Search Results
30656 articles found
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
lung adenocarcinoma; macrophage; PD-L1; GM-CSF; STAT3
Online: 11 June 2021 (13:08:03 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0502.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
mushroom; immune checkpoints; Axl receptor; lung cancer; dendritic cells; immune response.
Online: 21 July 2021 (15:43:11 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0097.v1
Subject:
Chemistry And Materials Science,
Other
Keywords:
CO oxidation; Methanol oxidation; Spray impregnation; Core-shell; Cobalt oxide; Palladium
Online: 1 December 2023 (16:32:29 CET)
ARTICLE
|
doi:10.20944/preprints201809.0458.v2
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Suzuki coupling reaction; Layered double hydroxides; Solid base catalyst; Microwave irradiation
Online: 8 January 2019 (15:13:46 CET)
ARTICLE
|
doi:10.20944/preprints202208.0103.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Resveratrol; antioxidant metabolism; scavengome; biomimetic oxidation; bioactivity-guided isolation; NMR spectroscopy; xanthine oxidase
Online: 4 August 2022 (05:33:52 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1208.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
colorectal neoplasms; microsatellite instability; immune checkpoint proteins; immunotherapy
Online: 21 February 2024 (15:00:37 CET)
REVIEW
|
doi:10.20944/preprints202108.0112.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Epitranscriptomics, Immune checkpoint blockage (ICB) therapy, anti-PD-1/PD-L1 drug resistance, Personalized medicine, CISH, microRNAs
Online: 4 August 2021 (13:02:22 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0050.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
OSRM; nickel; bimetallic catalyst; heterogeneous catalysis; Pd-Ni
Online: 2 August 2018 (16:54:10 CEST)
ARTICLE
|
doi:10.20944/preprints202401.1075.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
indoor fingerprint localization; WKNN; fingerprint distances
Online: 15 January 2024 (06:13:23 CET)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints202308.1413.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
diabetes; cardiovascular; renal; SGLT1; SGLT2; therapy.
Online: 22 August 2023 (07:45:50 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0383.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; medicinal chemistry; probe development
Online: 15 December 2020 (12:56:31 CET)
ARTICLE
|
doi:10.20944/preprints202012.0354.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; uHTS
Online: 14 December 2020 (16:36:57 CET)
HYPOTHESIS
|
doi:10.20944/preprints202004.0151.v2
Online: 22 April 2020 (09:46:54 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0116.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
In vivo; Alpha-glucosidase; Alpha-amylase; hyperglycemia
Online: 16 March 2017 (09:35:36 CET)
ARTICLE
|
doi:10.20944/preprints201810.0274.v1
Subject:
Social Sciences,
Language And Linguistics
Keywords:
Bilingual program; Academic performance; Learning competence; English proficiency; Student workload
Online: 12 October 2018 (14:51:07 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0609.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immune checkpoint inhibitors; immune-related adverse events (irAEs); tolerance; ipilimumab; nivolumab; interleukin-2; hyperthermia; low-dose-combination therapy
Online: 28 November 2018 (10:23:31 CET)
ARTICLE
|
doi:10.20944/preprints202301.0421.v3
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncology; Immune Checkpoint Inhibition; PD-1; PD-L1; CTLA-4; Immune Related Adverse Events; Immunotherapy; Tumor Plasticity; Tumor Microenvironment; Optimum Therapy Duration
Online: 6 March 2023 (01:53:16 CET)
REVIEW
|
doi:10.20944/preprints202311.0295.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Atrial fibrillation, SGLT2 inhibitors, cardiovascular outcomes, hemodynamic effects, AF risk reduction
Online: 6 November 2023 (08:13:49 CET)
ARTICLE
|
doi:10.20944/preprints201909.0250.v1
Subject:
Chemistry And Materials Science,
Chemical Engineering
Keywords:
ch4 temperature-programmed reduction; methane combustion; pd/zro2 catalyst; reduction; calcination
Online: 21 September 2019 (09:36:45 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0785.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
enteroviruses, coxsackievirus, leucoverdazyls, antioxidant, antiviral, 2C protein
Online: 11 April 2024 (09:22:02 CEST)
REVIEW
|
doi:10.20944/preprints202401.1697.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
DOAC; FXIa; mAbs; ASO; drug-drug interactions
Online: 23 January 2024 (12:31:04 CET)
ARTICLE
|
doi:10.20944/preprints202302.0423.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell; autoimmune disease; drug repurposing
Online: 24 February 2023 (09:11:37 CET)
ARTICLE
|
doi:10.20944/preprints202101.0480.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
organoid; induced pluripotent stem cell; Parkinson’s disease; neurotransmission; neuroimmunity; neuroinflammation; viral infection
Online: 25 January 2021 (10:55:03 CET)
REVIEW
|
doi:10.20944/preprints202402.1535.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
DNA polymerase I; Polymerase θ ; reverse transcriptase; homologous recombination; antibiotics; apicoplast
Online: 27 February 2024 (12:29:29 CET)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1978.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
enfortumab vedotin; urothelial carcinoma; database; real‐world; immune checkpoint
Online: 28 July 2023 (11:46:48 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0519.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Auger Electron Therapy; Palladium-103; Partial Pressure; Radioisotope Separation; Diffusion.
Online: 8 January 2024 (06:33:48 CET)
ARTICLE
|
doi:10.20944/preprints202001.0122.v1
Subject:
Physical Sciences,
Biophysics
Keywords:
cervical adenocarcinoma; immune-checkpoint inhibitor; programmed cell death-1(PD-1); programmed cell death-ligand 1(PD-L1); CD8 expression; lymphocyte; survival analysis
Online: 12 January 2020 (15:01:23 CET)
ARTICLE
|
doi:10.20944/preprints202311.0688.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
melanoma; metastasis; overall survival; progression-free survival; side effects; Nivolumab; Ipilimumab; anti-programmed death-1 antibodies; anti-cytotoxic T-lymphocyte antigen-4 antibodies.
Online: 10 November 2023 (11:05:56 CET)
ARTICLE
|
doi:10.20944/preprints202402.1288.v2
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
SGLT2 Inhibitors; Empagliflozin; Renal fibrosis; Connective tissue growth factor; Epithelial-mesenchymal transition
Online: 23 February 2024 (13:25:01 CET)
ARTICLE
|
doi:10.20944/preprints202311.0437.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
6-methyl-2-thiouracil, 6-propyl-2-thiouracil; complexation, copper(II) complexes, palladium(II) complexes, antimicrobial activity
Online: 7 November 2023 (10:37:37 CET)
ARTICLE
|
doi:10.20944/preprints201704.0014.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
tin oxide pellets; doping; HRTEM analysis; CO; sensitivity
Online: 4 April 2017 (08:16:13 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0240.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID19; 2019-nCov, 3CLpro inhbitors
Online: 15 April 2020 (10:00:52 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
REVIEW
|
doi:10.20944/preprints201805.0145.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase, enzyme inhibition, metalloenzymes, amino acid, glaucoma, tumors
Online: 9 May 2018 (13:55:15 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0483.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
MRONJ; CDK4/6 inhibitors; metastatic breast cancer; oral epidemiology
Online: 8 November 2023 (08:42:55 CET)
ARTICLE
|
doi:10.20944/preprints202307.2034.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bcl-2; Anti-apoptotic protein; Indole; Cancer drug discovery
Online: 28 July 2023 (14:36:37 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0270.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
drug design; falcipain; malaria; peptidomimetics; Plasmodium falciparum; virtual screening; pharmacophore.
Online: 12 July 2021 (14:48:13 CEST)
REVIEW
|
doi:10.20944/preprints202106.0158.v1
Online: 7 June 2021 (09:29:06 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
ARTICLE
|
doi:10.20944/preprints202401.1843.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
standardized Brassica juncea; 3T3-L1; C57BL/6J; anti-obesity; mechanism
Online: 25 January 2024 (14:24:23 CET)
ARTICLE
|
doi:10.20944/preprints202307.1251.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ascorbic acid; pharmacologic ascorbate; pancreatic cancer; epigenetics; DNA methyltransferase (DNMT); ten-eleven translocation (TET) methylcytosine dioxygenase
Online: 18 July 2023 (13:51:14 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0286.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
pd doped graphyne; dissolved gases; adsorption; density functional theory (dft)
Online: 25 September 2019 (16:01:58 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0097.v1
Subject:
Chemistry And Materials Science,
Electrochemistry
Keywords:
WO3; electrocatalysts; alkaline; Pd-W alloy; oxygen reduction reaction; reduction-oxidation method
Online: 9 April 2018 (04:06:25 CEST)
ARTICLE
|
doi:10.20944/preprints201912.0368.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
V(D)J recombination; vAbl cells; B lymphocytes; mouse genetics; genetic interaction
Online: 29 December 2019 (04:36:17 CET)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Virology,
Biology And Life Sciences
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0468.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
dasatinib; imatinib; nilotibin; ponatinib; children; therapeutic drug monitoring; sex and gender pharmacology; personalized medicine.
Online: 7 August 2023 (11:53:12 CEST)
REVIEW
|
doi:10.20944/preprints202305.1151.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
fusion proteins; inhibitor; therapeutic; cancer
Online: 16 May 2023 (10:32:09 CEST)
REVIEW
|
doi:10.20944/preprints202211.0448.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
alpha-1-antitrypsin (AAT); neutrophil elastase (NE); NETosis, PAD4, ARDS, COPD; neutrophils; COVID-19; TMPRSS2.
Online: 24 November 2022 (02:50:25 CET)
ARTICLE
|
doi:10.20944/preprints201911.0375.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
synthesis; 2-mercaptabezimidazole; sulfonamide; molecular docking study; α-amylase; sa
Online: 29 November 2019 (10:28:22 CET)
ARTICLE
|
doi:10.20944/preprints201801.0196.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
comorbid diseases; erectile dysfunction; penile duplex doppler ultrasound; penile pathology; phosphodiesterase type 5 inhibitors
Online: 22 January 2018 (09:03:17 CET)
ARTICLE
|
doi:10.20944/preprints202403.1095.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
KRAS inhibitor; metastasis; colorectal cancer; machine learning; meta analysis
Online: 21 March 2024 (03:50:20 CET)
ARTICLE
|
doi:10.20944/preprints202308.0290.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RNA-binding protein; human antigen R (HuR); high-throughput virtual screening; small molecule inhibitors; RNA pulldown assay
Online: 3 August 2023 (10:11:15 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0433.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
PCNA; p15; FRET; inhibitor screening; ATLD2; disease; variant; stability; aggregation
Online: 6 July 2023 (11:53:02 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0109.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
triple negative breast cancer; MCAK/KIF2C; aneuploidy; chromosomal instability; drug discovery
Online: 1 June 2023 (15:47:29 CEST)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
REVIEW
|
doi:10.20944/preprints201806.0056.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
mTOR; mTORC1; mTORC2; rapamycin; rapalogues; rapalogs; mTOR inhibitors; senescence; ageing; aging; cancer; neurodegeneration; immunosenescence; senolytics; biomarkers
Online: 5 June 2018 (09:49:19 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0561.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Nivolumab; immunotherapy; head and neck cancers; HNSCC; chemotherapy; neutrophil to lymphocyt ratio; NLR; second primary malignancy; Cetuximab
Online: 9 May 2023 (04:21:38 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1626.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Proton pump inhibitors; Clopidogrel; Stroke; Myocardial infarction
Online: 25 July 2023 (07:26:31 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0765.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
4-amino-7-chloroquinoline; 1,3,4-oxadiazole; anthranilic acid; synthesis; quorum sensing; anti-biofilm; P. aeruginosa; PQS
Online: 12 July 2023 (21:25:14 CEST)
REVIEW
|
doi:10.20944/preprints202306.0614.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
frailty, comorbidities, Crohn's disease, ulcerative colitis, infections, malignancies
Online: 8 June 2023 (09:30:13 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0097.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
KV1.3; potassium ion channels; antiproliferative activity; apoptosis; anticancer drugs
Online: 9 May 2022 (03:35:09 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0598.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
physical unclonable function; bloom filter; hardware security; PUF; memristor
Online: 27 August 2020 (08:05:03 CEST)
REVIEW
|
doi:10.20944/preprints202307.0136.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
Checkpoint Inhibitor; Philadelphia Chromosome; Myeloproliferative Neoplasm
Online: 4 July 2023 (04:49:05 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1702.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
vascular prosthesis; AEBSF; puromycin; Staphylococcus aureus; FTIR analysis
Online: 22 December 2023 (08:03:49 CET)
REVIEW
|
doi:10.20944/preprints202306.1426.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Trypanosomatids; squalene synthase; farnesyl diphosphate synthase; target-based approach; neglected tropical diseases.
Online: 20 June 2023 (10:27:48 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0218.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Scutellaria baicalensis; phytochemicals; glioblastoma multiforme; in silico
Online: 15 September 2022 (03:55:58 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0243.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
aqueous micellar system; trypsin inhibitor; isoflavone extraction; non-ionic surfactant; multifactorial optimization
Online: 17 January 2022 (16:01:53 CET)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
ARTICLE
|
doi:10.20944/preprints201909.0130.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Synthesis; triazinoindole; thiosemicarbazide; alpha-glucosidase; molecular docking study; SAR
Online: 13 September 2019 (10:54:30 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0200.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Thiazolidinones; ORAC assay; Metalloproteinase-9; Docking study; Keratinocytes cultures; Nuclear factor -kB.
Online: 31 October 2017 (16:36:16 CET)
ARTICLE
|
doi:10.20944/preprints201709.0070.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Coumarin; Mycobacterium tuberculosis; Cholinesterase inhibitor; Monoamine oxidase B inhibitor; Structure activity relationship; Albumin binding, Neuroprotection
Online: 15 September 2017 (17:34:38 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0485.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
bandgap; doping; palladium; platinum; stoichiometric NiO
Online: 22 October 2018 (10:02:55 CEST)
REVIEW
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hyperoxaluria; oxalate; inhibitor; small molecule drug; glycolate oxidase; lactate dehydrogenase; liver selective distribution
Online: 31 December 2020 (08:59:47 CET)
COMMUNICATION
|
doi:10.20944/preprints202004.0146.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Coronavirus Disease 2019; SARS-CoV-2; main protease; molecular docking-based virtual screening
Online: 9 April 2020 (09:34:45 CEST)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)
ARTICLE
|
doi:10.20944/preprints202310.0471.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
monomethyltyrosine; dimethyltyrosine; catalysis; peptides
Online: 9 October 2023 (10:53:37 CEST)
CASE REPORT
|
doi:10.20944/preprints202005.0220.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
checkpoint inhibitors; tuberculosis; non-small cell lung cancer (NSCLC); Anti-PD-1; toxicity management; immunotherapy; pembrolizumab
Online: 13 May 2020 (04:38:50 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0131.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
pharmacogenomics; immune checkpoint blockade; immunotherapy; drug response prediction; algorithm; mathematical model; precision medicine; personalized medicine
Online: 11 August 2019 (14:51:14 CEST)
COMMUNICATION
|
doi:10.20944/preprints202404.1027.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
galectin-1; small molecule glycomimetics; surface plasmon resonance; fluorescence polarisation
Online: 16 April 2024 (10:01:02 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1802.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
diabetes; terpenes; docking; MD simulation; MM-GBSA; DFT
Online: 27 October 2023 (11:50:06 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0006.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
branched chain 2-oxo acids; 2-oxoglutarate dehydrogenase; pyruvate dehydrogenase; phospho-nate and phosphinate analogs of pyruvate; protein succinylation; protein acetylation; protein glutarylation; sirtuin 3; sirtuin 5; anxiety
Online: 3 October 2022 (12:11:50 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0359.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
JAK/STAT3 signaling pathway; Meridianin derivatives; Isothiouronium; Anti-tumor activity
Online: 24 January 2022 (14:06:38 CET)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
REVIEW
|
doi:10.20944/preprints202004.0331.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; associated comorbidities; treatment; ACE2 inhibitors; Type 2 diabetes
Online: 19 April 2020 (05:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0308.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SARS-CoV-2; COVID-19; 3CL protease; molecular docking; molecular dynamics and simulations
Online: 23 February 2020 (02:17:46 CET)
ARTICLE
|
doi:10.20944/preprints202002.0062.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Integrase; HIV-1; Naturally occurring polymorphism; diversity; Molecular Modelling; Molecular Docking
Online: 5 February 2020 (11:02:15 CET)
REVIEW
|
doi:10.20944/preprints201910.0255.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antimicrobial resistance; biofilm; efflux pump inhibitors; antibiotic potentiation; eskapee pathogens; gram-negative bacteria
Online: 22 October 2019 (10:22:56 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0238.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
aurora kinase A; molecular docking; DFT; MD simulation
Online: 23 August 2019 (05:01:40 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ALK5 inhibitor; TGF-β; kinase assay; selectivity; docking
Online: 30 August 2018 (05:52:08 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0215.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
FGFR1; inhibitor; kinase inhibitor; pyrazine; hinge binder
Online: 30 March 2017 (04:13:45 CEST)
ARTICLE
|
doi:10.20944/preprints202404.2012.v1
Subject:
Energy And Fuel Technology,
Engineering
Keywords:
Biogas dry reforming; Membrane reactor; Ni/Cr/Ru catalyst; Ni/Cr catalyst; Operation condition
Online: 30 April 2024 (14:35:43 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0199.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
ammonia fuel cells; ammonia; SOFC; Impregnation; solid oxide
Online: 5 March 2021 (21:30:34 CET)
ARTICLE
|
doi:10.20944/preprints202104.0110.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hydrodechlorination; CHClF2; Pd-Pt/C; thermally modified carbon; effect of catalyst oxidation; pore structure changes
Online: 5 April 2021 (12:12:38 CEST)