BRIEF REPORT
|
doi:10.20944/preprints202002.0242.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; molecular docking; HIV protease inhibitor; nucleotide analogues
Online: 29 February 2020 (12:43:40 CET)
ARTICLE
|
doi:10.20944/preprints202002.0438.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Simeprevir; Protease inhibitor; Virtual screening; Docking
Online: 28 February 2020 (13:14:38 CET)
ARTICLE
|
doi:10.20944/preprints202003.0347.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
nsp12; RNA-dependent-RNA polymerase; SARS-CoV-2; inhibitor; vitamin B12
Online: 23 March 2020 (07:46:54 CET)
ARTICLE
|
doi:10.20944/preprints202003.0024.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
SARS-CoV-2; nonstructural proteins (NSP); NSP12; NSP7; NSP8; virtual screening; inhibitor
Online: 2 March 2020 (03:11:33 CET)
REVIEW
|
doi:10.20944/preprints201707.0019.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
affective disorders; alzheimer’s disease; l-Deprenyl (Selegiline); donepezil; galantamine; value; inhibitor constant; mechanism-based inhibition; multitarget-directed ligand (MTDL); rasagiline; rivastigmine
Online: 11 July 2017 (05:58:53 CEST)
HYPOTHESIS
|
doi:10.20944/preprints202004.0180.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
COVID-19; prostaglandins; mPGES1 inhibitor; ARDS; sonlicromanol; KH176
Online: 12 April 2020 (04:36:48 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0122.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cancer; FGFR; Inhibitor; 4‐Substituted‐1H‐indazole
Online: 29 September 2016 (15:42:08 CEST)
REVIEW
|
doi:10.20944/preprints201610.0100.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
BET; bromodomain; histone acetylation; gene transcription; BET inhibitor
Online: 24 October 2016 (05:06:56 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0591.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
adverse events; immune checkpoint inhibitor; myasthenia gravis; myopathy; neuropathy; nivolumab; pembrolizumab
Online: 29 September 2018 (11:28:00 CEST)
REVIEW
|
doi:10.20944/preprints201703.0148.v1
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
microcystin; saxitoxin; cylindrospermopsin; anatoxin-a; anatoxin-a(S); cyanobacteria; organic anion transporting polypeptide; phosphatase inhibitor; acetylcholinesterase; neurotoxicity; water quality; eutrophication; drinking water
Online: 20 March 2017 (06:17:48 CET)
REVIEW
|
doi:10.20944/preprints201705.0127.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Cholangiocarcinoma; DNA methylation; Tumor suppressor gene; microRNA; DNA methylation inhibitor
Online: 16 May 2017 (18:08:59 CEST)
TECHNICAL NOTE
|
doi:10.20944/preprints201706.0085.v1
Subject:
Engineering,
Civil Engineering
Keywords:
finite element modeling; electrochemical chloride extraction (ECE); electrical injection of corrosion inhibitor (EICI); rebar corrosion; repair mortar
Online: 19 June 2017 (13:40:09 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; SARS-CoV-2; 3CLpro; PLpro; RdRp; AAK1; inhibitor; dock; molecular dynamics
Online: 15 March 2020 (02:34:14 CET)
ARTICLE
|
doi:10.20944/preprints202004.0084.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
in silico repositioning; dual inhibitor; Covid-19; 3CLpro; PLpro; remdesivir
Online: 7 April 2020 (10:44:11 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0211.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Metalloproteinase; phenanthroline; metalloproteinase inhibitor; zebrafish; aryl hydrocarbon receptor; poly aromatic hydrocarbon toxicity; angiogenesis; neural crest; in vivo study
Online: 26 August 2016 (11:19:51 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0215.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
FGFR1; inhibitor; kinase inhibitor; pyrazine; hinge binder
Online: 30 March 2017 (04:13:45 CEST)
ARTICLE
|
doi:10.20944/preprints201709.0070.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Coumarin; Mycobacterium tuberculosis; Cholinesterase inhibitor; Monoamine oxidase B inhibitor; Structure activity relationship; Albumin binding, Neuroprotection
Online: 15 September 2017 (17:34:38 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0177.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Ebola; influenza virus; HIV; envelope protein; membrane fusion inhibitor; HR2; pentacyclic triterpenoids
Online: 19 January 2018 (04:02:15 CET)
SHORT NOTE
|
doi:10.20944/preprints201707.0096.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
corrosion inhibitor; coumarin; resonance
Online: 31 July 2017 (16:37:19 CEST)
ARTICLE
|
doi:10.20944/preprints201708.0021.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
3-((2-chlorobenzylidene)amino)coumarin; corrosion inhibitor; damage reduction
Online: 7 August 2017 (10:51:42 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0180.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
primary Sjögren's syndrome; alpha-1-antitrypsin; inhibitor; 4-hydroxy-2-nonenal; autoantibody isotypes; serum
Online: 30 October 2017 (04:30:59 CET)
ARTICLE
|
doi:10.20944/preprints201710.0127.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
WNT pathway; porcupine inhibitor ETC-1922159; sensitivity analysis; colorectal cancer; unknown biological hypotheses; combinatorial search space; support vector ranking
Online: 18 October 2017 (05:58:17 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0053.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
1,10-Phenanthroline-5,6-diamine; corrosion inhibitor; weight loss method
Online: 8 January 2018 (09:08:46 CET)
ARTICLE
|
doi:10.20944/preprints201805.0088.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
p53; proteasome inhibitor; endometrial cancer; ovarian cancer; gain-of-function mutation
Online: 4 May 2018 (09:03:27 CEST)
CASE REPORT
|
doi:10.20944/preprints201801.0227.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
Lactate dehydrogenase (LDH), Computed Tomography (CT), Glomerular filtration rate (GFR), C reactive protein (CRP), Angiotensin converting enzyme inhibitor (ACEI) Angiotensin receptor blocker (ARB), Kidney Urinary bladder ( KUB), Dimercapto Succinic Acid (DMSA)
Online: 24 January 2018 (11:41:15 CET)
ARTICLE
|
doi:10.20944/preprints201908.0134.v1
Subject:
Chemistry And Materials Science,
Electrochemistry
Keywords:
aluminium alloy; corrosion inhibitor; alkaline environment; impedance analysis; adsorption; dihydroxybenzene
Online: 12 August 2019 (03:58:57 CEST)
REVIEW
|
doi:10.20944/preprints202007.0314.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
hepatic fibrosis; Mac-2 binding protein glycated isomer; apoptosis inhibitor of macrophage; patatin-like phospholipase domain-containing protein 3; α-fetoprotein; PIVKA-II
Online: 14 July 2020 (13:55:16 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0123.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Snake venomics; Viperidae; Protobothrops flavoviridis; Habu pit viper; Bottom-Up; Top-Down; BPP; Tripeptide metalloprotease inhibitor; Cytotoxicity
Online: 6 July 2018 (16:34:48 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0008.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
WNT pathway; porcupine inhibitor ETC-1922159; sensitivity analysis; colorectal cancer; unknown biological hypotheses; combinatorial search space; support vector ranking; DNA repair and genomic stability factor RAD51
Online: 1 November 2017 (05:08:04 CET)
ARTICLE
|
doi:10.20944/preprints201802.0026.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pig eye perfusion model; pigmentary glaucoma; ocular hypertension; ocular hypotension; phagocytosis; rho-kinase inhibitor
Online: 5 February 2018 (03:39:57 CET)
ARTICLE
|
doi:10.20944/preprints201709.0061.v2
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
expired drug; corrosion inhibitor; potentiodynamic polarization; electrochemical impedance spectroscopy; AFM
Online: 17 October 2017 (04:18:30 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0314.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
MELK inhibitor; OTS167; LC-MS/MS; Pharmacokinetics, mouse serum
Online: 17 August 2018 (15:15:12 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints201804.0358.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
snakebite; antidote; inhibitor; small molecule therapeutics; SMT; secretory phospholipase; sPLA2; Neglected Tropical Disease; NTD
Online: 27 April 2018 (09:00:55 CEST)
COMMENTARY
|
doi:10.3390/sci2030070
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
small molecule inhibitor; personalized medicine; precision medicine; oncology; targeted therapy; drug delivery; drug screening; chemotherapy
Online: 8 September 2020 (00:00:00 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0065.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
hypothalamus; insulin resistance; inflammation; docosahexaenoic acid; PI3K inhibitor; AKT
Online: 4 July 2018 (09:58:03 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0131.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pigmentary glaucoma; ROCK kinase inhibitor; RKI-1447; trabecular meshwork; phagocytosis; cytoskeleton
Online: 9 July 2018 (11:27:28 CEST)
REVIEW
|
doi:10.20944/preprints202106.0176.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
chronic hepatitis B; covalently closed circular DNA; viral integration; transcription factor; nuclear receptor; transcriptional inhibitor; RNA interference
Online: 7 June 2021 (12:43:06 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0374.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
STAT3 as a drug target; cyclic STAT3 decoy; oligodeoxynucleotide inhibitor; head and neck cancer
Online: 29 April 2018 (10:10:00 CEST)
REVIEW
|
doi:10.20944/preprints202101.0393.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Breast cancer; Angiogenesis; Lymphangiogenesis; Cancer Stem cells, microRNA; EP4 receptor; Immune check-point inhibitor
Online: 19 January 2021 (17:40:53 CET)
ARTICLE
|
doi:10.20944/preprints201803.0144.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
sea anemone; drug discovery; cancer; antiangiogenic; endothelial cells; RGD motif; Kunitz type inhibitor
Online: 19 March 2018 (08:15:38 CET)
ARTICLE
|
doi:10.20944/preprints202009.0382.v1
Subject:
Social Sciences,
Behavior Sciences
Keywords:
donepezil; acetylcholinesterase inhibitor; dementia; zebrafish; behavior
Online: 17 September 2020 (07:41:35 CEST)
REVIEW
|
doi:10.20944/preprints201807.0254.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
endocrine disruptor, environmental health sciences, gene-environment, inhibitor of differentiation, neurocognitive disorders
Online: 14 July 2018 (23:30:36 CEST)
REVIEW
|
doi:10.20944/preprints201804.0359.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
oncolytic virus; in situ autovaccination; cytokine; immune checkpoint inhibitor; immune co-stimulator
Online: 27 April 2018 (09:18:37 CEST)
REVIEW
|
doi:10.20944/preprints201909.0120.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Lysophosphatidic acid; Autotaxin; inhibitor; allosteric; orthosteric; lipid chaperone; signalling, GPCR
Online: 11 September 2019 (13:18:21 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ALK5 inhibitor; TGF-β; kinase assay; selectivity; docking
Online: 30 August 2018 (05:52:08 CEST)
REVIEW
|
doi:10.20944/preprints202001.0030.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
histone deacetylase 6 inhibitor; personalized treatment; heat shock protein 90α; leukemia stem cells; imatinib resistance; targeted therapy
Online: 4 January 2020 (06:18:22 CET)
CASE REPORT
|
doi:10.20944/preprints202311.1692.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
mavacamten; cardiac myosin inhibitor; hypertrophic cardiomyopathy; heart failure
Online: 27 November 2023 (11:50:17 CET)
ARTICLE
|
doi:10.20944/preprints202002.0124.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
glycemic variability; continuous glucose monitoring; dipeptidyl Peptidase-4 inhibitor; metformin
Online: 10 February 2020 (10:06:31 CET)
REVIEW
|
doi:10.20944/preprints201809.0281.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
axon guidance; growth cone; cytoskeleton; caspases; apoptosis; signal integration; basal level of caspase activity; death associated inhibitor of apoptosis; axon branching; Netrin; DCC; frazzled; slit; robo; Drosophila
Online: 16 September 2018 (09:43:52 CEST)
REVIEW
|
doi:10.20944/preprints201811.0179.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
calorie restriction mimetics; anti-aging; lifespan extension; glucose metabolism modulation; chitosan; acarbose; SGLT2 inhibitor; 2-deoxy-D-glucose; D-allulose; D-glucosamine
Online: 7 November 2018 (15:26:42 CET)
REVIEW
|
doi:10.20944/preprints202107.0497.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
lung cancer; immune checkpoint inhibitor; perioperative therapy; neoadjuvant therapy; adjuvant therapy
Online: 21 July 2021 (14:58:36 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0333.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Corrosion inhibitor; Synergistic effect; Electrochemical measurements; Theoretical calculation
Online: 14 November 2018 (10:23:29 CET)
ARTICLE
|
doi:10.20944/preprints201808.0146.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
histone deacetylase inhibitor, MHY2256, p53, apoptosis, autophagy, Ishikawa, endometrial cancer
Online: 7 August 2018 (14:37:46 CEST)
REVIEW
|
doi:10.20944/preprints202104.0742.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Diabetes mellitus; Glucose metabolism; Histone deacetylase; HDACs; Histone deacetylase inhibitor; HDACi, Insulin release; Sirtuins, Sirtuin activation
Online: 28 April 2021 (10:23:12 CEST)
REVIEW
|
doi:10.20944/preprints201806.0163.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SIRT6, Diabetes, Gluconeogenesis, Cancer, Aging, Heart Disease, Pharmacological SIRT6 Inhibitor, Cardiac Hypertrophy, Tumorigenesis, Neurodegeneration, Neurodegenerative Diseases, AD
Online: 29 August 2018 (13:04:23 CEST)
REVIEW
|
doi:10.20944/preprints202101.0151.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
complement system; proteolytic cascade; convertase; inhibitor; structural biology; molecular mechanism
Online: 8 January 2021 (11:54:36 CET)
ARTICLE
|
doi:10.20944/preprints202009.0006.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID-19; SARS-CoV-2; protein design; complementarity; competitive inhibitor; homology-based threading in rational protein design
Online: 4 March 2021 (10:14:39 CET)
ARTICLE
|
doi:10.20944/preprints201810.0391.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
wheat; alpha-amylase/trypsin inhibitor; heterologous expression; Pichia pastoris; allergy
Online: 17 October 2018 (17:15:23 CEST)
REVIEW
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hyperoxaluria; oxalate; inhibitor; small molecule drug; glycolate oxidase; lactate dehydrogenase; liver selective distribution
Online: 31 December 2020 (08:59:47 CET)
ARTICLE
|
doi:10.20944/preprints201812.0369.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
serine proteinase inhibitor; Kunitz; bikunin; inter-α-trypsin inhibitor; pre-α-trypsin inhibitor.
Online: 31 December 2018 (11:03:39 CET)
ARTICLE
|
doi:10.20944/preprints201901.0020.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
osteopontin; THP-1; brefelamide; inhibitor; tuberculosis
Online: 3 January 2019 (13:07:14 CET)
ARTICLE
|
doi:10.20944/preprints202105.0600.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
heparan sulfate; glycosaminoglycan; carbohydrate biosynthesis; azido sugar; small molecule inhibitor
Online: 25 May 2021 (10:17:59 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0570.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
bone resorption; butyric acid; HDAC inhibitor; osteoblasts; osteoprotegerin/RANKL; periodontal/root canal pathogens
Online: 24 October 2018 (11:21:42 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0374.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Keywords: Tumor microenvironment (TME), glioblastoma multiforme (GBM), GBM- associated macrophages (GAMs), exosomes, oncomiR-21, STAT3 inhibitor.
Online: 31 May 2019 (08:18:33 CEST)
REVIEW
|
doi:10.20944/preprints202305.1507.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Radionuclide therapy; nuclear medicine; radiopharmaceutical; antibody; peptide; small molecule inhibitor; tumor; microenvironment
Online: 22 May 2023 (10:51:48 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0088.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
There are many molecules used as drug carrier. TUD-1 is a newly synthesized mesoporous silica (SM) molecule possess two important features; consists of mesoporous so it is very suitable to be drug carrier in addition to that it has the ability to induce apoptosis in cancer cells. However, the effect of TUD-1 appears to act as cell death inducer, regardless of whether it is necrosis or apoptosis. Unfortunately, recent studies indicate that a proportion of cells undergo necrosis rather than apoptosis, which limits the use of TUD-1 as a secure treatment. On the other hand, lithium considered as necrosis inhibitor element. Hence, current study based on the idea of production a new Li/TUD-1 by incorporated mesoporous silica (TUD-1 type) with lithium in order to produce a new compound that has the ability to activate apoptosis by mesoporous silica (TUD-1 type) and at the same time can inhibit the activity of necrosis by lithium. Herein, lithium was incorporated in TUD-1 mesoporous silica by
Online: 4 October 2018 (15:54:02 CEST)
REVIEW
|
doi:10.20944/preprints201810.0732.v1
Subject:
Social Sciences,
Behavior Sciences
Keywords:
depression; estrogenic endocrine disruptor; environmental factor; inhibitor of differentiation; mental disorder
Online: 31 October 2018 (04:51:16 CET)
REVIEW
|
doi:10.20944/preprints201907.0081.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Heat shock protein 27; HSP27 inhibitor; Anti-cancer drugs, Resistance
Online: 4 July 2019 (13:19:51 CEST)
REVIEW
|
doi:10.20944/preprints202110.0450.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Fibrosis; Integrin; TGFβ; Therapeutic target; Drug; Inhibitor; Monoclonal antibody; α8β1; α11β1; Hepatic stellate cell
Online: 29 October 2021 (10:16:13 CEST)
ARTICLE
|
doi:10.20944/preprints201903.0166.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Structure-based design; glycogen phosphorylase inhibitor; glycogen metabolism; type 2 diabetes; X-ray crystallography; N-acyl-β-D-glucopyranosylamine
Online: 15 March 2019 (14:06:06 CET)
ARTICLE
|
doi:10.20944/preprints201909.0037.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
EGFR; ErbB3; Src; phosphorylation; TK inhibitor; cetuximab
Online: 4 September 2019 (03:21:39 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0177.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
chronic myeloid leukemia; tyrosine kinase inhibitor; adverse drug event; quality of life; second-generation tyrosine kinase inhibitor; nilotinib
Online: 16 August 2019 (08:09:07 CEST)
REVIEW
|
doi:10.20944/preprints201907.0256.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
PI 3-kinase; chromosomal instability; PI3K inhibitor; cancer; tumour evolution; centrosome
Online: 23 July 2019 (11:01:34 CEST)
COMMUNICATION
|
doi:10.20944/preprints201908.0126.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
protein-protein interaction; protein-peptide interaction; triglycine; substrate binding site; peptide; inhibitor; Proteinase K
Online: 11 August 2019 (08:37:08 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0124.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Heat shock factor (HSF-1) knockdown; heat shock proteins 70 and 27; radiosensitization; Hsp90 inhibitor NVP-AUY922; homologous recombination (HR)
Online: 11 September 2019 (13:37:00 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0122.v1
Subject:
Physical Sciences,
Biophysics
Keywords:
cervical adenocarcinoma; immune-checkpoint inhibitor; programmed cell death-1(PD-1); programmed cell death-ligand 1(PD-L1); CD8 expression; lymphocyte; survival analysis
Online: 12 January 2020 (15:01:23 CET)
REVIEW
|
doi:10.20944/preprints202209.0296.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
non-small-cell lung cancer; performance status; cytotoxic chemotherapy; immune checkpoint inhibitor; cancer cachexia
Online: 20 September 2022 (05:53:12 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0732.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Epidermal Growth Factor Receptor (EGFR); mutations, EGFR tyrosine kinase inhibitor; molecular epidemiology; Non-small-cell lung cancer
Online: 28 April 2021 (07:55:22 CEST)
COMMUNICATION
|
doi:10.20944/preprints202103.0113.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
blood-based mutation burden (bTMB); cancer immunotherapy; immune checkpoint inhibitor (ICI); biomarker; mutation
Online: 2 March 2021 (21:45:40 CET)
REVIEW
|
doi:10.20944/preprints202302.0123.v2
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
WNT; NF-κ B, Ion Channels; Anthrax toxin recep- tors; Poliovirus receptors; Porcupine inhibitor ETC-1922159; Sensitivity analysis; Colorectal cancer; Unknown biological hypotheses; Combinatorial search space; Support vector ranking
Online: 20 September 2024 (11:03:20 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0582.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Liquid-based 3D culture; tumoroid; cisplatin resistance; imatinib (gleevec); tyrosine kinase inhibitor (TKI); organoid; spheroid; metastatic colorectal cancer (mCRC)
Online: 23 December 2020 (10:15:46 CET)
REVIEW
|
doi:10.20944/preprints202209.0113.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Cancer; Immunotherapy; Microbiome; Immune Checkpoint Inhibitor; Immunology; Therapy
Online: 7 September 2022 (12:42:28 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1403.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer’s Disease; Tauopathy; Cell penetrating peptide; Polyarginine; TAT; Liposomes; Nanoparticles; Tau pathology; Tau aggregation inhibitor; Endocytosis
Online: 19 May 2023 (08:06:10 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0009.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
microbiome; melanoma; immune checkpoint inhibitor; diet; immunotherapy
Online: 3 October 2022 (12:19:54 CEST)
REVIEW
|
doi:10.20944/preprints202307.0430.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Hodgkin lymphoma; relapsed/refractory; brentuximab vedotin; checkpoint inhibitor; PD-1 inhibitor; nivolumab; pembrolizumab; autologous hematopoietic cell transplantation
Online: 6 July 2023 (11:44:13 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0585.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
glioblastoma; cancer stem cells; EMT; MGMT; temozolomide; doxorubicin; STAT3; EGFR inhibitor (AG1478)
Online: 31 January 2023 (12:01:04 CET)
REVIEW
|
doi:10.20944/preprints202401.1219.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
biofuel; insecticides; pesticides; catalytic reduction of CO2; green economy; sustainability; biodegradation; nanoparticles; corrosion inhibitor; nanofertilizer; heavy metal detection
Online: 16 January 2024 (13:35:19 CET)
REVIEW
|
doi:10.20944/preprints202305.1151.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
fusion proteins; inhibitor; therapeutic; cancer
Online: 16 May 2023 (10:32:09 CEST)
CASE REPORT
|
doi:10.20944/preprints202206.0266.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
PARP inhibitor; angiogenesis; immune suppression; recurrent ovarian cancer
Online: 20 June 2022 (10:02:09 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Kinase Inhibitor; NEK2; Chemoresistance; Avicennia marina; Marine compounds; Molecular docking; Cancer
Online: 7 June 2020 (11:16:35 CEST)
REVIEW
|
doi:10.20944/preprints202107.0353.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Lung cancer; Adjuvant treatment; Non-small-cell lung carcinoma (NSCLC); Epidermal growth factor receptor (EGFR); Tyrosine kinase inhibitor (TKI)
Online: 15 July 2021 (10:16:30 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0208.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Plasma PD-L1; liquid biopsy; cfRNA; immune checkpoint inhibitor; predictive immune biomarker; NSCLC
Online: 11 August 2022 (06:10:34 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0581.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Wheat; RNAi silencing; amylase/trypsin inhibitor (ATI); allergy; Non Celiac Wheat Sensitivity (NCWS)
Online: 24 July 2020 (11:51:53 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0559.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Nori; human ovarian tetracarcinoma (PA1); Tatridin B; NSD2 inhibitor
Online: 29 December 2022 (09:57:46 CET)
ARTICLE
|
doi:10.20944/preprints202306.1387.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
press cake; soy; extrusion; meat analogue; texture; water-holding capacity; oil-binding capacity; trypsin inhibitor activity
Online: 20 June 2023 (07:20:50 CEST)
REVIEW
|
doi:10.20944/preprints202004.0181.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
renal cell carcinoma; angiogenesis; immune-checkpoint inhibitor; tumor microenvironment; molecular subtypes; prognostic-biomarkers; predictive factors
Online: 12 April 2020 (04:48:44 CEST)
ARTICLE
|
doi:10.20944/preprints202010.0021.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Pioglitazone; DPP4-inhibitor; ESRD; Cardiovascular outcome; Mortality
Online: 1 October 2020 (15:41:50 CEST)
REVIEW
|
doi:10.20944/preprints202106.0609.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Chronic myeloid leukaemia; chronic phase; Tyrosine kinase inhibitor; Treatment free remission; deep molecular response; BCR-ABL.
Online: 25 June 2021 (08:13:40 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Azanucleoside; DMSO; DNA methylation, epigenetics; phosphorylation; restriction factor; triphosphohydrolase; methyltransferase inhibitor
Online: 4 January 2021 (08:19:38 CET)
ARTICLE
|
doi:10.20944/preprints202407.1116.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hepatitis C virus; MD Simulations; Covalent inhibitor; Drug resistance; Pharmacophore-based virtual screening
Online: 16 July 2024 (04:54:08 CEST)