REVIEW
|
doi:10.20944/preprints202401.0513.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Extracellular ubiquitin; monomeric ubiquitin; immunomodulatory drugs; sepsis; biotherapeutic proteins
Online: 8 January 2024 (02:23:44 CET)
ARTICLE
|
doi:10.20944/preprints202307.2144.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Streptozotocin; vanillic acid; silver nanoparticles; and antidiabetic drugs
Online: 1 August 2023 (03:46:33 CEST)
REVIEW
|
doi:10.20944/preprints202211.0147.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
topoisomerase; anticancer; cancer; anticancer drugs; enzyme
Online: 8 November 2022 (06:22:07 CET)
ARTICLE
|
doi:10.20944/preprints202308.1882.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
fSP3; drug design; bioavailability; non-systemic drugs; druglikeness; cheminformatics
Online: 29 August 2023 (03:25:53 CEST)
REVIEW
|
doi:10.20944/preprints202302.0030.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
angiogenesis inhibitors; VEGF inhibitors; ovarian cancer; progression-free survival; overall sur-vival; toxicity; systematic review; meta-analysis; randomized controlled trials; FDA approval of cancer drugs
Online: 2 February 2023 (05:26:47 CET)
REVIEW
|
doi:10.20944/preprints202310.1973.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
cornea; neovascularization; steroids; anti-VEGF drugs; keratoplasty; angiogenic factors; anti-angiogenic factors
Online: 30 October 2023 (17:25:56 CET)
ARTICLE
|
doi:10.20944/preprints202306.0784.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
antiepileptic drugs; age; autism spectrum disorder; epilepsy; ketogenic diet; mitochondrial dysfunction; modified Atkins diet; neurodevelopmental regression, seizures
Online: 12 June 2023 (07:23:54 CEST)
REVIEW
|
doi:10.20944/preprints202401.2185.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Avian Influenza; Pandemic Management; Epidemiology; Virology; Pathogenesis; Antiviral Drugs; Influenza Vaccines; Immune Response; Antigenic Drift; Antigenic Shift
Online: 31 January 2024 (08:04:16 CET)
REVIEW
|
doi:10.20944/preprints202306.1965.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Meningioma; Seizure prophylaxis; Antiepileptic drugs
Online: 28 June 2023 (10:57:21 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0115.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
dental pulp stem cells; nonsteroidal anti-inflammatory drugs; ibuprofen; diclofenac; angiogenesis; apoptosis
Online: 1 April 2024 (17:22:44 CEST)
REVIEW
|
doi:10.20944/preprints202401.1465.v1
Subject:
Biology And Life Sciences,
Behavioral Sciences
Keywords:
intracranial self-stimulation; brain-stimulation reward; optogenetics; optical ICSS;
reward; aversion; drugs of abuse; new psychoactive substances
reward; aversion; drugs of abuse; new psychoactive substances
Online: 19 January 2024 (07:08:28 CET)
ARTICLE
|
doi:10.20944/preprints202309.0432.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Brain; Caffeine; Cytokines; Ibuprofen; Intermittent Hypoxia; Myelination; Neuroinflammation; Non-steroidal Anti-inflammatory Drugs
Online: 6 September 2023 (11:12:33 CEST)
REVIEW
|
doi:10.20944/preprints202308.0951.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pulmonary arterial hypertension associated with connective tissue diseases; drugs; novel drugs; therapy; treatment; prognosis
Online: 11 August 2023 (13:25:08 CEST)
REVIEW
|
doi:10.20944/preprints202404.0437.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
neurodegenerative diseases; Parkinson’ s disease; Alzheimer’ s disease; drug discovery; disease-modifying drugs
Online: 5 April 2024 (12:39:57 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0034.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
pain; non-steroidal anti-inflammatory drugs; dysmenorrhea; edema; inflammation; over-the-counter drugs
Online: 1 August 2023 (14:21:27 CEST)
REVIEW
|
doi:10.20944/preprints202304.0933.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Spirocycles; three-dimensional; high-Fsp3; spirocyclizations; cyclodehydration; ketalization; intramolecular Claisen condensation; intramolecular alkylation; approved drugs
Online: 26 April 2023 (03:09:08 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0513.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
DNMT3A, QM/MM, covalent drugs, reaction mechanism
Online: 7 July 2023 (15:51:33 CEST)
REVIEW
|
doi:10.20944/preprints202305.0130.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
Obesity; hypothalamus; appetite; glucose homeostasis; weight-loss drugs; AGRP; POMC; NTS; incretins
Online: 3 May 2023 (10:22:49 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0457.v1
Subject:
Medicine And Pharmacology,
Veterinary Medicine
Keywords:
Newcastle disease virus; natural compounds; antiviral drugs; NDV; MD simulation; Hemagglutinin Neuraminidase; biological activity; ADMET; pharmacophore; screening
Online: 8 March 2024 (03:56:28 CET)
REVIEW
|
doi:10.20944/preprints202309.1061.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
prodrugs; HIV; AIDS; Nucleoside Reverse Transcriptase Inhibitors (NRTI); co-drugs; new drugs; medicinal chemistry
Online: 18 September 2023 (05:47:07 CEST)
ARTICLE
|
doi:10.20944/preprints202312.2072.v1
Subject:
Medicine And Pharmacology,
Tropical Medicine
Keywords:
Bothrops jararaca; Snakebite; Local Lesions; Inflammation; Leukocyte-endothelium interactions; Antivenom; Anti-inflammatory drugs; Microcirculation.
Online: 27 December 2023 (09:47:41 CET)
ARTICLE
|
doi:10.20944/preprints202209.0121.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Cathinones; Designer drugs; Bath salts; Neuronal injury; astroglial injury; Calpain; Caspase
Online: 8 September 2022 (09:14:34 CEST)
REVIEW
|
doi:10.20944/preprints202402.0853.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Artificial intelligence; Cancer; Covid.19; Chemotherapy; Target prediction drugs
Online: 16 February 2024 (02:28:25 CET)
REVIEW
|
doi:10.20944/preprints202403.1692.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
aryl hydrocarbon receptor; dopamine; antipsychotic drugs; naturally occurring antipsychotics; senotherapeutics
Online: 28 March 2024 (12:24:09 CET)
ARTICLE
|
doi:10.20944/preprints202308.0462.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Platinum drugs; acetylation; oxidation; immune response; mass spectrometry; chromatography
Online: 7 August 2023 (10:10:09 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1460.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Onchocerciasis; drug discovery; anthelmintics; O. gutturosa; motility and MTT inhibition; FDA approved drugs
Online: 23 November 2023 (09:31:11 CET)
ARTICLE
|
doi:10.20944/preprints202306.1149.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
platelets; blood coagulation; fibrin; thrombin generation; antiplatelet drugs; acetylsalicylic acid; ticagrelor; glycoprotein IIb-IIIa antagonists
Online: 15 June 2023 (13:13:19 CEST)
REVIEW
|
doi:10.20944/preprints202401.1141.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Osteporososis; diabetes mellitus; antihyperglycemic drugs; bone metabolism
Online: 15 January 2024 (16:32:34 CET)
SHORT NOTE
|
doi:10.20944/preprints202212.0230.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
monoamine oxidase; inhibitors; indole; 1,2,4-oxadiazole; drug research; neuroprotective drugs; Parkinson’s disease; MAO
Online: 13 December 2022 (07:12:01 CET)
ARTICLE
|
doi:10.20944/preprints202212.0467.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
azole drugs; cryptococcal meningitis; resistance; synergism; synthetic antifungal peptides
Online: 26 December 2022 (03:44:06 CET)
REVIEW
|
doi:10.20944/preprints202403.0030.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
alcohol; oxidative stress; inflammation; gut dysbiosis; biological drugs; probiotics
Online: 4 March 2024 (06:18:36 CET)
ARTICLE
|
doi:10.20944/preprints202402.1524.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Coccomyxa subellipsoidea KJ; metallothioneins; Th17 cytokines; T cell activation; immunoregulation; transcriptome analysis; peripheral blood mononuclear cells; inflammatory factors; toxic shock syndrome toxin-1; immune regulatory drugs
Online: 27 February 2024 (10:26:51 CET)
REVIEW
|
doi:10.20944/preprints202305.0014.v1
Subject:
Public Health And Healthcare,
Physical Therapy, Sports Therapy And Rehabilitation
Keywords:
HBV/HDV coinfection; Evolving antiviral drugs; innovative immune therapeutic agents; combination of antiviral and immune therapy
Online: 1 May 2023 (04:18:06 CEST)
REVIEW
|
doi:10.20944/preprints202305.1405.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
mitochondrial stress; insulin resistance; natural drugs
Online: 19 May 2023 (08:08:53 CEST)
REVIEW
|
doi:10.20944/preprints202401.1135.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
asthma; insulin resistance; antidiabetic drugs; metabolic dysfunction; obesity
Online: 15 January 2024 (14:52:22 CET)
REVIEW
|
doi:10.20944/preprints202304.0901.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
PCa; taxanes-based drugs; combination therapy; transmembrane proteins
Online: 25 April 2023 (08:34:03 CEST)
REVIEW
|
doi:10.20944/preprints202306.0011.v1
Subject:
Medicine And Pharmacology,
Transplantation
Keywords:
Desensitization; Donor specific antibodies; HLA system; antibodies identification; B cells; Plasma cells; Complement; New drugs; Desensitization; Donor specific antibodies; HLA system; B cells; Plasma cells; Complemennt; New drugs
Online: 1 June 2023 (03:17:00 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0151.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
hepatitis B; hepatitis delta; people who use drugs; people who inject drugs; harm reduction; population health; viral hepatitis; liver cancer
Online: 2 April 2024 (08:53:02 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1638.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
Gestational Diabetes Mellitus; pregnancy; antidiabetic drugs; prescription pattern
Online: 25 September 2023 (09:27:25 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0540.v1
Subject:
Biology And Life Sciences,
Aquatic Science
Keywords:
Emerging contaminants; Non-antibiotic drugs; Antimicrobial activity.
Online: 8 January 2024 (10:10:30 CET)
REVIEW
|
doi:10.20944/preprints202403.1857.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Microbiota; Diabetes; Gestational Diabetes; Probiotics, Drugs.
Online: 29 March 2024 (11:33:25 CET)
ARTICLE
|
doi:10.20944/preprints202312.0054.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Ex Vivo Resistance Platform; CAF-mediated Resistance; Combinations of cytotoxic and targeted drugs
Online: 1 December 2023 (07:57:41 CET)
ARTICLE
|
doi:10.20944/preprints202403.1394.v1
Subject:
Social Sciences,
Psychology
Keywords:
Doping; Performance-Enhancing Drugs; Psychometry; Sport Psychology
Online: 23 March 2024 (09:35:00 CET)
ARTICLE
|
doi:10.20944/preprints202309.1300.v1
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
semaglutide; drug misuse; drug abuse; pharmacovigilance; image- and performance-enhancing (IPED) drugs; glucagon-like peptide-1 (GLP-1) agonists
Online: 20 September 2023 (05:05:11 CEST)
REVIEW
|
doi:10.20944/preprints202312.2247.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Nonsteroidal anti-inflammatory drugs; pregnancy; adverse effects; analgesics; self-medication
Online: 29 December 2023 (04:01:29 CET)
ARTICLE
|
doi:10.20944/preprints202308.1019.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
1,2,3-triazoles; anti-cancer drugs; vibrational analysis; scaling; dimer calculation
Online: 14 August 2023 (10:36:19 CEST)
REVIEW
|
doi:10.20944/preprints202310.0168.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
IL-17; fibrosis; autoimmune; epigenetics; biological drugs.
Online: 3 October 2023 (15:25:03 CEST)
COMMUNICATION
|
doi:10.20944/preprints202403.0296.v1
Subject:
Environmental And Earth Sciences,
Other
Keywords:
detection technology of drugs in urban sewage; magnetic solid phase extraction; acoustic ejection mass spectrometry analysis method; fast detection
Online: 6 March 2024 (11:08:13 CET)
CASE REPORT
|
doi:10.20944/preprints202402.0716.v1
Subject:
Medicine And Pharmacology,
Orthopedics And Sports Medicine
Keywords:
Sinus Tarsi syndrome; Heel pain; Extracorporeal pulse-activated therapy (EPAT); Standard-of-care treatments; Non-steroidal anti-inflammatory drugs (NSAIDs); Foot orthosis; Laser therapy
Online: 13 February 2024 (08:01:19 CET)
ARTICLE
|
doi:10.20944/preprints202401.1005.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
designer receptors exclusively activated by designer drugs (DREADDs); infralimbic cortex; sleep; stress; transcranial direct current stimulation (tDCS); ventrolateral preoptic area
Online: 15 January 2024 (02:28:51 CET)
CASE REPORT
|
doi:10.20944/preprints202307.0658.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
hypertriglyceridemia; dyslipidemia; evinacumab; ANGPTL3-inhibitors; lipid-lowering drugs
Online: 11 July 2023 (10:45:58 CEST)
REVIEW
|
doi:10.20944/preprints202405.0326.v1
Subject:
Pharmacology And Toxicology,
Medicine And Pharmacology
Keywords:
SARS-CoV-2; 3CLpro; Novel Mechanism of Catalysis; FDA-approved drugs; Triad
Online: 7 May 2024 (16:44:24 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1441.v1
Subject:
Complementary And Alternative Medicine,
Medicine And Pharmacology
Keywords:
essential oils; GC-MS; antibacterial activity; gram-positive and gram-negative bacteria; diffusimetric antibiogram; antibacterial drugs; combinations; interactions
Online: 23 April 2024 (12:52:32 CEST)
REVIEW
|
doi:10.20944/preprints202405.0001.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Graves' disease; hyperthyroidism; Graves' ophthalmopathy; antithyroid drugs; stress
Online: 1 May 2024 (02:30:35 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1851.v1
Subject:
Complementary And Alternative Medicine,
Medicine And Pharmacology
Keywords:
platelet-activating factor acetyl hydrolase; non-steroidal anti-inflammatory drugs; cancer
Online: 29 April 2024 (03:43:14 CEST)