Networks; Metadata Networks; Visual mining; Cluster analysis; Motif discovery; StarPep toolbox; Peptide drug discovery
Online: 17 March 2023 (10:05:05 CET)
ARTICLE
|
doi:10.20944/preprints202303.0253.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
ASFV; humoral responses; ASFV capsid proteins; ASFV vaccines; ASFV immunity; antigen discovery; luciferase antibody capture assay; luciferase immunoprecipitation assay; viral hemorrhagic fever.
Online: 14 March 2023 (09:43:57 CET)
ARTICLE
|
doi:10.20944/preprints202303.0193.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Antibiofilm peptide; chemical space; StarPep toolbox; complex network; centrality measure; motif discovery
Online: 10 March 2023 (09:36:30 CET)
ARTICLE
|
doi:10.20944/preprints202303.0048.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Minimum Inhibitory Concentrations; Deep Learning; Regression; Antimicrobial peptides; Drug Discovery
Online: 3 March 2023 (01:29:51 CET)
ARTICLE
|
doi:10.20944/preprints202302.0250.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
AI drug discovery; mTOR; rapalog; C. elegans; cancer; longevity
Online: 15 February 2023 (02:42:57 CET)
REVIEW
|
doi:10.20944/preprints202302.0234.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
lipid metabolism; Apicomplexa; drug discovery; calcium signaling; acidocalcisomes; parasite
Online: 14 February 2023 (04:42:12 CET)
ARTICLE
|
doi:10.20944/preprints202301.0221.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Ion channels; Membrane proteins; Transmembrane proteins; Drug discovery; Protein language models; Convolutional Neural Network
Online: 12 January 2023 (09:21:08 CET)
ARTICLE
|
doi:10.20944/preprints202301.0039.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
somatic point mutations; non-coding RNA; biomarker discovery; driver genes; non-coding RNAs prioritization; health data analytics
Online: 4 January 2023 (02:22:00 CET)
ARTICLE
|
doi:10.20944/preprints202211.0296.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antimicrobial resistance; broad-spectrum antibiotics; antibacterial drug discovery; gram-negative bacteria; pyrrolobenzodiazepines
Online: 16 November 2022 (04:20:55 CET)
BRIEF REPORT
|
doi:10.20944/preprints202211.0063.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
melanoma; drug discovery; spliceosomal inhibition; acute toxicity; blood chemistry; organ histopathology
Online: 3 November 2022 (01:43:05 CET)
REVIEW
|
doi:10.20944/preprints202208.0230.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; compound databases; chemical space; diversity; drug discovery; openscience; pseudo-natural product
Online: 12 August 2022 (08:39:40 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0349.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Docking; lead discovery; molecular dynamic simulation; tuberculosis; coupled assay
Online: 25 May 2022 (10:11:26 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0146.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
ubiquitous exposure; diagnosis; research design; quality of health care; habitat injuries; discovery
Online: 11 May 2022 (05:40:27 CEST)
ARTICLE
|
doi:10.20944/preprints202204.0224.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID-19; SARS-CoV-2; drug discovery; multitargeting; computational drug repurposing
Online: 26 April 2022 (03:39:06 CEST)
REVIEW
|
doi:10.20944/preprints202204.0151.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Isocyanide-based multicomponent reactions; Antimicrobial Discovery; Antibiotic Resistance; Public Health
Online: 18 April 2022 (03:38:08 CEST)
ARTICLE
|
doi:10.20944/preprints202202.0349.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Hypoxia-inducible factor; cancer; hypoxia; drug discovery; medicinal chemistry; virtual screening; molecular dynamics simulation; MM-PBSA; Drug discovery
Online: 28 February 2022 (08:40:24 CET)
REVIEW
|
doi:10.20944/preprints202202.0067.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Antimalarial Drug; Malaria Vaccine; Drug Discovery; Artimisnine; K13; Malaria
Online: 4 February 2022 (10:22:34 CET)
ARTICLE
|
doi:10.20944/preprints202202.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cancer; tumor homing peptide; in silico drug discovery; complex network; chemical space network; centrality measure; similarity searching, group fusion; motif discovery; starPep toolbox software
Online: 3 February 2022 (10:14:05 CET)
REVIEW
|
doi:10.20944/preprints202201.0440.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
electrophiles; signaling; profiling; drug mechanism; drug discovery; T-REX
Online: 28 January 2022 (14:57:08 CET)
ARTICLE
|
doi:10.20944/preprints202111.0467.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
myxobacteria; secondary metabolites; biarylitide; natural product discovery; RiPPs; genome mining; myxarylin
Online: 25 November 2021 (10:42:39 CET)
ARTICLE
|
doi:10.20944/preprints202111.0329.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Machine Learning; Deep Learning; Molecular Modeling; Virtual Screening; Drug Discovery
Online: 18 November 2021 (13:59:09 CET)
ARTICLE
|
doi:10.20944/preprints202111.0266.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Pan-Cancer; somatic point mutations; cancer subtyping; biomarker discovery; driver genes; per-sonalized medicine; health data analytics
Online: 15 November 2021 (13:51:33 CET)
ARTICLE
|
doi:10.20944/preprints202111.0125.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
artificial intelligence; de novo design; fragment-based drug discovery; HIV-1 inhibitors; pseudo natural products
Online: 8 November 2021 (09:23:49 CET)
REVIEW
|
doi:10.20944/preprints202109.0501.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Antigen Selection; Epitope Selection; Antibody Targeting; Epitope Accessibility; Antibody Engineering; Protein Engineering; Drug Targeting; Model-Informed Drug Discovery and Development
Online: 3 November 2021 (08:26:47 CET)
REVIEW
|
doi:10.20944/preprints202109.0491.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Tuberculosis; Mycobacterium; Diagnostics; Drug Discovery; Antibiotics; Antimicrobial Re-sistance; Microfluidics; Single-Cell Analysis; Bioengineered Models
Online: 29 September 2021 (11:34:04 CEST)
ARTICLE
|
doi:10.20944/preprints202109.0138.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Agaricus Bisporus; Button Mushroom; Molecular docking; PyRx software; BIOVIA Discovery studio
Online: 8 September 2021 (10:14:03 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0512.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
oyster mushroom (Pleurotus sp.); PARP protein; 4UND protein; molecular docking; PyRx; BIOVIA drug discovery
Online: 26 August 2021 (16:15:06 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0770.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
BRF2; cancer; molecular dynamics simulation; drug repurposing; drug discovery
Online: 16 July 2021 (11:40:34 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0315.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Myxobacteria; myxochelin; nicotinic acid; secondary metabolites; natural product discovery; precursor-directed biosynthesis; total synthesis
Online: 14 July 2021 (10:03:32 CEST)
REVIEW
|
doi:10.20944/preprints202106.0305.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
dietary flavonoids; cardioprotective effects; ROS scavenging; myocardial dysfunction; bioavailability and drug metabolism; toxicity; drug discovery
Online: 11 June 2021 (08:44:01 CEST)
REVIEW
|
doi:10.20944/preprints202105.0567.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Artificial intelligence AI; machine learning; algorithms; QSAR; drug discovery
Online: 24 May 2021 (13:02:21 CEST)
REVIEW
|
doi:10.20944/preprints202105.0346.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
drug discovery; drug repurposing; bioinformatics; machine learning; artificial intelligence; biomedical discoveries etc.
Online: 14 May 2021 (15:17:50 CEST)
REVIEW
|
doi:10.20944/preprints202104.0244.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Staphylococcus aureus; MRSA; genome-scale metabolic models; model-driven discovery; strain-specific models
Online: 8 April 2021 (14:25:31 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0084.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
price discovery; financial economics; clearing; credit default swaps; collateralization; OTC; risk premium; CCP.
Online: 2 March 2021 (12:05:53 CET)
ARTICLE
|
doi:10.20944/preprints202103.0059.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Metallothionein (MT); Scientific discovery; Scientific pursuit; Research strategies; upward looking research; Exploratory research; Protein function; Compensation; Moonlighting; multifunctional proteins; Vestiges
Online: 2 March 2021 (09:39:39 CET)
REVIEW
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
web server; rational design; functionalizing enzymes; enzyme discovery; user-friendly tools
Online: 28 January 2021 (07:51:45 CET)
ARTICLE
|
doi:10.20944/preprints202101.0209.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
leafy greens; spinach; metabolomics; metabolic profiling; food pathogens; biomarker discovery
Online: 12 January 2021 (08:20:35 CET)
REVIEW
|
doi:10.20944/preprints202012.0372.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Vicia faba; genomic resources; mapping population; gene discovery; breeding
Online: 15 December 2020 (10:38:24 CET)
ARTICLE
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
COVID-19; SARS-CoV-2; in silico drug discovery; gene expression profile; tensor decomposition; feature extraction
Online: 8 December 2020 (10:17:05 CET)
ARTICLE
|
doi:10.20944/preprints202010.0196.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
drug discovery; artificial intelligence; protein discovery; binding prediction; synthetic molecule generation; synthetic drug
Online: 20 November 2020 (11:30:03 CET)
CONCEPT PAPER
|
doi:10.20944/preprints202011.0250.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
antibiotic discovery; STEM education; biosynthetic gene cluster; molecular networking; multi-omics
Online: 6 November 2020 (16:50:46 CET)
REVIEW
|
doi:10.20944/preprints202010.0179.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Non Michaelis-Menten Kinetics; High-throughput screening; allostery; cooperativity; processive kinetics; distributive kinetics; single-molecule; auto-catalytic; drug discovery
Online: 8 October 2020 (13:34:16 CEST)
ARTICLE
|
doi:10.20944/preprints202006.0258.v2
Subject:
Engineering,
Civil Engineering
Keywords:
Conservation laws; Data inference; Data discovery; Dimensionless form; PINN
Online: 30 September 2020 (03:51:25 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0602.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; Genomes; microRNA; SARS-CoV-2; Variant discovery
Online: 25 September 2020 (10:14:46 CEST)
REVIEW
|
doi:10.20944/preprints202008.0320.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Data Science; Machine Learning; Deep Learning; Genomics; COVID-19; Drug Discovery; Image Analysis; Interactomics; Epidemiology
Online: 14 August 2020 (11:01:56 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0213.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Clustering; Pattern Discovery; Time series; Multi-Level Spectral Clustering; English Channel
Online: 8 August 2020 (18:00:26 CEST)
REVIEW
|
doi:10.20944/preprints202007.0523.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
discovery proteomics; targeted proteomics; mass spectrometry; fish allergens; crustacean allergens; mollusk allergens
Online: 22 July 2020 (11:23:40 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0172.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
COVID-19; Twitter; Topic Discovery; Arabic
Online: 9 July 2020 (07:25:19 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0326.v2
Subject:
Environmental And Earth Sciences,
Remote Sensing
Keywords:
GEO label; serverless; semantic sensor web; discovery; visualisation; sensor web
Online: 30 June 2020 (08:06:39 CEST)