REVIEW
|
doi:10.20944/preprints201910.0144.v6
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus; antiviral drug; drug discovery; drug development; broad-spectrum antivirals
Online: 14 February 2020 (02:27:24 CET)
REVIEW
|
doi:10.20944/preprints202010.0179.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Non Michaelis-Menten Kinetics; High-throughput screening; allostery; cooperativity; processive kinetics; distributive kinetics; single-molecule; auto-catalytic; drug discovery
Online: 8 October 2020 (13:34:16 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0025.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
drug repurposing; translational bioinformatics; transcriptomics; transcriptome analysis; drug discovery; protocol; gene expression
Online: 9 October 2016 (08:42:23 CEST)
REVIEW
|
doi:10.20944/preprints201805.0011.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
computational drug repositioning; drug repositioning; drug repurposing; machine learning; deep learning; crowdsourcing; open innovation; drug discovery
Online: 1 May 2018 (12:27:22 CEST)
REVIEW
|
doi:10.20944/preprints202105.0346.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
drug discovery; drug repurposing; bioinformatics; machine learning; artificial intelligence; biomedical discoveries etc.
Online: 14 May 2021 (15:17:50 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1523.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Biomarker discovery; disease pathogenesis; autoimmunity; antigenic mimicry; machine learning
Online: 23 November 2023 (11:10:59 CET)
CONCEPT PAPER
|
doi:10.20944/preprints202011.0250.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
antibiotic discovery; STEM education; biosynthetic gene cluster; molecular networking; multi-omics
Online: 6 November 2020 (16:50:46 CET)
ARTICLE
|
doi:10.20944/preprints202006.0258.v2
Subject:
Engineering,
Civil Engineering
Keywords:
Conservation laws; Data inference; Data discovery; Dimensionless form; PINN
Online: 30 September 2020 (03:51:25 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0132.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
arylamine N-acetyltransferases; cancer; tuberculosis; drug discovery; traditional Chinese medicine; virtual screening; molecular dynamics simulation; MM-PBSA
Online: 30 June 2017 (11:36:22 CEST)
REVIEW
|
doi:10.20944/preprints202008.0320.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Data Science; Machine Learning; Deep Learning; Genomics; COVID-19; Drug Discovery; Image Analysis; Interactomics; Epidemiology
Online: 14 August 2020 (11:01:56 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0602.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; Genomes; microRNA; SARS-CoV-2; Variant discovery
Online: 25 September 2020 (10:14:46 CEST)
REVIEW
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
web server; rational design; functionalizing enzymes; enzyme discovery; user-friendly tools
Online: 28 January 2021 (07:51:45 CET)
ARTICLE
|
doi:10.20944/preprints201704.0117.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
Body sensor network; Smart home, knowledge discovery in BSN data; frequent patterns; periodic patterns and productive pattern.
Online: 18 April 2017 (18:15:50 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0191.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
High-dimensional data analysis, Multiple hypothesis testing, False discovery rate, Optimum significance threshold, Maximum for reasonable number of rejected hypotheses, Big data analysis
Online: 24 March 2017 (18:29:35 CET)
REVIEW
|
doi:10.20944/preprints202012.0372.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Vicia faba; genomic resources; mapping population; gene discovery; breeding
Online: 15 December 2020 (10:38:24 CET)
ARTICLE
|
doi:10.20944/preprints201902.0140.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus discovery; Chlamydia pecorum; Koala; picornavirus; phylogeny
Online: 15 February 2019 (07:33:16 CET)
REVIEW
|
doi:10.20944/preprints202105.0567.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Artificial intelligence AI; machine learning; algorithms; QSAR; drug discovery
Online: 24 May 2021 (13:02:21 CEST)
REVIEW
|
doi:10.20944/preprints201812.0273.v3
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
mutations; disease-causing mutations; polymorphism; folding free energy change; binding free energy change; drug discovery; in silico screening
Online: 28 January 2019 (11:39:23 CET)
ARTICLE
|
doi:10.20944/preprints202004.0524.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
unsupervised learning; tensor decomposition; feature selection; COVID-19; drug discovery; gene expression
Online: 3 June 2020 (05:29:09 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
COVID-19; SARS-CoV-2; in silico drug discovery; gene expression profile; tensor decomposition; feature extraction
Online: 8 December 2020 (10:17:05 CET)
REVIEW
|
doi:10.20944/preprints202005.0342.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
seaweed; metabolites; neuroprotection; Alzheimer’s disease; Parkinson’s disease; ischemic stroke; computer-aided drug discovery
Online: 21 May 2020 (09:49:29 CEST)
REVIEW
|
doi:10.20944/preprints201804.0126.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
pharmaceutical market; drugs; drug discovery; solid-phase peptide synthesis
Online: 10 April 2018 (10:14:33 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0343.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
GALAXY; Assembly; Annotation; Genomic Variants Discovery; Workflow
Online: 21 May 2020 (09:57:42 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0172.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
COVID-19; Twitter; Topic Discovery; Arabic
Online: 9 July 2020 (07:25:19 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0512.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
oyster mushroom (Pleurotus sp.); PARP protein; 4UND protein; molecular docking; PyRx; BIOVIA drug discovery
Online: 26 August 2021 (16:15:06 CEST)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)
REVIEW
|
doi:10.20944/preprints201901.0273.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Mycobacterium abscessus; non-tuberculous mycobacteria; antimicrobial drug discovery; cystic fibrosis
Online: 28 January 2019 (10:05:28 CET)
ARTICLE
|
doi:10.20944/preprints201811.0627.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemical space; chemical data set; chemoinformatics; consensus diversity plot; drug discovery; molecular diversity; visualization
Online: 30 November 2018 (10:06:15 CET)
ARTICLE
|
doi:10.20944/preprints201908.0100.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cancer biomarker discovery; gene expression data; Ingenuity Knowledge Base (IKB); transfer learning; interpretable classification rules
Online: 8 August 2019 (05:28:26 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0160.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
false discovery rate; machine learning; protein function prediction; support vector machine; BLAST
Online: 24 November 2017 (11:14:05 CET)
ARTICLE
|
doi:10.20944/preprints202005.0007.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
process mining; business process; fastText; email logs; Process Model Discovery
Online: 2 May 2020 (12:19:14 CEST)
ARTICLE
|
doi:10.20944/preprints201803.0144.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
sea anemone; drug discovery; cancer; antiangiogenic; endothelial cells; RGD motif; Kunitz type inhibitor
Online: 19 March 2018 (08:15:38 CET)
ARTICLE
|
doi:10.20944/preprints202302.0250.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
AI drug discovery; mTOR; rapalog; C. elegans; cancer; longevity
Online: 15 February 2023 (02:42:57 CET)
ARTICLE
|
doi:10.20944/preprints201811.0561.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cheminformatics, drugs, drug-likeness, drug discovery, natural products
Online: 23 November 2018 (13:56:32 CET)
REVIEW
|
doi:10.20944/preprints202104.0244.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Staphylococcus aureus; MRSA; genome-scale metabolic models; model-driven discovery; strain-specific models
Online: 8 April 2021 (14:25:31 CEST)
ARTICLE
|
doi:10.20944/preprints202010.0196.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
drug discovery; artificial intelligence; protein discovery; binding prediction; synthetic molecule generation; synthetic drug
Online: 20 November 2020 (11:30:03 CET)
ARTICLE
|
doi:10.20944/preprints202210.0223.v3
Subject:
Biology And Life Sciences,
Virology
Keywords:
Drug discovery; Systems biology; SARS-CoV-2; Dengue; Influenza A; RSV; cell viability analysis; antivirals; in vitro validation; in vivo validation
Online: 22 March 2024 (16:46:59 CET)
ARTICLE
|
doi:10.20944/preprints202107.0315.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Myxobacteria; myxochelin; nicotinic acid; secondary metabolites; natural product discovery; precursor-directed biosynthesis; total synthesis
Online: 14 July 2021 (10:03:32 CEST)
ARTICLE
|
doi:10.20944/preprints201806.0143.v1
Subject:
Arts And Humanities,
Philosophy
Keywords:
induction; naturalism; evidence and justification; epistemic norms; induction and concept formation; induction and discovery of laws
Online: 8 June 2018 (16:24:17 CEST)
ARTICLE
|
doi:10.20944/preprints201911.0024.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
Iranian traditional medicine; Persian medicine; ontology; knowledge-base; Mizaj; temperament; new drug discovery
Online: 3 November 2019 (17:07:50 CET)
REVIEW
|
doi:10.20944/preprints202004.0012.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; chemical space; database; LANaPD; molecular diversity; drug discovery; natural sources
Online: 2 April 2020 (04:47:13 CEST)
ARTICLE
|
doi:10.20944/preprints202202.0349.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Hypoxia-inducible factor; cancer; hypoxia; drug discovery; medicinal chemistry; virtual screening; molecular dynamics simulation; MM-PBSA; Drug discovery
Online: 28 February 2022 (08:40:24 CET)
ARTICLE
|
doi:10.20944/preprints202101.0209.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
leafy greens; spinach; metabolomics; metabolic profiling; food pathogens; biomarker discovery
Online: 12 January 2021 (08:20:35 CET)
REVIEW
|
doi:10.20944/preprints202006.0078.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
COVID-19; vaccine; vaccine development; vaccine discovery; systems biology; machine learning; platform technologies; adjuvants; smart clinical trials; human genetics; regulatory convergence; real world evidence; vaccines safety
Online: 7 June 2020 (10:11:02 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0063.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
FABP4; A-FABP; aP2; antidiabetes; antiobesity; antiatherosclerosis; anticancer; computational tools; computer-aided drug discovery
Online: 5 September 2019 (15:39:58 CEST)
REVIEW
|
doi:10.20944/preprints202106.0305.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
dietary flavonoids; cardioprotective effects; ROS scavenging; myocardial dysfunction; bioavailability and drug metabolism; toxicity; drug discovery
Online: 11 June 2021 (08:44:01 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0574.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
activity cliff; activity landscape plotter; epigenetics; docking; drug discovery; D-tools; molecular dynamics; Epi-polypharmacology; SmART; structure-activity relationships
Online: 26 November 2018 (07:14:05 CET)
REVIEW
|
doi:10.20944/preprints202006.0229.v1
Subject:
Public Health And Healthcare,
Health Policy And Services
Keywords:
SARS-CoV-2; COVID-19; Recovery trial; Discovery trial
Online: 18 June 2020 (09:23:27 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0059.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Metallothionein (MT); Scientific discovery; Scientific pursuit; Research strategies; upward looking research; Exploratory research; Protein function; Compensation; Moonlighting; multifunctional proteins; Vestiges
Online: 2 March 2021 (09:39:39 CET)
ARTICLE
|
doi:10.20944/preprints201809.0587.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
machine learning; conotoxins; cone snails; venom; drug discovery
Online: 29 September 2018 (07:39:42 CEST)
ARTICLE
|
doi:10.20944/preprints201907.0220.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
diversity; fragment-based drug discovery; library design; library size
Online: 19 July 2019 (07:54:41 CEST)
REVIEW
|
doi:10.20944/preprints202001.0324.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
natural products; sirtuin; drug discovery; epigenetics; structure–activity relationship
Online: 27 January 2020 (09:21:29 CET)
REVIEW
|
doi:10.20944/preprints202204.0151.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Isocyanide-based multicomponent reactions; Antimicrobial Discovery; Antibiotic Resistance; Public Health
Online: 18 April 2022 (03:38:08 CEST)
ARTICLE
|
doi:10.20944/preprints202111.0329.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Machine Learning; Deep Learning; Molecular Modeling; Virtual Screening; Drug Discovery
Online: 18 November 2021 (13:59:09 CET)
ARTICLE
|
doi:10.20944/preprints201912.0302.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
papillomavirus; feline; cat; felid; cancer; squamous cell carcinoma; phylogeny; discovery; pathogen; oncogenic
Online: 23 December 2019 (12:01:11 CET)
ARTICLE
|
doi:10.20944/preprints202109.0138.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Agaricus Bisporus; Button Mushroom; Molecular docking; PyRx software; BIOVIA Discovery studio
Online: 8 September 2021 (10:14:03 CEST)
HYPOTHESIS
|
doi:10.20944/preprints201808.0127.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Big Data, Systems Models, Cancer metabolism, Cancer personalized treatment, Drug Discovery.
Online: 6 August 2018 (15:09:15 CEST)
ARTICLE
|
doi:10.20944/preprints202204.0224.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID-19; SARS-CoV-2; drug discovery; multitargeting; computational drug repurposing
Online: 26 April 2022 (03:39:06 CEST)
ARTICLE
|
doi:10.20944/preprints202202.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cancer; tumor homing peptide; in silico drug discovery; complex network; chemical space network; centrality measure; similarity searching, group fusion; motif discovery; starPep toolbox software
Online: 3 February 2022 (10:14:05 CET)
ARTICLE
|
doi:10.20944/preprints201910.0074.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Pseudomonas aeruginosa; Quorum sensing; Virtual screening; E-pharmacophore; Drug discovery.
Online: 7 October 2019 (12:33:33 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0770.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
BRF2; cancer; molecular dynamics simulation; drug repurposing; drug discovery
Online: 16 July 2021 (11:40:34 CEST)
ARTICLE
Subject:
Environmental And Earth Sciences,
Paleontology
Keywords:
islands, discovery, settlement, colonization, Easter Island, Rapa Nui, Pacific Ocean, Polynesians, Amerindians
Online: 28 March 2019 (11:22:33 CET)
ARTICLE
|
doi:10.20944/preprints201811.0499.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
music acoustics, melody discovery, pitch tracking, Indian classical music
Online: 20 November 2018 (11:31:10 CET)
REVIEW
|
doi:10.20944/preprints202202.0067.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Antimalarial Drug; Malaria Vaccine; Drug Discovery; Artimisnine; K13; Malaria
Online: 4 February 2022 (10:22:34 CET)
REVIEW
|
doi:10.20944/preprints202109.0491.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Tuberculosis; Mycobacterium; Diagnostics; Drug Discovery; Antibiotics; Antimicrobial Re-sistance; Microfluidics; Single-Cell Analysis; Bioengineered Models
Online: 29 September 2021 (11:34:04 CEST)
ARTICLE
|
doi:10.20944/preprints201903.0121.v1
Online: 11 March 2019 (09:00:00 CET)
ARTICLE
|
doi:10.20944/preprints202205.0349.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Docking; lead discovery; molecular dynamic simulation; tuberculosis; coupled assay
Online: 25 May 2022 (10:11:26 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0322.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Hemolytic peptide; Network science; Half-Space Proximal Networks; Metadata Networks; Visual mining; Cluster analysis; Motif discovery; StarPep toolbox; Peptide drug discovery
Online: 17 March 2023 (10:05:05 CET)
ARTICLE
|
doi:10.20944/preprints202103.0084.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
price discovery; financial economics; clearing; credit default swaps; collateralization; OTC; risk premium; CCP.
Online: 2 March 2021 (12:05:53 CET)
REVIEW
|
doi:10.20944/preprints202304.0209.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Gut microbiome; Machine learning; Deep learning; Metagenomics; Autoimmune diseases; Biomarkers discovery; Diagnostic models
Online: 23 April 2023 (02:59:58 CEST)
REVIEW
|
doi:10.20944/preprints202201.0440.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
electrophiles; signaling; profiling; drug mechanism; drug discovery; T-REX
Online: 28 January 2022 (14:57:08 CET)
REVIEW
|
doi:10.20944/preprints201810.0701.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
tuberculosis; latency; non-replicating persistent; antibiotic; drug discovery; mycobacterium tuberculosis
Online: 14 November 2018 (10:24:31 CET)
REVIEW
|
doi:10.20944/preprints202208.0213.v2
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
GIBAC; Biophysics; Structural Biology; Drug discovery \& design; Artificial intelligence-integrated drug discovery
Online: 19 October 2023 (13:38:05 CEST)
ARTICLE
|
doi:10.20944/preprints202111.0266.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Pan-Cancer; somatic point mutations; cancer subtyping; biomarker discovery; driver genes; per-sonalized medicine; health data analytics
Online: 15 November 2021 (13:51:33 CET)
ARTICLE
|
doi:10.20944/preprints202205.0146.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
ubiquitous exposure; diagnosis; research design; quality of health care; habitat injuries; discovery
Online: 11 May 2022 (05:40:27 CEST)
ARTICLE
|
doi:10.20944/preprints201912.0049.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
natural product; drug discovery; protoflavonoid; continuous-flow chemistry; oxime; antitumor; antiviral; epstein-barr virus; lytic cycle
Online: 4 December 2019 (11:40:33 CET)
ARTICLE
|
doi:10.20944/preprints202111.0467.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
myxobacteria; secondary metabolites; biarylitide; natural product discovery; RiPPs; genome mining; myxarylin
Online: 25 November 2021 (10:42:39 CET)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
USP14; molecular docking; molecular dynamic simulation; cancer; ubiquitin; drug discovery
Online: 23 December 2019 (12:36:38 CET)
ARTICLE
|
doi:10.20944/preprints202303.0048.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Minimum Inhibitory Concentrations; Deep Learning; Regression; Antimicrobial peptides; Drug Discovery
Online: 3 March 2023 (01:29:51 CET)
REVIEW
|
doi:10.20944/preprints202109.0501.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Antigen Selection; Epitope Selection; Antibody Targeting; Epitope Accessibility; Antibody Engineering; Protein Engineering; Drug Targeting; Model-Informed Drug Discovery and Development
Online: 3 November 2021 (08:26:47 CET)
ARTICLE
|
doi:10.20944/preprints202111.0125.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
artificial intelligence; de novo design; fragment-based drug discovery; HIV-1 inhibitors; pseudo natural products
Online: 8 November 2021 (09:23:49 CET)
ARTICLE
|
doi:10.20944/preprints201811.0429.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
drug repurposing; drug repositioning; computational biology; drug discovery; computational pharmacology; malaria; multitargeting; malaria treatment
Online: 19 November 2018 (07:31:08 CET)
REVIEW
|
doi:10.20944/preprints202007.0523.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
discovery proteomics; targeted proteomics; mass spectrometry; fish allergens; crustacean allergens; mollusk allergens
Online: 22 July 2020 (11:23:40 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0326.v2
Subject:
Environmental And Earth Sciences,
Remote Sensing
Keywords:
GEO label; serverless; semantic sensor web; discovery; visualisation; sensor web
Online: 30 June 2020 (08:06:39 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0218.v1
Subject:
Business, Economics And Management,
Econometrics And Statistics
Keywords:
agricultural commodity futures; price discovery; market reflexivity; Hawkes process
Online: 13 May 2020 (03:35:53 CEST)
REVIEW
|
doi:10.20944/preprints202005.0408.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
drug discovery; machine learning; in silico; pharmacology
Online: 25 May 2020 (04:55:24 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0213.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Clustering; Pattern Discovery; Time series; Multi-Level Spectral Clustering; English Channel
Online: 8 August 2020 (18:00:26 CEST)
ARTICLE
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
c-src-tyrosine kinase; QSAR; molecular descriptors; virtual screening; drug discovery; cancer; molecular docking
Online: 25 October 2019 (11:21:43 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0253.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
ASFV; humoral responses; ASFV capsid proteins; ASFV vaccines; ASFV immunity; antigen discovery; luciferase antibody capture assay; luciferase immunoprecipitation assay; viral hemorrhagic fever.
Online: 14 March 2023 (09:43:57 CET)
ARTICLE
|
doi:10.20944/preprints202308.2113.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
herbs; spices; flavonoids; antioxidants; diabetes; volatile compounds; drug discovery; phytochemicals; human health
Online: 31 August 2023 (10:12:18 CEST)
REVIEW
|
doi:10.20944/preprints202304.0677.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Metabolomics; Simultaneous Quantitation and Discovery (SQUAD); Targeted Metabolomics; Untargeted Metabolomics
Online: 21 April 2023 (07:29:13 CEST)
REVIEW
|
doi:10.20944/preprints202401.1357.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
HIV-1; AIDS; FDA; Combination antiretroviral therapy; latent reservoirs; apoptosis; drug resistance; anti-HIV-1 drug design and discovery
Online: 18 January 2024 (10:29:57 CET)
REVIEW
|
doi:10.20944/preprints202307.0757.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Lippia javanica; Pharmacological; metabolites; ethnobotanical; drug discovery
Online: 12 July 2023 (05:42:56 CEST)
REVIEW
|
doi:10.20944/preprints202302.0234.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
lipid metabolism; Apicomplexa; drug discovery; calcium signaling; acidocalcisomes; parasite
Online: 14 February 2023 (04:42:12 CET)
REVIEW
|
doi:10.20944/preprints202208.0230.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; compound databases; chemical space; diversity; drug discovery; openscience; pseudo-natural product
Online: 12 August 2022 (08:39:40 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0907.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
cancer; protein degradation; degraders; drug discovery; PROTAC; CDK9
Online: 11 January 2024 (10:20:13 CET)
ARTICLE
|
doi:10.20944/preprints202301.0221.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Ion channels; Membrane proteins; Transmembrane proteins; Drug discovery; Protein language models; Convolutional Neural Network
Online: 12 January 2023 (09:21:08 CET)
ARTICLE
|
doi:10.20944/preprints202303.0193.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Antibiofilm peptide; chemical space; StarPep toolbox; complex network; centrality measure; motif discovery
Online: 10 March 2023 (09:36:30 CET)
ARTICLE
|
doi:10.20944/preprints202310.0425.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
hepatitis B; antiviral; drug discovery; HBc protein; pharmacophore-based screening; drug repurposing
Online: 8 October 2023 (05:11:37 CEST)
REVIEW
|
doi:10.20944/preprints202308.0887.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Drug Discovery; Drug Repurposing; SARS-CoV-2; COVID; Molecular Docking; QSAR; Molecular Dynamic; Virtual Screening; Drug Design
Online: 11 August 2023 (09:03:55 CEST)