ARTICLE
|
doi:10.20944/preprints202005.0057.v2
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; treatment; drug; survival; antiviral; hydroxychloroquine
Online: 9 May 2020 (04:45:37 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0544.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
Bodybuilding; Drug Free; Competing; Peaking; Carbohydrate Loading; Water Loading; Sodium Loading; Fat Loading: Vitamin C; Fibre Restriction
Online: 27 September 2018 (12:58:34 CEST)
REVIEW
|
doi:10.20944/preprints202012.0452.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RNA; self-amplifying RNA; replicon; vaccine; drug delivery
Online: 18 December 2020 (11:12:44 CET)
ARTICLE
|
doi:10.20944/preprints202003.0349.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
novel coronavirus; COVID-19; protease; molecular docking; drug designing; ADME; drug repurposing
Online: 23 March 2020 (09:47:49 CET)
REVIEW
|
doi:10.20944/preprints202012.0242.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; SARS-CoV-2; long-haul; inflammation; tissue damage; drug repurposing
Online: 10 December 2020 (09:42:20 CET)
COMMUNICATION
|
doi:10.20944/preprints202002.0418.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
virtual screening; molecular docking; drug repurposing; drug repositioning; anti-viral drugs; Coronavirus; COVID-19; 2019-nCoV; SARS-CoV-2
Online: 9 March 2020 (02:29:04 CET)
REVIEW
|
doi:10.20944/preprints202012.0062.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Trop 2; targeted therapy; antibody-drug conjugate; solid tumors
Online: 2 December 2020 (12:35:36 CET)
REVIEW
|
doi:10.20944/preprints202010.0179.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Non Michaelis-Menten Kinetics; High-throughput screening; allostery; cooperativity; processive kinetics; distributive kinetics; single-molecule; auto-catalytic; drug discovery
Online: 8 October 2020 (13:34:16 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0360.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SARS-CoV-2; transcriptional inhibition; COVID-19; drug repurposing; TMPRSS2
Online: 28 April 2020 (09:39:02 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0061.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Coronavirus; Deep learning; Drug screening; homology modeling; main protease
Online: 5 February 2020 (10:59:09 CET)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
ARTICLE
|
doi:10.20944/preprints202003.0440.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; SARS-CoV-2; 2019-nCoV; novel corona virus; drug repurposing; chloroquine; high-risk group; asymptomatic
Online: 30 March 2020 (07:24:16 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0071.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
2019-nCoV; novel corona virus; Wuhan virus; drug; vaccine; spike protein; epitope; vaccine design
Online: 5 February 2020 (15:34:15 CET)
ARTICLE
|
doi:10.20944/preprints202003.0413.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
coronavirus; drug; COVID-19; SARS; MERS; ontology; ChEBI; NDF-RT; DrON; bioinformatics
Online: 29 March 2020 (01:58:40 CET)
REVIEW
|
doi:10.20944/preprints201812.0170.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
bacterial nanocellulose; nanofibrillated nanocellulose; animal nanocellulose; algal nanocellulose; tissue engineering; tissue repair; wound dressing; cell delivery; drug delivery; antimicrobial properties
Online: 14 December 2018 (06:44:53 CET)
REVIEW
|
doi:10.20944/preprints202005.0376.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus bioinformatics; SARS-CoV-2; sequencing; epidemiology; drug design; tools
Online: 23 May 2020 (11:01:11 CEST)
REVIEW
|
doi:10.20944/preprints202004.0122.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
melatonin; coronavirus; pandemic; SARS-CoV-2; bat; lung; apoptosis; programmed cell death; mortality; morbidity; COVID-19; drug
Online: 9 April 2020 (09:24:47 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
REVIEW
|
doi:10.20944/preprints202008.0312.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
SARS-CoV-2(COVID-19); + ssRNA; ribosomal – framshift; Pseudoknot; replication; model; drug; vaccine
Online: 14 August 2020 (08:26:31 CEST)
REVIEW
|
doi:10.20944/preprints202105.0311.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Angiotensin converting enzyme 2; breast feeding; drug therapy; pregnancy; severe acute respiratory syndrome coronavirus 2
Online: 13 May 2021 (15:26:34 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0157.v1
Subject:
Business, Economics And Management,
Accounting And Taxation
Keywords:
National Centralized Drug Procurement; "4+7" policy; drug price; interrupted time series; volume-based procurement.
Online: 6 April 2021 (08:18:10 CEST)
REVIEW
|
doi:10.20944/preprints201807.0233.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
nanocrystals; poorly soluble drug; nanotechnology; stability
Online: 13 July 2018 (11:16:15 CEST)
REVIEW
|
doi:10.20944/preprints202112.0315.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Nanotechnology; Niosomes; Targeted Drug Delivery
Online: 20 December 2021 (14:18:53 CET)
ARTICLE
|
doi:10.20944/preprints202107.0229.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
HPLC; NSAIDs; Isocratic; Short column; Drug mixture
Online: 9 July 2021 (15:23:57 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
monoglyceride colloidal liquid crystals; release profile; mathematical models; drug delivery systems; release kinetic; square root laws
Online: 17 September 2018 (09:33:52 CEST)
REVIEW
|
doi:10.20944/preprints202101.0503.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
CNS; Drug receptors; GABA; Cannabinoid; Opioid; Serotonin; Dopamine
Online: 25 January 2021 (14:15:20 CET)
REVIEW
|
doi:10.20944/preprints202102.0265.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Peptides; Clinical Practice; Drug Therapy; Therapeutic
Online: 10 February 2021 (15:51:13 CET)
ARTICLE
|
doi:10.20944/preprints202203.0117.v3
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
active pharmaceutical ingredient; compounded drug; compounding; extemporaneous formulation; manufactured material; medication; monograph; pediatric; reference standards
Online: 5 April 2022 (10:17:10 CEST)
REVIEW
|
doi:10.20944/preprints201805.0426.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
biological activity; crosslinking; drug delivery; cosmetic; food-supplement; functionalization; hyaluronan applications; hyaluronan derivatives; hyaluronan synthases; hyaluronic acid; hyaluronidases; physico-chemical properties
Online: 29 May 2018 (12:13:48 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0393.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV2; RNA depended RNA polymerase; Valproic acid Co-A; drug repurposing
Online: 26 March 2020 (15:04:22 CET)
REVIEW
|
doi:10.20944/preprints202007.0108.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
COVID-19; SARS-CoV-2; coronavirus; hypothesis; pathophysiology; drug repurposing
Online: 7 July 2020 (02:50:55 CEST)
REVIEW
|
doi:10.20944/preprints202105.0346.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
drug discovery; drug repurposing; bioinformatics; machine learning; artificial intelligence; biomedical discoveries etc.
Online: 14 May 2021 (15:17:50 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0075.v3
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
azithromycin; HPLC; robust; isocratic; drug stability; degradation products
Online: 4 January 2017 (10:08:52 CET)
REVIEW
|
doi:10.20944/preprints202104.0652.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Enzymatic reaction; crosslinking; Hydrogel; Biomedical application; Tissue engineering; Wound healing; Drug delivery
Online: 26 April 2021 (10:52:24 CEST)
REVIEW
|
doi:10.20944/preprints202005.0234.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
SIRD; Twitter; GHSI; Pre-symptomatic; EHR; Contact tracing; On-line survey; qRT-PCR; X-ray; CT/HRCT; CNN; Autoencoder; Drug affinity; CPI; and Inflation.
Online: 14 May 2020 (11:25:57 CEST)
REVIEW
|
doi:10.20944/preprints202305.1084.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
antibody-drug conjugate; lysosome; cathepsin; legumain; self-immolation; payload release; peptidomimetic; linker
Online: 16 May 2023 (04:51:34 CEST)
CASE REPORT
|
doi:10.20944/preprints202012.0596.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Covid-19, SARS-CoV-2, drug repurposing
Online: 23 December 2020 (15:58:38 CET)
REVIEW
|
doi:10.20944/preprints202105.0567.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Artificial intelligence AI; machine learning; algorithms; QSAR; drug discovery
Online: 24 May 2021 (13:02:21 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0023.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
gelatin-oleic conjugate; self-assembled biodegradable nanoparticles; biomimetic shear stress; cell dynamic environment; cellular drug delivery; paclitaxel
Online: 4 April 2017 (10:59:02 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0025.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
drug repurposing; translational bioinformatics; transcriptomics; transcriptome analysis; drug discovery; protocol; gene expression
Online: 9 October 2016 (08:42:23 CEST)
REVIEW
|
doi:10.20944/preprints201807.0241.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
biomaterial; bone regeneration; drug release; hydrogel; lignin; multivariate data processing; osteogenesis; scaffolds; stem cells; tissue engineering
Online: 13 July 2018 (15:07:37 CEST)
ARTICLE
|
doi:10.20944/preprints202101.0490.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
CD44; Cancer Stem Cells; Tumorigenesis; Drug Resistance; Immune Markers; Epithelial to Mesenchymal Transition; Therapeutic Targeting
Online: 25 January 2021 (12:23:49 CET)
ARTICLE
|
doi:10.20944/preprints201610.0083.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
stroke; antioxidant; co-drug; animal model
Online: 20 October 2016 (08:46:38 CEST)
ARTICLE
|
doi:10.20944/preprints201705.0174.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
steroid; metabolism; anti-inflammatory drug; inhibition
Online: 24 May 2017 (08:25:26 CEST)
REVIEW
|
doi:10.20944/preprints201702.0036.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
pulmonary arterial hypertension; prostacyclin; nanoparticle; drug delivery system
Online: 13 February 2017 (09:27:09 CET)
REVIEW
|
doi:10.20944/preprints201705.0129.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
cell fate decision; cancer attractors; gene network dynamics; EMT; drug resistance; intrinsically disordered proteins
Online: 17 May 2017 (06:25:17 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0310.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
primary open angle glaucoma; dorzolamide/timolol fixed combination; drug efficacy; safety
Online: 24 April 2018 (08:36:58 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0490.v1
Subject:
Computer Science And Mathematics,
Computer Vision And Graphics
Keywords:
drug release simulation; disintegration simulation; poorly water soluble drug; mefenamic acid; Noyes-Whitney equation; cellular automata; synchrotron microtomography
Online: 22 October 2018 (11:38:04 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0199.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SARS-CoV-2; COVID-19; CADD; virtual screening; approved drugs; drug repurposing; essential targets; molecular docking; molecular dynamics simulations
Online: 11 May 2020 (13:14:18 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0132.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
arylamine N-acetyltransferases; cancer; tuberculosis; drug discovery; traditional Chinese medicine; virtual screening; molecular dynamics simulation; MM-PBSA
Online: 30 June 2017 (11:36:22 CEST)
REVIEW
|
doi:10.20944/preprints202003.0345.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; lysosomotropic agents; endosome; antiviral; drug repurposing
Online: 24 March 2020 (06:26:54 CET)
ARTICLE
|
doi:10.20944/preprints201709.0102.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
drug screening; bone mineralization; osteoclast; zebrafish
Online: 21 September 2017 (06:34:11 CEST)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
REVIEW
|
doi:10.20944/preprints202005.0342.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
seaweed; metabolites; neuroprotection; Alzheimer’s disease; Parkinson’s disease; ischemic stroke; computer-aided drug discovery
Online: 21 May 2020 (09:49:29 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0028.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
lanthanides; fluorapatite; drug loading; nano carrier
Online: 5 April 2017 (11:26:48 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0170.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Spreading parameter; Cellular proliferation; Drug sensitivity; Substrates; Cancer cells
Online: 26 April 2017 (17:38:07 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0297.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
lignin; drug release; paracetamol; disintegration
Online: 24 May 2019 (12:40:01 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
REVIEW
|
doi:10.20944/preprints202006.0232.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Adverse drug reactions; Anti-COVID drugs; Coronavirus; Drug repurposing; Drug toxicity; Pharmacotherapy
Online: 18 June 2020 (12:43:43 CEST)
REVIEW
|
doi:10.20944/preprints201804.0126.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
pharmaceutical market; drugs; drug discovery; solid-phase peptide synthesis
Online: 10 April 2018 (10:14:33 CEST)
REVIEW
|
doi:10.20944/preprints202001.0324.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
natural products; sirtuin; drug discovery; epigenetics; structure–activity relationship
Online: 27 January 2020 (09:21:29 CET)
ARTICLE
|
doi:10.20944/preprints202009.0459.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; coronavirus; drug repositioning; pathway enrichment
Online: 19 September 2020 (11:34:12 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0283.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Adverse drug reaction; COVID-19 treatment
Online: 12 August 2020 (11:12:41 CEST)
REVIEW
|
doi:10.20944/preprints201805.0011.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
computational drug repositioning; drug repositioning; drug repurposing; machine learning; deep learning; crowdsourcing; open innovation; drug discovery
Online: 1 May 2018 (12:27:22 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0447.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
spike protein; SARS-CoV-2; mutation; drug repurposing; digitoxin
Online: 20 August 2020 (08:24:41 CEST)
ARTICLE
|
doi:10.20944/preprints202006.0358.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Enzyme inhibition; Secondary Metabolites; In-silico Analysis; Molecular docking; Drug candidates
Online: 30 June 2020 (08:11:28 CEST)
REVIEW
|
doi:10.20944/preprints202008.0320.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Data Science; Machine Learning; Deep Learning; Genomics; COVID-19; Drug Discovery; Image Analysis; Interactomics; Epidemiology
Online: 14 August 2020 (11:01:56 CEST)
REVIEW
|
doi:10.20944/preprints201807.0143.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
Aromatic hydroxy metabolites; arenolic drug metabolites; metabolic O-dealkylation; metabolic aromatic ring hydroxylation; primary and auxiliary pharmacophores; auxophores; metabolic modification of drug activity
Online: 9 July 2018 (13:28:16 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0319.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
adverse drug reactions; spontaneous reporting; causality; ADR; severity
Online: 18 August 2018 (05:17:05 CEST)
REVIEW
|
doi:10.20944/preprints201807.0226.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
galvanic replacement; photothermal therapy; drug delivery; nanoparticles; cancer treatment
Online: 13 July 2018 (05:11:21 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0466.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
COVID-19; coronavirus; ACE2; bioinformatics analysis; drug prediction
Online: 26 April 2020 (03:14:50 CEST)
REVIEW
|
doi:10.20944/preprints201812.0032.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cannabis; cannabinoids; THC; CBD, drug-drug interactions; pharmacokinetic; cytochrome P450; UDP- glucuronosyltransferases; glucoprotein-P
Online: 3 December 2018 (16:07:43 CET)
REVIEW
|
doi:10.20944/preprints201910.0296.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
nasal delivery; glioblastoma multiforme; drug delivery; nanoparticles; nose-to-brain delivery; pre-clinical studies; clinical evaluation
Online: 27 October 2019 (09:36:27 CET)
REVIEW
|
doi:10.20944/preprints202108.0558.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
chitosan; chitin; biological activit; drug delivery; antioxidant; antimicrobial; biocatalysis; nanoparticles
Online: 31 August 2021 (11:07:28 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0279.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Blood-Brain Barrier, Penetrating Peptides, Machine learning techniques, Drug delivery, Therapeutic peptides
Online: 10 June 2021 (08:13:15 CEST)
REVIEW
|
doi:10.20944/preprints201709.0050.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's-disease; dementia; drug targeting; nanoemulsion; neuroinflammation; oxidative stress; scavenger receptors; sonoporation; transcranial ultrasound
Online: 13 September 2017 (05:44:29 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Covid-19; proteins; normal-modes; protein-drug interactions; chloroquine; ivermectin; remdesivir; sofosbuvir; boceprevir; α-difluoromethylornithine (DMFO)
Online: 11 August 2020 (04:09:43 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
humans; infection control; therapy; coronavirus; immunoglobulins; drug therapy; therapeutic use; corticosteroid
Online: 8 March 2020 (17:04:19 CET)
REVIEW
|
doi:10.20944/preprints201808.0155.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
amyloid diseases; biocomputing; drug design; natural antiamyloids
Online: 8 August 2018 (04:27:10 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0561.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cheminformatics, drugs, drug-likeness, drug discovery, natural products
Online: 23 November 2018 (13:56:32 CET)
REVIEW
|
doi:10.20944/preprints202004.0395.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
coronavirus disease 2019; chloroquine; drug repurposing; HIV; Africa
Online: 22 April 2020 (08:33:34 CEST)
REVIEW
|
doi:10.20944/preprints202203.0071.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
rheumatoid arthritis; precision medicine; new treatment; drug development; method development
Online: 25 May 2022 (04:59:01 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0307.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
TiO2 nanoparticles; antibacterial activity; multi-drug-resistance pathogens; MRSA; E. coli. P. aeruginosa; genotoxicity
Online: 10 November 2020 (12:09:17 CET)
REVIEW
|
doi:10.20944/preprints201810.0507.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
liposomes, exosomes, extracellular vesicles, drug delivery, drug targeting, bioinspired systems, engineered systems.
Online: 22 October 2018 (15:35:20 CEST)
REVIEW
|
doi:10.20944/preprints201810.0577.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
myeloma; daratumumab; elotuzumab; isatuximab; CD38; JNJ- 63723283; denosumab; checkpoint inhibitors; BCMA; bispecific T-cell engager; antibody-drug conjugates
Online: 24 October 2018 (12:11:23 CEST)
REVIEW
|
doi:10.20944/preprints201910.0144.v6
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus; antiviral drug; drug discovery; drug development; broad-spectrum antivirals
Online: 14 February 2020 (02:27:24 CET)
CONCEPT PAPER
|
doi:10.20944/preprints202004.0213.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
covid-19; rlmE MTase; new drug target; corona diagnosis; corona pandemic
Online: 13 April 2020 (12:33:22 CEST)
REVIEW
|
doi:10.20944/preprints201801.0218.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Biocompatibility; Biodegradability; Biopolyesters; Biopolymers; Composites; Drug Release; Implants; Polyhydroxyalkanoates; Scaffolds; Tissue Engineering
Online: 23 January 2018 (16:49:05 CET)
ARTICLE
|
doi:10.20944/preprints202106.0675.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
pharmacogenes; transcripts; sex-bias; drug metabolism; sex differences
Online: 28 June 2021 (15:08:38 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1300.v1
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
semaglutide; drug misuse; drug abuse; pharmacovigilance; image- and performance-enhancing (IPED) drugs; glucagon-like peptide-1 (GLP-1) agonists
Online: 20 September 2023 (05:05:11 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0395.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Deep-Learning; Interpretability; Omics; Biophysics; Drug Synergy; Cancer
Online: 14 April 2021 (17:44:40 CEST)
REVIEW
|
doi:10.20944/preprints202206.0147.v3
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Designed Ankyrin Repeat protein; DARPin; drug development; ensovibep; abicipar pegol
Online: 21 June 2022 (10:21:27 CEST)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0245.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
Chitosan-g-PMMA amphiphilic nanoparticles; thiolated polymers; mucoadhesion; mucosal drug delivery; Caco2 and HT29-MTX cell lines; apparent permeability in vitro.
Online: 18 April 2018 (16:28:21 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0397.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SARS-CoV-2; Drug repurposing; N-acetyl-D-glucosamine; ORF1ab; Biodata mining; Protein modelling
Online: 24 May 2020 (18:49:41 CEST)
REVIEW
|
doi:10.20944/preprints202007.0016.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
myeloma; BCMA; bispecific T-cell engager; antibody-drug conjugates; chimeric antigen receptor T-cells; belantamab mafodotin; idecabtagene vicleucel; JNJ-68284528
Online: 3 July 2020 (07:30:57 CEST)
REVIEW
|
doi:10.20944/preprints202107.0506.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Drug repositioning; Molecular modelling; Beauvericin
Online: 22 July 2021 (07:48:33 CEST)
REVIEW
|
doi:10.20944/preprints201810.0360.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Molecular Dynamics, CoSolvent Molecular Dynamics, Drug design, Fragment Screening, Docking
Online: 16 October 2018 (12:15:17 CEST)
REVIEW
|
doi:10.20944/preprints201908.0271.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
GPCRs; membrane protein; molecular dynamics; protein structure; drug design; biased-signaling pathway; allosteric sites
Online: 26 August 2019 (15:34:57 CEST)
REVIEW
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
nucleoid-associated proteins (NAPs); moonlighting proteins; drug target; biofilm; specificity determination; phylogenetic analysis
Online: 7 June 2020 (09:07:56 CEST)