ARTICLE
|
doi:10.20944/preprints202005.0057.v2
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; treatment; drug; survival; antiviral; hydroxychloroquine
Online: 9 May 2020 (04:45:37 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0544.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
Bodybuilding; Drug Free; Competing; Peaking; Carbohydrate Loading; Water Loading; Sodium Loading; Fat Loading: Vitamin C; Fibre Restriction
Online: 27 September 2018 (12:58:34 CEST)
REVIEW
|
doi:10.20944/preprints202012.0452.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RNA; self-amplifying RNA; replicon; vaccine; drug delivery
Online: 18 December 2020 (11:12:44 CET)
ARTICLE
|
doi:10.20944/preprints202003.0349.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
novel coronavirus; COVID-19; protease; molecular docking; drug designing; ADME; drug repurposing
Online: 23 March 2020 (09:47:49 CET)
REVIEW
|
doi:10.20944/preprints202012.0242.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; SARS-CoV-2; long-haul; inflammation; tissue damage; drug repurposing
Online: 10 December 2020 (09:42:20 CET)
COMMUNICATION
|
doi:10.20944/preprints202002.0418.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
virtual screening; molecular docking; drug repurposing; drug repositioning; anti-viral drugs; Coronavirus; COVID-19; 2019-nCoV; SARS-CoV-2
Online: 9 March 2020 (02:29:04 CET)
REVIEW
|
doi:10.20944/preprints202012.0062.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Trop 2; targeted therapy; antibody-drug conjugate; solid tumors
Online: 2 December 2020 (12:35:36 CET)
REVIEW
|
doi:10.20944/preprints202010.0179.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Non Michaelis-Menten Kinetics; High-throughput screening; allostery; cooperativity; processive kinetics; distributive kinetics; single-molecule; auto-catalytic; drug discovery
Online: 8 October 2020 (13:34:16 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0360.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SARS-CoV-2; transcriptional inhibition; COVID-19; drug repurposing; TMPRSS2
Online: 28 April 2020 (09:39:02 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0061.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Coronavirus; Deep learning; Drug screening; homology modeling; main protease
Online: 5 February 2020 (10:59:09 CET)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
ARTICLE
|
doi:10.20944/preprints202003.0440.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; SARS-CoV-2; 2019-nCoV; novel corona virus; drug repurposing; chloroquine; high-risk group; asymptomatic
Online: 30 March 2020 (07:24:16 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0071.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
2019-nCoV; novel corona virus; Wuhan virus; drug; vaccine; spike protein; epitope; vaccine design
Online: 5 February 2020 (15:34:15 CET)
ARTICLE
|
doi:10.20944/preprints202003.0413.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
coronavirus; drug; COVID-19; SARS; MERS; ontology; ChEBI; NDF-RT; DrON; bioinformatics
Online: 29 March 2020 (01:58:40 CET)
REVIEW
|
doi:10.20944/preprints201812.0170.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
bacterial nanocellulose; nanofibrillated nanocellulose; animal nanocellulose; algal nanocellulose; tissue engineering; tissue repair; wound dressing; cell delivery; drug delivery; antimicrobial properties
Online: 14 December 2018 (06:44:53 CET)
REVIEW
|
doi:10.20944/preprints202005.0376.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus bioinformatics; SARS-CoV-2; sequencing; epidemiology; drug design; tools
Online: 23 May 2020 (11:01:11 CEST)
REVIEW
|
doi:10.20944/preprints202004.0122.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
melatonin; coronavirus; pandemic; SARS-CoV-2; bat; lung; apoptosis; programmed cell death; mortality; morbidity; COVID-19; drug
Online: 9 April 2020 (09:24:47 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
ARTICLE
|
doi:10.20944/preprints201608.0162.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
bacterial ghosts (BGs); Vibrio parahaemolyticus; chemically induced lysis; minimum inhibition concentration (MIC); sodium hydroxide (NaOH); lipopolysaccharides (LPS); endotoxic activity; macrophages; cytotoxicity; cytokine
Online: 17 August 2016 (10:26:00 CEST)
REVIEW
|
doi:10.20944/preprints202008.0312.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
SARS-CoV-2(COVID-19); + ssRNA; ribosomal – framshift; Pseudoknot; replication; model; drug; vaccine
Online: 14 August 2020 (08:26:31 CEST)
REVIEW
|
doi:10.20944/preprints202105.0311.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Angiotensin converting enzyme 2; breast feeding; drug therapy; pregnancy; severe acute respiratory syndrome coronavirus 2
Online: 13 May 2021 (15:26:34 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0157.v1
Subject:
Business, Economics And Management,
Accounting And Taxation
Keywords:
National Centralized Drug Procurement; "4+7" policy; drug price; interrupted time series; volume-based procurement.
Online: 6 April 2021 (08:18:10 CEST)
REVIEW
|
doi:10.20944/preprints201807.0233.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
nanocrystals; poorly soluble drug; nanotechnology; stability
Online: 13 July 2018 (11:16:15 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0224.v2
Subject:
Engineering,
Marine Engineering
Keywords:
propeller; cavitation pattern; unsteady cavitation; induced pressure fluctuations; high-speed visualization; volume acceleration; cavitation-pressure correlations
Online: 5 September 2016 (09:37:05 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
monoglyceride colloidal liquid crystals; release profile; mathematical models; drug delivery systems; release kinetic; square root laws
Online: 17 September 2018 (09:33:52 CEST)
ARTICLE
|
doi:10.20944/preprints201906.0069.v1
Subject:
Engineering,
Mechanical Engineering
Keywords:
winglets; lift-induced drag; wing tip device; non-planar lifting surface; performance optimization; aircraft performance; regional aircraft
Online: 9 June 2019 (03:48:26 CEST)
REVIEW
|
doi:10.20944/preprints201703.0125.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
Extracellular vesicles (EVs); Peptidylarginine deiminases (PADs); Chlor-amidine (Cl-Am); cancer; neurodegeneration; deimination; cytoskeleton; induced pluripotent stem cells (iPSCs); histone H3; epigenetics
Online: 16 March 2017 (17:54:15 CET)
REVIEW
|
doi:10.20944/preprints202112.0315.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Nanotechnology; Niosomes; Targeted Drug Delivery
Online: 20 December 2021 (14:18:53 CET)
REVIEW
|
doi:10.20944/preprints202102.0265.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Peptides; Clinical Practice; Drug Therapy; Therapeutic
Online: 10 February 2021 (15:51:13 CET)
ARTICLE
|
doi:10.20944/preprints202102.0280.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Double stranded RNA; Nano clay; Phytophthora infestans; Potato; Spray Induced gene silencing (SIGS)
Online: 11 February 2021 (11:07:19 CET)
ARTICLE
|
doi:10.20944/preprints201701.0095.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
polymeric composite; surface initiated atom transfer radical polymerization; photo-induced; living radical polymerization; metal-free atom transfer radical polymerization
Online: 22 January 2017 (04:56:44 CET)
ARTICLE
|
doi:10.20944/preprints201801.0278.v1
Subject:
Arts And Humanities,
Humanities
Keywords:
resettlement; psychological risks; development-induced displacement
Online: 30 January 2018 (06:48:20 CET)
REVIEW
|
doi:10.20944/preprints201805.0426.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
biological activity; crosslinking; drug delivery; cosmetic; food-supplement; functionalization; hyaluronan applications; hyaluronan derivatives; hyaluronan synthases; hyaluronic acid; hyaluronidases; physico-chemical properties
Online: 29 May 2018 (12:13:48 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0393.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV2; RNA depended RNA polymerase; Valproic acid Co-A; drug repurposing
Online: 26 March 2020 (15:04:22 CET)
ARTICLE
|
doi:10.20944/preprints202107.0229.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
HPLC; NSAIDs; Isocratic; Short column; Drug mixture
Online: 9 July 2021 (15:23:57 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0075.v3
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
azithromycin; HPLC; robust; isocratic; drug stability; degradation products
Online: 4 January 2017 (10:08:52 CET)
REVIEW
|
doi:10.20944/preprints202007.0108.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
COVID-19; SARS-CoV-2; coronavirus; hypothesis; pathophysiology; drug repurposing
Online: 7 July 2020 (02:50:55 CEST)
REVIEW
|
doi:10.20944/preprints202101.0503.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
CNS; Drug receptors; GABA; Cannabinoid; Opioid; Serotonin; Dopamine
Online: 25 January 2021 (14:15:20 CET)
REVIEW
|
doi:10.20944/preprints202005.0234.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
SIRD; Twitter; GHSI; Pre-symptomatic; EHR; Contact tracing; On-line survey; qRT-PCR; X-ray; CT/HRCT; CNN; Autoencoder; Drug affinity; CPI; and Inflation.
Online: 14 May 2020 (11:25:57 CEST)
ARTICLE
|
doi:10.20944/preprints202203.0117.v3
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
active pharmaceutical ingredient; compounded drug; compounding; extemporaneous formulation; manufactured material; medication; monograph; pediatric; reference standards
Online: 5 April 2022 (10:17:10 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0025.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
drug repurposing; translational bioinformatics; transcriptomics; transcriptome analysis; drug discovery; protocol; gene expression
Online: 9 October 2016 (08:42:23 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0026.v1
Subject:
Environmental And Earth Sciences,
Geophysics And Geology
Keywords:
seismic hazard; openquake; GMPE; basin-induced amplification; SPECFEM2D
Online: 4 January 2018 (10:04:35 CET)
CASE REPORT
|
doi:10.20944/preprints202012.0596.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Covid-19, SARS-CoV-2, drug repurposing
Online: 23 December 2020 (15:58:38 CET)
REVIEW
|
doi:10.20944/preprints202104.0652.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Enzymatic reaction; crosslinking; Hydrogel; Biomedical application; Tissue engineering; Wound healing; Drug delivery
Online: 26 April 2021 (10:52:24 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0023.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
gelatin-oleic conjugate; self-assembled biodegradable nanoparticles; biomimetic shear stress; cell dynamic environment; cellular drug delivery; paclitaxel
Online: 4 April 2017 (10:59:02 CEST)
REVIEW
|
doi:10.20944/preprints202105.0567.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Artificial intelligence AI; machine learning; algorithms; QSAR; drug discovery
Online: 24 May 2021 (13:02:21 CEST)
REVIEW
|
doi:10.20944/preprints201807.0241.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
biomaterial; bone regeneration; drug release; hydrogel; lignin; multivariate data processing; osteogenesis; scaffolds; stem cells; tissue engineering
Online: 13 July 2018 (15:07:37 CEST)
REVIEW
|
doi:10.20944/preprints201905.0130.v1
Subject:
Biology And Life Sciences,
Plant Sciences
Keywords:
induced mutagenesis; fast neutron irradiation; mutation mapping; deletagene; next-generation sequencing technologies; reverse genetics
Online: 10 May 2019 (14:38:21 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0083.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
stroke; antioxidant; co-drug; animal model
Online: 20 October 2016 (08:46:38 CEST)
ARTICLE
|
doi:10.20944/preprints201705.0174.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
steroid; metabolism; anti-inflammatory drug; inhibition
Online: 24 May 2017 (08:25:26 CEST)
REVIEW
|
doi:10.20944/preprints201705.0129.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
cell fate decision; cancer attractors; gene network dynamics; EMT; drug resistance; intrinsically disordered proteins
Online: 17 May 2017 (06:25:17 CEST)
REVIEW
|
doi:10.20944/preprints202105.0346.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
drug discovery; drug repurposing; bioinformatics; machine learning; artificial intelligence; biomedical discoveries etc.
Online: 14 May 2021 (15:17:50 CEST)
REVIEW
|
doi:10.20944/preprints201702.0036.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
pulmonary arterial hypertension; prostacyclin; nanoparticle; drug delivery system
Online: 13 February 2017 (09:27:09 CET)
ARTICLE
|
doi:10.20944/preprints202101.0490.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
CD44; Cancer Stem Cells; Tumorigenesis; Drug Resistance; Immune Markers; Epithelial to Mesenchymal Transition; Therapeutic Targeting
Online: 25 January 2021 (12:23:49 CET)
ARTICLE
|
doi:10.20944/preprints201804.0310.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
primary open angle glaucoma; dorzolamide/timolol fixed combination; drug efficacy; safety
Online: 24 April 2018 (08:36:58 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0003.v1
Subject:
Physical Sciences,
Atomic And Molecular Physics
Keywords:
laser-induced plasma; stark broadening; electron density; nanomaterial; atomic spectroscopy; silver; hydrogen
Online: 1 August 2018 (08:02:03 CEST)
REVIEW
|
doi:10.20944/preprints201711.0015.v1
Subject:
Biology And Life Sciences,
Plant Sciences
Keywords:
RGSV; movement proteins; gene silencing; transgenic mechanism; virus-induced small interfering RNA; RNA silencing pathway; antiviral plant defenses
Online: 2 November 2017 (03:05:04 CET)
ARTICLE
|
doi:10.20944/preprints201810.0490.v1
Subject:
Computer Science And Mathematics,
Computer Vision And Graphics
Keywords:
drug release simulation; disintegration simulation; poorly water soluble drug; mefenamic acid; Noyes-Whitney equation; cellular automata; synchrotron microtomography
Online: 22 October 2018 (11:38:04 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0108.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
contrast induced nephropath; acute myocardial infarction
Online: 21 November 2016 (12:13:30 CET)
ARTICLE
|
doi:10.20944/preprints202005.0199.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SARS-CoV-2; COVID-19; CADD; virtual screening; approved drugs; drug repurposing; essential targets; molecular docking; molecular dynamics simulations
Online: 11 May 2020 (13:14:18 CEST)
ARTICLE
|
doi:10.20944/preprints201709.0102.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
drug screening; bone mineralization; osteoclast; zebrafish
Online: 21 September 2017 (06:34:11 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0132.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
arylamine N-acetyltransferases; cancer; tuberculosis; drug discovery; traditional Chinese medicine; virtual screening; molecular dynamics simulation; MM-PBSA
Online: 30 June 2017 (11:36:22 CEST)
REVIEW
|
doi:10.20944/preprints202003.0345.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; lysosomotropic agents; endosome; antiviral; drug repurposing
Online: 24 March 2020 (06:26:54 CET)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0170.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Spreading parameter; Cellular proliferation; Drug sensitivity; Substrates; Cancer cells
Online: 26 April 2017 (17:38:07 CEST)
REVIEW
|
doi:10.20944/preprints202005.0342.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
seaweed; metabolites; neuroprotection; Alzheimer’s disease; Parkinson’s disease; ischemic stroke; computer-aided drug discovery
Online: 21 May 2020 (09:49:29 CEST)
ARTICLE
|
doi:10.20944/preprints201704.0028.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
lanthanides; fluorapatite; drug loading; nano carrier
Online: 5 April 2017 (11:26:48 CEST)
REVIEW
|
doi:10.20944/preprints202305.1084.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
antibody-drug conjugate; lysosome; cathepsin; legumain; self-immolation; payload release; peptidomimetic; linker
Online: 16 May 2023 (04:51:34 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0297.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
lignin; drug release; paracetamol; disintegration
Online: 24 May 2019 (12:40:01 CEST)
REVIEW
|
doi:10.20944/preprints202001.0324.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
natural products; sirtuin; drug discovery; epigenetics; structure–activity relationship
Online: 27 January 2020 (09:21:29 CET)
REVIEW
|
doi:10.20944/preprints201804.0126.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
pharmaceutical market; drugs; drug discovery; solid-phase peptide synthesis
Online: 10 April 2018 (10:14:33 CEST)
REVIEW
|
doi:10.20944/preprints202006.0232.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Adverse drug reactions; Anti-COVID drugs; Coronavirus; Drug repurposing; Drug toxicity; Pharmacotherapy
Online: 18 June 2020 (12:43:43 CEST)
REVIEW
|
doi:10.20944/preprints201805.0011.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
computational drug repositioning; drug repositioning; drug repurposing; machine learning; deep learning; crowdsourcing; open innovation; drug discovery
Online: 1 May 2018 (12:27:22 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0283.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Adverse drug reaction; COVID-19 treatment
Online: 12 August 2020 (11:12:41 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0447.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
spike protein; SARS-CoV-2; mutation; drug repurposing; digitoxin
Online: 20 August 2020 (08:24:41 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0459.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; coronavirus; drug repositioning; pathway enrichment
Online: 19 September 2020 (11:34:12 CEST)
ARTICLE
|
doi:10.20944/preprints202006.0358.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Enzyme inhibition; Secondary Metabolites; In-silico Analysis; Molecular docking; Drug candidates
Online: 30 June 2020 (08:11:28 CEST)
REVIEW
|
doi:10.20944/preprints201807.0143.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
Aromatic hydroxy metabolites; arenolic drug metabolites; metabolic O-dealkylation; metabolic aromatic ring hydroxylation; primary and auxiliary pharmacophores; auxophores; metabolic modification of drug activity
Online: 9 July 2018 (13:28:16 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0319.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
adverse drug reactions; spontaneous reporting; causality; ADR; severity
Online: 18 August 2018 (05:17:05 CEST)
REVIEW
|
doi:10.20944/preprints202008.0320.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Data Science; Machine Learning; Deep Learning; Genomics; COVID-19; Drug Discovery; Image Analysis; Interactomics; Epidemiology
Online: 14 August 2020 (11:01:56 CEST)
REVIEW
|
doi:10.20944/preprints201807.0226.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
galvanic replacement; photothermal therapy; drug delivery; nanoparticles; cancer treatment
Online: 13 July 2018 (05:11:21 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0466.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
COVID-19; coronavirus; ACE2; bioinformatics analysis; drug prediction
Online: 26 April 2020 (03:14:50 CEST)
REVIEW
|
doi:10.20944/preprints201812.0032.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cannabis; cannabinoids; THC; CBD, drug-drug interactions; pharmacokinetic; cytochrome P450; UDP- glucuronosyltransferases; glucoprotein-P
Online: 3 December 2018 (16:07:43 CET)
REVIEW
|
doi:10.20944/preprints201910.0296.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
nasal delivery; glioblastoma multiforme; drug delivery; nanoparticles; nose-to-brain delivery; pre-clinical studies; clinical evaluation
Online: 27 October 2019 (09:36:27 CET)
ARTICLE
|
doi:10.20944/preprints201801.0204.v1
Subject:
Chemistry And Materials Science,
Metals, Alloys And Metallurgy
Keywords:
metastable Ti alloy; high temperature deformation; stress-induced ω; stress-induced α˝ martensite; transmission electron microscopy; slip; X-ray diffraction.
Online: 22 January 2018 (17:17:03 CET)
REVIEW
|
doi:10.20944/preprints202108.0558.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
chitosan; chitin; biological activit; drug delivery; antioxidant; antimicrobial; biocatalysis; nanoparticles
Online: 31 August 2021 (11:07:28 CEST)
REVIEW
|
doi:10.20944/preprints201709.0050.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's-disease; dementia; drug targeting; nanoemulsion; neuroinflammation; oxidative stress; scavenger receptors; sonoporation; transcranial ultrasound
Online: 13 September 2017 (05:44:29 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Covid-19; proteins; normal-modes; protein-drug interactions; chloroquine; ivermectin; remdesivir; sofosbuvir; boceprevir; α-difluoromethylornithine (DMFO)
Online: 11 August 2020 (04:09:43 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0279.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Blood-Brain Barrier, Penetrating Peptides, Machine learning techniques, Drug delivery, Therapeutic peptides
Online: 10 June 2021 (08:13:15 CEST)
REVIEW
|
doi:10.20944/preprints201808.0155.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
amyloid diseases; biocomputing; drug design; natural antiamyloids
Online: 8 August 2018 (04:27:10 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
humans; infection control; therapy; coronavirus; immunoglobulins; drug therapy; therapeutic use; corticosteroid
Online: 8 March 2020 (17:04:19 CET)
REVIEW
|
doi:10.20944/preprints202203.0071.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
rheumatoid arthritis; precision medicine; new treatment; drug development; method development
Online: 25 May 2022 (04:59:01 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0087.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Mongolian oak cups; ethanol crude extract (ECE); ellagic acid- and kaempferol-derivatives; alloxan-induced rats; type 1 diabetes; hypoglycemic effect
Online: 8 April 2018 (08:45:39 CEST)
REVIEW
|
doi:10.20944/preprints202004.0395.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
coronavirus disease 2019; chloroquine; drug repurposing; HIV; Africa
Online: 22 April 2020 (08:33:34 CEST)
REVIEW
|
doi:10.20944/preprints201810.0577.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
myeloma; daratumumab; elotuzumab; isatuximab; CD38; JNJ- 63723283; denosumab; checkpoint inhibitors; BCMA; bispecific T-cell engager; antibody-drug conjugates
Online: 24 October 2018 (12:11:23 CEST)
REVIEW
|
doi:10.20944/preprints201910.0144.v6
Subject:
Biology And Life Sciences,
Virology
Keywords:
virus; antiviral drug; drug discovery; drug development; broad-spectrum antivirals
Online: 14 February 2020 (02:27:24 CET)
ARTICLE
|
doi:10.20944/preprints201811.0561.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cheminformatics, drugs, drug-likeness, drug discovery, natural products
Online: 23 November 2018 (13:56:32 CET)
REVIEW
|
doi:10.20944/preprints201810.0507.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
liposomes, exosomes, extracellular vesicles, drug delivery, drug targeting, bioinspired systems, engineered systems.
Online: 22 October 2018 (15:35:20 CEST)
ARTICLE
|
doi:10.20944/preprints201907.0001.v1
Subject:
Engineering,
Aerospace Engineering
Keywords:
Variable cant angle; Winglets; Drag reduction; Lift-induced drag; CFD
Online: 1 July 2019 (11:02:29 CEST)