REVIEW
|
doi:10.20944/preprints202003.0378.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
China's COVID-19 Guide; Remdesivir; Xuebijing; Hydroxychloroquine; IL6 inhibitors; COVID-19
Online: 26 March 2020 (01:48:42 CET)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0003.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
SARS-CoV-2; protease; virtual screening; pharmacophore; inhibitors; natural compounds
Online: 17 April 2020 (11:00:55 CEST)
REVIEW
|
doi:10.20944/preprints202004.0160.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; ACE; ACE2; Angiotensin II; Bradykinin; RAS inhibitors; ACE inhibitors; AT1 receptor blockers; Losartan; Bradykinin Antagonists; Ang II loading; Giapreza; Icatibant.
Online: 14 April 2020 (14:34:43 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0023.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
anti-yeast; enzyme inhibitors; Terminalia mantaly; Combretaceae
Online: 3 November 2016 (09:35:17 CET)
ARTICLE
|
doi:10.20944/preprints202005.0016.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; elderly; proton pump inhibitors; antipsychotics; metformin; oral antidiabetics
Online: 2 May 2020 (15:48:33 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0022.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
HPPD inhibitors; pharmacophore model; molecule docking; HipHop model; virtual screening; ChemDiv
Online: 5 June 2017 (05:16:39 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
REVIEW
|
doi:10.20944/preprints201902.0101.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
age-related macular degeneration; anti-inflammatory agents; dry AMD; geographic atrophy; intravitreal injection; complement inhibitors; neuroprotective agents; non-exudative AMD
Online: 12 February 2019 (11:00:52 CET)
ARTICLE
|
doi:10.20944/preprints202004.0439.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV-2; COVID-19; spike glycoprotein; variability; molecular docking; molecular dynamics; inhibitors
Online: 24 April 2020 (11:42:01 CEST)
REVIEW
|
doi:10.20944/preprints201805.0129.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
BET inhibitors; HDAC inhibitors; pancreatic cancer; aberrant transcription; enhancers; transcription factors; distal regulatory elements; MYC; FOXA1; BRD4
Online: 8 May 2018 (10:47:27 CEST)
REVIEW
|
doi:10.20944/preprints202102.0150.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
CTLA-4; Treg cells: Immune checkpoint inhibitors; CD28; Antigen Presenting Cells
Online: 5 February 2021 (09:35:47 CET)
ARTICLE
|
doi:10.20944/preprints202103.0752.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Mixture toxicity; Neurotoxicity; Antagonism; Organophosphate; Acetylcholinesterase inhibitors; GABA; Behavior; Risk assessment; Spontaneous movement activity
Online: 31 March 2021 (07:52:05 CEST)
ARTICLE
|
doi:10.20944/preprints201812.0362.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Antibiotic resistance, efflux pump inhibitors, Escherichia coli, efflux pumps, multidrug resistance, Staphylococcus aureus
Online: 31 December 2018 (09:55:32 CET)
ARTICLE
|
doi:10.20944/preprints201807.0199.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
ALS-inhibitors; horseweed; multiple-resistance; alternative chemical control
Online: 11 July 2018 (11:56:59 CEST)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)
REVIEW
|
doi:10.20944/preprints201803.0227.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Antivenom; snakebite; small molecule toxin inhibitors; oligonucleotides; antibodies; phage display; next generation antivenom; recombinant antivenom
Online: 27 March 2018 (13:41:46 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0196.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
comorbid diseases; erectile dysfunction; penile duplex doppler ultrasound; penile pathology; phosphodiesterase type 5 inhibitors
Online: 22 January 2018 (09:03:17 CET)
REVIEW
|
doi:10.20944/preprints202004.0331.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; associated comorbidities; treatment; ACE2 inhibitors; Type 2 diabetes
Online: 19 April 2020 (05:42:22 CEST)
REVIEW
|
doi:10.20944/preprints202103.0262.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
immune checkpoint inhibitors; immune checkpoint radiolabeled antibodies; PD-1; PD-L1; immune PET; immunotherapy; AI; Radiomics; Deep learning; CAR-T cells
Online: 9 March 2021 (11:12:55 CET)
ARTICLE
|
doi:10.20944/preprints201908.0223.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
LSD1; molecular inhibitors; thieno[3,2-b]pyrrole-5-carboxamide derivatives; Molecular docking; 3D-QSAR; Molecular dynamics simulations
Online: 21 August 2019 (09:54:43 CEST)
REVIEW
|
doi:10.20944/preprints202012.0343.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; platelet activating factor; thrombosis; inflammation; Mediterranean diet; PAF-inhibitors
Online: 14 December 2020 (14:16:37 CET)
ARTICLE
|
doi:10.20944/preprints201911.0094.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
hPSCs; ROCK inhibitors; fasudil; cell survival; metabolism; differentiation
Online: 8 November 2019 (10:41:13 CET)
REVIEW
|
doi:10.20944/preprints201903.0288.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Enhancers; BET inhibitors; CDK7 inhibitors; HDAC inhibitors; Transcription factors; eRNAs; cancer
Online: 30 March 2019 (08:33:07 CET)
ARTICLE
|
doi:10.20944/preprints201806.0131.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
histone demethylase inhibitors; DNA damage; epigenetic drugs; breast cancer
Online: 8 June 2018 (12:29:10 CEST)
ARTICLE
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
kinase inhibitors; pure drug nanoparticles; drug nanocrystals; bottom-up nanonization; nanoprecipitation; microfluidics; flow focusing technologies
Online: 2 March 2021 (11:29:18 CET)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201810.0103.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Nipah Virus, outbreak, inhibitors, QSAR, database, prediction algorithm
Online: 5 October 2018 (15:04:23 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0079.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer’s disease (AD); amyloid precursor protein (APP); familial AD (FAD); sporadic AD (SAD); BACE1 inhibitors; APP-independent generation of beta amyloid
Online: 6 April 2018 (15:16:08 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0027.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
microginins; cyanobacteria; Microcystis; aminopeptidase M inhibitors
Online: 5 January 2018 (04:16:23 CET)
ARTICLE
|
doi:10.20944/preprints201905.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminopeptidases; inhibitors; aminophosphonate; phenylglycine analogues; fluorine substituted; molecular modeling
Online: 6 May 2019 (10:16:45 CEST)
REVIEW
|
doi:10.20944/preprints201806.0056.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
mTOR; mTORC1; mTORC2; rapamycin; rapalogues; rapalogs; mTOR inhibitors; senescence; ageing; aging; cancer; neurodegeneration; immunosenescence; senolytics; biomarkers
Online: 5 June 2018 (09:49:19 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0319.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
cyanobacteria; protease inhibitors; digestive enzyme; daphnia; HPLC; UV/Vis
Online: 27 May 2019 (12:56:49 CEST)
REVIEW
|
doi:10.20944/preprints201809.0435.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Acute Myeloid Leukemia; FLT3; Tyrosine kinase inhibitors; resistance
Online: 21 September 2018 (10:28:34 CEST)
REVIEW
|
doi:10.20944/preprints201905.0358.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
alloimmune response; immunosuppressants; calcineurin inhibitors; corticosteroids; mTOR inhibitors; neurotoxicity; neuroprotective effects
Online: 29 May 2019 (16:37:44 CEST)
REVIEW
|
doi:10.20944/preprints202108.0364.v1
Subject:
Medicine And Pharmacology,
Tropical Medicine
Keywords:
dengue virus; antiviral targets; NS5; flavivirus; polymerase; nucleoside inhibitors; non-nucleoside inhibitors
Online: 17 August 2021 (14:07:29 CEST)
ARTICLE
|
doi:10.20944/preprints201906.0074.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
agrobacterium tumefaciens-mediated transformation; citrus fruit; metal ion chelators; fruit-fungal interaction; transcription factor; virulence; protease inhibitors
Online: 10 June 2019 (09:56:16 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0609.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immune checkpoint inhibitors; immune-related adverse events (irAEs); tolerance; ipilimumab; nivolumab; interleukin-2; hyperthermia; low-dose-combination therapy
Online: 28 November 2018 (10:23:31 CET)
ARTICLE
|
doi:10.20944/preprints202102.0408.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
NhaP2-type cation-proton antiporter; Vibrio cholerae; Amiloride Analogs; Inhibitors against NhaP-type antiporters
Online: 18 February 2021 (10:39:07 CET)
ARTICLE
|
doi:10.20944/preprints202108.0327.v3
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Melanoma; Core regulatory network; in silico perturbationSystems pharmacology; Boolean model; Small molecule inhibitors; Virtual screening; ADME; E2F1
Online: 12 June 2023 (10:22:29 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0540.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
3-hydroxy-3-methylglutaryl-coenzyme-A inhibitors; Sepsis
Online: 27 July 2018 (13:07:17 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Antivirals; coronavirus; COVID-19; covalent drugs; dynamic light scattering; inhibitors; main protease; natural products
Online: 28 November 2022 (13:40:01 CET)
REVIEW
|
doi:10.20944/preprints201903.0256.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immunocheckpoint inhibitors; chemotherapy; tirosin kinase inhibitors; angiogenesis
Online: 28 March 2019 (06:48:37 CET)
ARTICLE
|
doi:10.20944/preprints201911.0010.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
aromatase inhibitors; anastrozole; levonorgestrel-iud; endometriosis; endometriomas; clinical trial
Online: 1 November 2019 (12:47:34 CET)
REVIEW
|
doi:10.20944/preprints202204.0202.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Metabolic syndrome; SGLT2 inhibitors; Dapagliflozin; Empagliflozin; Canagliflozin; Translational modeling
Online: 21 April 2022 (10:12:04 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0251.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Vorinostat, histone deacetylase, HDAC inhibitors, dibenzodiazocines, hydroxamic acid, selectivity
Online: 11 May 2021 (15:35:00 CEST)
ARTICLE
|
doi:10.20944/preprints201812.0064.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
combinatorial search forest; sensitivity analysis; support vector ranking algorithm; unknown biological hypotheses; Wnt pathway; PORCN-WNT inhibitors; ETC-1922159; Sobol indices; Hilbert Schmidt independence criterion indices (HSIC); F-divergence (Fdiv); systems biology
Online: 5 December 2018 (07:52:17 CET)
ARTICLE
|
doi:10.20944/preprints202201.0380.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Therapeutic biomarkers; circulating tumor cells; Immunocytochemistry; targeted therapy; Fluorescence in situ hybridization (FISH); Immune Checkpoint Inhibitors; Liquid Biopsy; Hormonal Treatments; Breast Cancer; Lung Cancer
Online: 25 January 2022 (11:31:05 CET)
REVIEW
|
doi:10.20944/preprints201902.0245.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cyclin-dependent kinases; cyclin-dependent kinase 4 and 6 inhibitors; targeted therapies; breast cancer
Online: 27 February 2019 (04:48:54 CET)
REVIEW
|
doi:10.20944/preprints201810.0577.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
myeloma; daratumumab; elotuzumab; isatuximab; CD38; JNJ- 63723283; denosumab; checkpoint inhibitors; BCMA; bispecific T-cell engager; antibody-drug conjugates
Online: 24 October 2018 (12:11:23 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0209.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Vezf1; angiogenesis; vascular biology; endothelial cells; MSS31, tube formation, small molecule inhibitors computational modeling.
Online: 15 May 2018 (08:08:15 CEST)
REVIEW
|
doi:10.20944/preprints202108.0372.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immune checkpoint inhibitors; non-small cell lung carcinoma; PD-1; PD-L1; immune PET; immunotherapy; Radiomics; PET/CT
Online: 18 August 2021 (08:20:43 CEST)
REVIEW
|
doi:10.20944/preprints202104.0679.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Sildenafil; phosphodiesterase 5 inhibitors; drug repurposing; cancer; chemoadjuvant
Online: 26 April 2021 (15:02:08 CEST)
REVIEW
|
doi:10.20944/preprints202201.0468.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Flavivirus; NS2B-NS3; ZIKA Virus; Dengue Virus; West Nile Virus; Inhibitors
Online: 31 January 2022 (13:46:44 CET)
CASE REPORT
|
doi:10.20944/preprints202201.0298.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Checkpoint inhibitors; Immune related adverse events; Cholestasis; Severe ductopenia; Vanishing bile duct syndrome
Online: 20 January 2022 (11:07:21 CET)
ARTICLE
|
doi:10.20944/preprints202102.0525.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
HIV-RT; ribonuclease H; dual inhibitors; docking; putative binding
Online: 23 February 2021 (15:51:40 CET)
ARTICLE
|
doi:10.20944/preprints202104.0270.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Systemic amyloidosis; amyloid fibrils; amyloidogenesis inhibitors; antibody light chains; light chain stabilizers; doxycycline; EGCG; thioflavin T; filter trap; PAINS
Online: 9 April 2021 (15:07:24 CEST)
REVIEW
|
doi:10.20944/preprints202205.0290.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cholesterol; PCSK9 inhibitors; HMG-CoA; LDL receptor; statins
Online: 23 May 2022 (10:01:24 CEST)
REVIEW
|
doi:10.20944/preprints202105.0430.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ethylene biosynthesis; ethylene inhibitors; in vitro culture; plant hormones; S-adenosylmethionine; stress responses
Online: 19 May 2021 (07:50:29 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0307.v3
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Immune Checkpoint Inhibitors; anti-PD-1/PDL-1; anti-CTLA-4; gender; sex; Nivolumab; Pembrolizumab; Atezolizumab; Ipilimumab; Durvalumab
Online: 15 November 2018 (07:02:24 CET)
REVIEW
|
doi:10.20944/preprints201809.0364.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
clear cell renal cell carcinoma; hypoxia inducible factors (HIFs); selenium; PD-L1; miRNA; VEGF; mTOR inhibitors
Online: 19 September 2018 (05:10:22 CEST)
REVIEW
|
doi:10.20944/preprints201909.0140.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; immune checkpoint inhibitors; HCC; pembrolizumab; nivolumab; immune microenvironment; targeted therapies
Online: 14 September 2019 (18:37:29 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0565.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 transcription; HIV-1 Tat; TAR RNA; small molecule inhibitors
Online: 23 June 2021 (11:04:21 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0115.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
triterpenoids; Acacia stem bark; polypharmacology; protein kinase inhibitors
Online: 3 June 2021 (13:04:47 CEST)
REVIEW
|
doi:10.20944/preprints202108.0037.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ovarian cancer; checkpoint inhibitors; ICIs; immunotherapy; PARP; avelumab; pembrolizumab; nivolumab; bevacizumab; platinum
Online: 2 August 2021 (13:01:35 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0174.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Phosphodiesterase (PDE); natural products; inhibitors; Protein Kinase; selectivity; fluorescence polarization
Online: 6 April 2021 (12:07:58 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0221.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Fatty Acid Amide Hydrolase; cannabinoid; carboxamide inhibitors; 3D-QSAR; CoMSIA.
Online: 8 November 2018 (14:52:23 CET)
REVIEW
|
doi:10.20944/preprints201910.0255.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antimicrobial resistance; biofilm; efflux pump inhibitors; antibiotic potentiation; eskapee pathogens; gram-negative bacteria
Online: 22 October 2019 (10:22:56 CEST)
REVIEW
|
doi:10.20944/preprints202305.0751.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Skin pigmentation; melanin; Tyrosinase inhibitors; hypopigmentation; hyperpigmentation; Vitiligo; skin-lightening; Depigmentation
Online: 10 May 2023 (11:32:48 CEST)
REVIEW
|
doi:10.20944/preprints202005.0392.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
RAAS inhibitors; COVID-19; coronavirus; angiotensin; clinical outcome; antihypertensive
Online: 24 May 2020 (17:48:42 CEST)
REVIEW
|
doi:10.20944/preprints202012.0167.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Matrix metalloproteinase; MMPs; protease; TIMPs; exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; TAILS
Online: 24 March 2021 (16:23:28 CET)
REVIEW
|
doi:10.20944/preprints202103.0063.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
breast cancer, CDK inhibitors, liquid biopsy, resistance mechanisms, therapy
Online: 2 March 2021 (09:53:38 CET)
REVIEW
|
doi:10.20944/preprints202009.0449.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
oleaginous microorganisms; microbial lipids; lignocellulose pretreatment; enzymatic hydrolysis; inhibitors
Online: 19 September 2020 (05:16:42 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0133.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
aging; angiotensin-converting enzyme inhibitors; nutrient metabolism; genetic background; nutritional stress
Online: 29 October 2018 (10:33:59 CET)
REVIEW
|
doi:10.20944/preprints202105.0140.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Adsorption; Scale Inhibitors; Fine sands; Colloids; Reservoir
Online: 7 May 2021 (10:42:36 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 25 January 2021 (15:01:17 CET)
REVIEW
|
doi:10.20944/preprints202104.0016.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Immune checkpoint inhibitors; pediatric solid tumor; immune suppression
Online: 1 April 2021 (12:22:35 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0425.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cancer; immune checkpoint inhibitors; survival; antibiotic; meta-analysis
Online: 29 March 2020 (06:43:23 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0279.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
NS3 inhibitors; allosteric inhibitors; NS4A; peptidomimetics; imidazole; hepatitis C virus; molecular dynamics; Flaviviridae; DSLS; binding assay
Online: 24 January 2020 (11:11:46 CET)
ARTICLE
|
doi:10.20944/preprints202105.0638.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 26 May 2021 (13:14:06 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0142.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
glioblastoma; immunotherapy; radiotherapy; brain cancers; radioimmunotherapy; immune checkpoint inhibitors; temozolomide; durvalumab; immunoradiotherapy.
Online: 10 May 2022 (13:22:16 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0772.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitors; immune-related endocrine dysfunction; hypothyroidism; targeted therapy; malignancy
Online: 31 May 2021 (12:49:40 CEST)
REVIEW
|
doi:10.20944/preprints201907.0286.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 Gag; Gag inhibitors; Protease; Protease inhibitors; drug resistance mutations; drug design
Online: 25 July 2019 (10:05:03 CEST)
REVIEW
|
doi:10.20944/preprints202104.0667.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
breast cancer; CDK inhibitors; liquid biopsy; resistance mechanisms; therapy
Online: 26 April 2021 (12:57:01 CEST)
ARTICLE
|
doi:10.20944/preprints202110.0171.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
chronic myeloid leukemia; dasatinib; ponatinib; pimozide; STAT inhibitors; K562
Online: 11 October 2021 (16:17:32 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0221.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
hCA IX and XII; dual inhibitors; molecular modeling studies; in vitro assays
Online: 11 July 2020 (02:30:03 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0170.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SonoCloud; GL261 mouse model; ultrasound-mediated drug delivery; glioblastoma; immune checkpoint inhibitors
Online: 9 December 2022 (02:59:28 CET)
ARTICLE
|
doi:10.20944/preprints202109.0429.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; hepatic arterial infusion chemotherapy; cisplatin; sorafenib; multikinase inhibitors; risk factors; propensity score-matched analysis
Online: 24 September 2021 (12:38:25 CEST)
ARTICLE
|
doi:10.20944/preprints202109.0375.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
HIV-protease inhibitors; pseudo-symmetric core; heteroaryl carboxyamides; synthesis; biological screening; molecular modeling
Online: 22 September 2021 (10:44:16 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
REVIEW
|
doi:10.20944/preprints202111.0087.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virome; microbiota; cancer; bacteriophages; fecal microbiota transplantation; checkpoint inhibitors; immunotherapy
Online: 3 November 2021 (14:30:14 CET)
REVIEW
|
doi:10.20944/preprints201809.0291.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
CCR6, CCL20, Inhibitors, TH17, Treg, Inflammatory diseases, Cancer
Online: 17 September 2018 (09:31:43 CEST)
REVIEW
|
doi:10.20944/preprints201911.0264.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
cardiovascular risk; dipeptidyl peptidase-4 inhibitors; glucagon like peptide-1 receptor agonists; sodium glucose cotransporter-2 inhibitors; type 2 diabetes mellitus
Online: 24 November 2019 (04:26:47 CET)
COMMUNICATION
|
doi:10.20944/preprints202012.0365.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
corrosion; amino acids; inhibitors; steel; iron; Monte Carlo simulation
Online: 15 December 2020 (10:09:29 CET)
ARTICLE
|
doi:10.20944/preprints202109.0520.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Phytoene, Dunaliella salina, mitosis inhibitors, herbicides, red light
Online: 30 September 2021 (14:18:55 CEST)
ARTICLE
|
doi:10.20944/preprints202110.0297.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
gastric cancer; immunotherapy; immune checkpoint blockade (ICB); immune checkpoint inhibitors (ICI),; DNA repair gene signature (DRGS); prognostic biomarker; score system
Online: 20 October 2021 (22:47:19 CEST)
REVIEW
|
doi:10.20944/preprints202110.0298.v1
Subject:
Medicine And Pharmacology,
Orthopedics And Sports Medicine
Keywords:
Osteoarthritis; LithoLexal; Lithothamnion; Disease-modifying adjunctive therapy; Anti-inflammatory agents; Cytokine inhibitors
Online: 20 October 2021 (22:49:47 CEST)
ARTICLE
|
doi:10.20944/preprints202203.0405.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
α-amylase inhibitors; diabetes; hemi-pyocyanin; marine discards; microbial conversion
Online: 31 March 2022 (10:47:24 CEST)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)