ARTICLE
|
doi:10.20944/preprints201611.0121.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
tissue microarray; immunohistochemistry; cancer imaging; tyrosine kinase receptor; normal tissue; colon cancer
Online: 24 November 2016 (11:07:23 CET)
ARTICLE
|
doi:10.20944/preprints201703.0225.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
acute lung injury; fasudil, Rho kinase; endothelial function; inflammation
Online: 31 March 2017 (08:30:54 CEST)
REVIEW
|
doi:10.20944/preprints201705.0212.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
cancer; cell-surface receptor; EGFR; molecular mechanism; phosphorylation; receptor tyrosine kinase; transmembrane signal transduction
Online: 30 May 2017 (08:34:04 CEST)
ARTICLE
|
doi:10.20944/preprints201708.0015.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ischemia-reperfusion injury (IRI), ω3-PUFA, AMP-activated protein kinase (AMPK), autophagy
Online: 4 August 2017 (12:56:08 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0215.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
FGFR1; inhibitor; kinase inhibitor; pyrazine; hinge binder
Online: 30 March 2017 (04:13:45 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0018.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
pyruvate kinase M2; prostate cancer; cancer metabolism; mTOR; autophagy
Online: 3 January 2019 (12:32:52 CET)
ARTICLE
|
doi:10.20944/preprints201908.0238.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
aurora kinase A; molecular docking; DFT; MD simulation
Online: 23 August 2019 (05:01:40 CEST)
REVIEW
|
doi:10.20944/preprints201808.0044.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast tumor kinase (BRK); protein tyrosine kinase 6 (PTK6); breast cancer; pathways; therapeutics
Online: 2 August 2018 (09:58:55 CEST)
ARTICLE
|
doi:10.20944/preprints201707.0033.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
hepatic inflammation; high-fat-cholesterol diet; hypertension; mitogen-activated protein kinase; nonalcoholic steatohepatitis; nuclear factor erythroid 2-related factor 2 pathway; nuclear factor-kappa B; spontaneously hypertensive rat; stroke-prone spontaneously hypertensive5/Dmcr; Wistar Kyoto
Online: 14 July 2017 (10:54:38 CEST)
REVIEW
|
doi:10.20944/preprints201807.0237.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
TRPM7, kinase, inflammation, lymphocytes, calcium signalling, SMAD, TH17, hypersensitivity, regulatory T cells, thrombosis, graft versus host disease, T cells, innate immunity
Online: 13 July 2018 (14:14:56 CEST)
ARTICLE
|
doi:10.20944/preprints201911.0399.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
olivo-ponto-cerebellar atrophy (OPCA); Purkinje cells; Calcium/calmodulin dependent protein kinase II (CAMK2); Plastin (Fimbrin); Hirano bodies; Huntington’s disease
Online: 30 November 2019 (14:47:30 CET)
ARTICLE
|
doi:10.20944/preprints201802.0026.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pig eye perfusion model; pigmentary glaucoma; ocular hypertension; ocular hypotension; phagocytosis; rho-kinase inhibitor
Online: 5 February 2018 (03:39:57 CET)
REVIEW
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Parkinson’s disease; precision medicine; personalized medicine; GBA; Glucocerebrosidase; GCase; LRRK2; Leucine-rich repeat kinase-2; Dopamine; PD drug trials; PD risk variants
Online: 14 September 2020 (00:22:59 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0131.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pigmentary glaucoma; ROCK kinase inhibitor; RKI-1447; trabecular meshwork; phagocytosis; cytoskeleton
Online: 9 July 2018 (11:27:28 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0634.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
compound 3K; ovarian cancer; pyruvate kinase M2; autophagy; apoptosis
Online: 26 September 2020 (13:34:05 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0393.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
genetic code expansion, protein kinase B, phosphoinositide dependent kinase 1 (PDK1), phosphoseryl-tRNA synthetase (SepRS), tRNASep
Online: 21 July 2018 (12:35:26 CEST)
REVIEW
|
doi:10.20944/preprints201809.0435.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Acute Myeloid Leukemia; FLT3; Tyrosine kinase inhibitors; resistance
Online: 21 September 2018 (10:28:34 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0197.v1
Subject:
Biology And Life Sciences,
Plant Sciences
Keywords:
Cudratricusxanthone L; Cudrania tricuspidata; Neuroinflammation; Nuclear factor-kappa B (NF-κB); Mitogen-activated protein kinase (MAPK)
Online: 9 August 2018 (20:43:24 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ALK5 inhibitor; TGF-β; kinase assay; selectivity; docking
Online: 30 August 2018 (05:52:08 CEST)
REVIEW
|
doi:10.20944/preprints201903.0256.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immunocheckpoint inhibitors; chemotherapy; tirosin kinase inhibitors; angiogenesis
Online: 28 March 2019 (06:48:37 CET)
REVIEW
|
doi:10.20944/preprints201902.0245.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cyclin-dependent kinases; cyclin-dependent kinase 4 and 6 inhibitors; targeted therapies; breast cancer
Online: 27 February 2019 (04:48:54 CET)
REVIEW
|
doi:10.20944/preprints202012.0288.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
desmoplastic small round cell tumor; treatment; prognosis; surgery; radiotherapy; chemotherapy; tyrosine kinase receptor; target therapy; rare disease
Online: 11 December 2020 (15:53:20 CET)
ARTICLE
|
doi:10.20944/preprints201809.0322.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
p21-activated kinase (PAK); Pancreatic ductal adenocarcinoma (PDA); PF-3758309; gemcitabine
Online: 17 September 2018 (15:28:54 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0374.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
aldosterone; apoptosis; cardiac myocyte; eplerenone; fibrosis; finerenone; G protein-coupled receptor kinase (GRK)-5; mineralocorticoid receptor; mineralocorticoid receptor antagonist (MRA); signal transduction
Online: 17 September 2020 (05:24:29 CEST)
REVIEW
|
doi:10.20944/preprints201903.0138.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
extracellular signal-regulated kinase; MAPK/ERK signaling; intracellular signaling; kidney development; ureteric bud branching morphogenesis; nephrogenesis; progenitor cells; self-renewal; differentiation
Online: 13 March 2019 (09:00:32 CET)
REVIEW
|
doi:10.20944/preprints201811.0389.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
adverse remodeling; aldosterone; cardiac myocyte; crosstalk; G protein-coupled receptor (GPCR); GPCR-kinase (GRK); heart failure; inflammation; mineralocorticoid receptor; myocardial infarction; oxidative stress; signal transduction
Online: 16 November 2018 (07:54:04 CET)
ARTICLE
|
doi:10.20944/preprints201911.0061.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
rett syndrome; intrinsically disordered region; phylogenetic profile analysis; post-transcriptional modification; methyl-cpg-binding protein 2; cyclin-dependent kinase-like 5; forkhead box protein g1
Online: 6 November 2019 (10:58:54 CET)
ARTICLE
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
c-src-tyrosine kinase; QSAR; molecular descriptors; virtual screening; drug discovery; cancer; molecular docking
Online: 25 October 2019 (11:21:43 CEST)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
ARTICLE
|
doi:10.20944/preprints202203.0290.v2
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
host-virus interactions; tissue-specific model; COVID-19; SARS-CoV-2; antiviral targets; flux balance analysis; flux variability analysis; reaction knockout; host-derived enforcement; metabolic modeling; virus mutations; nucleoside diphosphate kinase; software engineering; Python
Online: 27 July 2022 (10:37:12 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0343.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
protein; exercise; muscle damage; creatine kinase; myoglobin; inflammation
Online: 16 July 2020 (06:33:18 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0349.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
MAP kinase; ERK5; Bmk1; SUMO; nuclear translocation; transcription; cell proliferation; cancer; Hsp90; Cdc37
Online: 29 January 2020 (05:00:39 CET)
ARTICLE
|
doi:10.20944/preprints202106.0115.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
triterpenoids; Acacia stem bark; polypharmacology; protein kinase inhibitors
Online: 3 June 2021 (13:04:47 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0278.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
astrocytes; glutamine; SN1 (SNAT3); Sp1; protein kinase C; ammonia; transport
Online: 12 November 2018 (10:02:12 CET)
COMMUNICATION
|
doi:10.20944/preprints202106.0309.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
mTORC1; RHEB; G-Protein; Allosteric activation; Kinase domain; Binding kinetics
Online: 11 June 2021 (09:14:14 CEST)
ARTICLE
|
doi:10.20944/preprints201907.0013.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Rett Syndrome; intrinsically disordered region; phylogenetic profile analysis; post-transcriptional modification; methyl-CpG-binding protein 2; cyclin-dependent kinase-like 5; forkhead box protein G1
Online: 1 July 2019 (11:59:56 CEST)
REVIEW
|
doi:10.20944/preprints201808.0403.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
p-21 activated kinase; pioglitazone, metformin, type 2 diabetes mellitus, cancer, chemoprevention, and inflammation.
Online: 23 August 2018 (05:10:55 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0251.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Trichoderma atroviride; mycoparasitism; secondary metabolites; 6-pentyl-alpha-pyrone; Tmk3 MAP kinase; light; dark
Online: 11 September 2020 (08:49:15 CEST)
REVIEW
|
doi:10.20944/preprints202112.0518.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell non-Hodgkin lymphoma (B-NHL); B-cell receptor (BCR); Bruton’s tyrosine kinase (BTK); spleen tyrosine kinase (SYK); phosphoinositide-3-kinase (PI3K); ibrutinib; acalabrutinib; copanlisib; idelalisib; umbralisib; fostamatinib; combination therapies
Online: 31 December 2021 (12:23:29 CET)
COMMUNICATION
|
doi:10.20944/preprints202104.0275.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
fludioxonil; fungicide; mode of action; high osmolarity glycerol (HOG) pathway; Magnaporthe oryzae; signal transduction; histidine kinase; MoHIK1; HIK1; phenylpyrrole
Online: 12 April 2021 (09:38:33 CEST)
REVIEW
|
doi:10.20944/preprints201809.0360.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
p-21 activated kinase; pioglitazone, metformin, type 2 diabetes mellitus, cancer, chemoprevention, and inflammation.
Online: 19 September 2018 (00:50:05 CEST)
REVIEW
|
doi:10.20944/preprints201907.0256.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
PI 3-kinase; chromosomal instability; PI3K inhibitor; cancer; tumour evolution; centrosome
Online: 23 July 2019 (11:01:34 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0339.v1
Subject:
Biology And Life Sciences,
Plant Sciences
Keywords:
Banana; fine mapping; quantitative trait locus; Musa acuminata ssp. malaccensis; Fusarium wilt; Fusarium oxysporum f. sp. cubense; Tropical Race 4; Subtropical Race 4; marker assisted selection; resistance gene expression; receptor-like kinase; RNAseq
Online: 5 May 2023 (09:51:49 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0177.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
chronic myeloid leukemia; tyrosine kinase inhibitor; adverse drug event; quality of life; second-generation tyrosine kinase inhibitor; nilotinib
Online: 16 August 2019 (08:09:07 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0729.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Gastric cancer; Cyclin-dependent protein kinase; Cluster of differentiation (CD) 47; Prognosis
Online: 31 May 2021 (10:13:20 CEST)
ARTICLE
|
doi:10.20944/preprints201910.0358.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
epithelial-to-mesenchymal transition; TGF-β1; cAMP; A-kinase anchoring protein; Ezrin; AKAP95; Yotiao; cigarette smoke; COPD
Online: 31 October 2019 (02:15:56 CET)
ARTICLE
|
doi:10.20944/preprints202104.0732.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Epidermal Growth Factor Receptor (EGFR); mutations, EGFR tyrosine kinase inhibitor; molecular epidemiology; Non-small-cell lung cancer
Online: 28 April 2021 (07:55:22 CEST)
COMMUNICATION
|
doi:10.20944/preprints202011.0174.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
MZA, Manzamine A; CTKD, C-terminal kinase domain; ras-ERK1/2 (extracellular-signal-regulated kinase 1/2) pathway; RSK1, 90kDa ribosomal protein S6 kinase 1; RSK2, 90kDa ribosomal protein S6 kinase 2; NTKD, N-terminal kinase domain
Online: 4 November 2020 (08:27:07 CET)
ARTICLE
|
doi:10.20944/preprints201905.0145.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Sprouty1; proliferation; tyrosine kinase
Online: 13 May 2019 (08:23:54 CEST)
REVIEW
|
doi:10.20944/preprints202103.0510.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RAF kinase independent; RAS; MST2; ASK; PLK; RHO-α; apoptosis; cell cycle; cancer therapy
Online: 22 March 2021 (10:29:37 CET)
ARTICLE
|
doi:10.20944/preprints202109.0474.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
NELL2; Preproenkephalin; Endoplasmic reticulum; Calcium ion; Protein kinase C; Extracellular signal-regulated kinase (ERK)
Online: 28 September 2021 (13:40:26 CEST)
REVIEW
|
doi:10.20944/preprints202207.0024.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
post-translation modifications; CK2; Huntington’s Disease; Kinase Inhibition; HTT phosphorylation
Online: 1 July 2022 (17:47:10 CEST)
ARTICLE
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
kinase inhibitors; pure drug nanoparticles; drug nanocrystals; bottom-up nanonization; nanoprecipitation; microfluidics; flow focusing technologies
Online: 2 March 2021 (11:29:18 CET)
ARTICLE
|
doi:10.20944/preprints202109.0156.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
circulating thymidine kinase 1; cell loss; biomarker; early treatment response; breast cancer
Online: 8 September 2021 (16:25:39 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0582.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Liquid-based 3D culture; tumoroid; cisplatin resistance; imatinib (gleevec); tyrosine kinase inhibitor (TKI); organoid; spheroid; metastatic colorectal cancer (mCRC)
Online: 23 December 2020 (10:15:46 CET)
COMMUNICATION
|
doi:10.20944/preprints201910.0068.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Frank-Starling; myopathy; Myosin Binding Protein-C; Kinase mechanism
Online: 7 October 2019 (12:15:26 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0297.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Protein Kinase Receptor (PKR); Mammarenavirus; Interferon; Innate immune response; Mx1; ISG15; CCL5
Online: 13 May 2021 (13:27:07 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0393.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
poxviruses; protein kinase R; evolution; translational regulation; eIF2
Online: 30 May 2022 (10:42:41 CEST)
REVIEW
|
doi:10.20944/preprints202107.0353.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Lung cancer; Adjuvant treatment; Non-small-cell lung carcinoma (NSCLC); Epidermal growth factor receptor (EGFR); Tyrosine kinase inhibitor (TKI)
Online: 15 July 2021 (10:16:30 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Kinase Inhibitor; NEK2; Chemoresistance; Avicennia marina; Marine compounds; Molecular docking; Cancer
Online: 7 June 2020 (11:16:35 CEST)
REVIEW
|
doi:10.20944/preprints202106.0609.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Chronic myeloid leukaemia; chronic phase; Tyrosine kinase inhibitor; Treatment free remission; deep molecular response; BCR-ABL.
Online: 25 June 2021 (08:13:40 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202107.0525.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Mucormycosis; AlkB; demethylase; virulence; dimorphism; protein kinase A; hyphae development; Mucor
Online: 23 July 2021 (07:57:16 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0638.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 26 May 2021 (13:14:06 CEST)
REVIEW
|
doi:10.20944/preprints201912.0412.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Frank-Starling; angiotensin receptor; muscle contraction; myosin light chain kinase; Protein Kinase C-βII; myosin light chain phosphatase; β-arrestin; MgATP; MgADP-phosphomyosin; myosin LC affinity for Ca2+
Online: 11 January 2020 (13:24:08 CET)
ARTICLE
|
doi:10.20944/preprints202104.0174.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Phosphodiesterase (PDE); natural products; inhibitors; Protein Kinase; selectivity; fluorescence polarization
Online: 6 April 2021 (12:07:58 CEST)
REVIEW
|
doi:10.20944/preprints202307.0990.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Bruton's tyrosine kinase (BTK); cognitive disorders; multiple sclerosis (MS); Neuroinflammation; immune system
Online: 14 July 2023 (13:24:12 CEST)
REVIEW
|
doi:10.20944/preprints202003.0251.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
gastric acid suppressant; chemotherapy; tyrosine kinase inhibitors; proton pump inhibitors
Online: 31 March 2020 (03:40:46 CEST)
REVIEW
|
doi:10.20944/preprints202304.1236.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
FLT3 mutations; resistant/relapsed acute myeloid leukemia; tyrosine kinase inhibitors; gilteritinib
Online: 29 April 2023 (10:55:21 CEST)
ARTICLE
|
doi:10.20944/preprints202304.1063.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
empagliflozin; vascular calcification; AMP-activated protein kinase; nuclear factor erythroid-2-related factor; heme oxygenase 1; chronic kidney disease
Online: 27 April 2023 (09:35:25 CEST)
REVIEW
|
doi:10.20944/preprints202305.0122.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Non-small cell lung cancer (NSCLC); EGFR; Tyrosine kinase inhibitors (TKIs); Uncommon mutation; Compound mutation; Intracranial activity; Immunotherapy
Online: 3 May 2023 (09:29:08 CEST)
REVIEW
|
doi:10.20944/preprints202307.2046.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CADD; SBDD; LBDD; kinase; small molecule kinase inhibitors
Online: 31 July 2023 (03:05:42 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0542.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
safety analysis; targeted therapy; monoclonal antibody therapy; immune checkpoint inhibibitors; tyrosine kinase inhibitors; breast cancer; gynecological cancer; Helixor; Viscum album L.; PARP inhibitors; CDK 4/6 inhibitors
Online: 30 December 2022 (12:00:35 CET)
ARTICLE
|
doi:10.20944/preprints202111.0108.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Plasmodium; malaria; type III beta phosphatidylinositol 4-kinase; virtual screening; homology modeling; molecular dynamics
Online: 5 November 2021 (08:44:31 CET)
ARTICLE
|
doi:10.20944/preprints202311.1488.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
tuberculosis; statins; host-directed therapy; foam cells; granulomas; NLRP3 inflammasome; mevalonate-kinase deficiencies
Online: 23 November 2023 (08:23:48 CET)
ARTICLE
|
doi:10.20944/preprints202305.0538.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Aging; Betaine; dBHMT; Drosophila; dSAMTOR; dTORC1; Kinase; Methionine; SAM
Online: 8 May 2023 (12:06:37 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 25 January 2021 (15:01:17 CET)
ARTICLE
|
doi:10.20944/preprints202306.0068.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
3D printed scaffolds; carbon nanotube; capped carbon nanotube; protein kinase A; pseudomonas elastase; exotoxin A; alpha-hemolysin; shiga toxin 2a
Online: 5 June 2023 (02:56:10 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0002.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Extracellular calpastatin, Ca2+/ calmodulin (CaM)-dependent protein kinase kinase 2, osteocytes, osteoclasts, bone remodeling
Online: 1 February 2023 (01:11:27 CET)
BRIEF REPORT
|
doi:10.20944/preprints202207.0144.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Protein Kinase C; PKCeta; autophagy; senescence; chemoresistance; oxidative stress; ER stress; 3MA; chloroquine
Online: 10 July 2022 (06:42:23 CEST)
REVIEW
|
doi:10.20944/preprints202306.1643.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
metastasis treatment; small molecules; tyrosine kinase inhibitors; integrins; siRNA
Online: 22 June 2023 (16:10:15 CEST)
REVIEW
|
doi:10.20944/preprints202306.0143.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Systemic sclerosis; treatment; Janus kinase inhibitors; fibrosis; anti-cytokine treatment
Online: 2 June 2023 (07:07:00 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1297.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Heart failure; β-adrenergic receptor; cardiac fibrosis; cardiac inflammation; Bruton’s tyrosine kinase; Zanubrutinib
Online: 19 June 2023 (05:23:12 CEST)
REVIEW
|
doi:10.20944/preprints202305.0606.v1
Subject:
Medicine And Pharmacology,
Anatomy And Physiology
Keywords:
alcoholic fatty liver; adenosine monophosphate activated kinase; sterol regulatory element binding protein 1c; peroxisome proliferator activated receptor , oxidative stress; cytochrome P450 2E1
Online: 9 May 2023 (08:38:13 CEST)
REVIEW
|
doi:10.20944/preprints202309.1260.v1
Subject:
Medicine And Pharmacology,
Pediatrics, Perinatology And Child Health
Keywords:
PANDAS; Pediatric Autoimmune Neuropsychiatric Disorders Associated with Streptococcal Infections; PANDAS syndrome; neuropsychiatric disorder; streptococci; molecular mimicry; CaM kinase; striatal cholinergic interneurons; obsessive-compulsive disorder; streptococcal infection; tic; tics
Online: 19 September 2023 (07:09:19 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1201.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Methicillin-resistant Staphylococcus aureus; poly-amidoamine dendrimers (PAMAM); anti-virulence agent, accessory gene regulator; histidine kinase inhibitor.
Online: 16 August 2023 (20:32:54 CEST)
REVIEW
|
doi:10.20944/preprints202402.1356.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
DNA replication; origin of replication; initiation; replication fork; Okazaki fragment; DNA damage signalling; ATR kinase; telomeres
Online: 23 February 2024 (09:33:26 CET)
REVIEW
|
doi:10.20944/preprints202403.0254.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
dichloroacetate; cancer; lactic acidosis; glioma; pyruvate dehydrogenase kinase; pyruvate dehydrogenase; pyruvate dehydrogenase phosphatase
Online: 5 March 2024 (13:03:15 CET)
REVIEW
|
doi:10.20944/preprints202311.0094.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Casein Kinase II; Musculoskeletal; Osteoarthritis; Osteoporosis; CX-4945; CIBG-300; Cell Signaling; Drug Development; Targeted therapy
Online: 1 November 2023 (13:18:42 CET)
REVIEW
|
doi:10.20944/preprints202305.1789.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PTK6; Colorectal cancer; Tyrosine Kinase Inhibitors
Online: 25 May 2023 (09:52:24 CEST)
REVIEW
|
doi:10.20944/preprints202308.0444.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Avenanthramide; AKT-Protein kinase B; Alzheimer's disease; Parkinson's disease; oxidative stress; neuroprotection
Online: 7 August 2023 (02:28:52 CEST)
REVIEW
|
doi:10.20944/preprints202307.0539.v3
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Hepatocellular carcinoma; tyrosine kinase inhibitors; immune checkpoint inhibitors; biomarkers
Online: 17 July 2023 (13:22:33 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0522.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Rabson-Mendenhall syndrome; insulin resistance; diabetes mellitus; acanthosis nigricans; tyrosine kinase; insulin; Insulin receptor; INSR
Online: 8 November 2023 (07:35:08 CET)
REVIEW
|
doi:10.20944/preprints202401.0297.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
dual leucine zipper kinase; phosphorylation; protein-protein interaction; proteasomal degradation; palmitoylation
Online: 4 January 2024 (09:32:03 CET)
ARTICLE
|
doi:10.20944/preprints202309.1199.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
protein-protein interaction; fragment molecular orbital method; polo-like kinase 1; molecular dynamics simulation
Online: 19 September 2023 (03:58:32 CEST)
REVIEW
|
doi:10.20944/preprints202312.0095.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Eosinophilia,; hematological neoplasm; myeloid/lymphoid neoplasm with eosinophilia; tyrosine kinase fusion genes; acute leukemia
Online: 1 December 2023 (16:34:12 CET)
REVIEW
|
doi:10.20944/preprints202309.1526.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
neurodegeneration with brain iron accumulation (NBIA); pantothenate kinaseassociated neurodegeneration (PKAN); pantothenate kinase 2 (PANK2); pantothenate; pantethine; vitamin E; omega 3; -lipoic acid; L-carnitine; thiamine; fibroblasts; induced neurons; precision medicine
Online: 22 September 2023 (09:18:39 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1059.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
corneal enendothelial dystrophy; Slc4a11; barrier function; lactate transporters; Src kinase; oxidative stress; Visomitin
Online: 15 May 2023 (15:50:03 CEST)
REVIEW
|
doi:10.20944/preprints202312.1057.v1
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
cardiotonic steroids; endogenous cardiotonic steroids; ouabain; blood; blood cells; red blood cells; Na,K-ATPase; Src-kinase; signalling cascades; immunogenic effects
Online: 14 December 2023 (06:14:30 CET)