REVIEW
|
doi:10.20944/preprints202305.0473.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Drug Discovery; Drug Design; Drug Development, Quantum Computing, Quantum Machine Learning
Online: 8 May 2023 (08:37:23 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0296.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antimicrobial resistance; broad-spectrum antibiotics; antibacterial drug discovery; gram-negative bacteria; pyrrolobenzodiazepines
Online: 16 November 2022 (04:20:55 CET)
ARTICLE
|
doi:10.20944/preprints202303.0322.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Hemolytic peptide; Network science; Half-Space Proximal Networks; Metadata Networks; Visual mining; Cluster analysis; Motif discovery; StarPep toolbox; Peptide drug discovery
Online: 17 March 2023 (10:05:05 CET)
ARTICLE
|
doi:10.20944/preprints202305.1006.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Melanoma; drug discovery; spliceosomal inhibition; BRAF; cell line xenograft; organ histopathology
Online: 15 May 2023 (09:19:54 CEST)
REVIEW
|
doi:10.20944/preprints202309.0943.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
arbovirus; monoclonal antibody; flavivirus; alphavirus; neutralizing antibody; antibody discovery
Online: 14 September 2023 (03:51:07 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202211.0063.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
melanoma; drug discovery; spliceosomal inhibition; acute toxicity; blood chemistry; organ histopathology
Online: 3 November 2022 (01:43:05 CET)
ARTICLE
|
doi:10.20944/preprints202008.0213.v1
Subject:
Computer Science And Mathematics,
Computer Science
Keywords:
Clustering; Pattern Discovery; Time series; Multi-Level Spectral Clustering; English Channel
Online: 8 August 2020 (18:00:26 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0193.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Antibiofilm peptide; chemical space; StarPep toolbox; complex network; centrality measure; motif discovery
Online: 10 March 2023 (09:36:30 CET)
REVIEW
|
doi:10.20944/preprints202308.0434.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
In silico studies; drug discovery; SARS-CoV-2; molecular docking; virtual screening; molecular dynamics simulations; drug candidates; antiviral activity; receptor-ligand complex; drug design
Online: 4 August 2023 (11:11:21 CEST)
REVIEW
|
doi:10.20944/preprints202310.0771.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 12 October 2023 (04:19:37 CEST)
REVIEW
|
doi:10.20944/preprints202311.0529.v1
Subject:
Public Health And Healthcare,
Primary Health Care
Keywords:
SARS-CoV-2; Papain-like protease; COVID-19; Molecular modelling; Molecular dynamics simulations; Drug discovery; Antiviral drugs; Inhibitors; Therapeutic agents; therapeutic targets; Irreversible inhibitors; Repurposing drugs
Online: 8 November 2023 (16:11:55 CET)
REVIEW
|
doi:10.20944/preprints202401.1443.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
The Blood-Brain Barrier (BBB); CNS drug discovery; passive diffusion; active transport; Efflux transporters; Influx Transporters; P-glycoproteins (P-gp); breast cancer resistance protein (BCRP); in silico models
Online: 19 January 2024 (09:32:31 CET)
ARTICLE
|
doi:10.20944/preprints202310.0425.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
hepatitis B; antiviral; drug discovery; HBc protein; pharmacophore-based screening; drug repurposing
Online: 8 October 2023 (05:11:37 CEST)
REVIEW
|
doi:10.20944/preprints202311.1051.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Toxoplasma gondii; proteomics; host-parasite interactions; PTMs; drug discovery
Online: 16 November 2023 (07:46:09 CET)
ARTICLE
|
doi:10.20944/preprints202205.0146.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
ubiquitous exposure; diagnosis; research design; quality of health care; habitat injuries; discovery
Online: 11 May 2022 (05:40:27 CEST)
REVIEW
|
doi:10.20944/preprints202305.0945.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Systems Pharmacology; Polypharmacology; Adverse Events; Drug Discovery; Functional genomics; Disease Modeling; Network analysis; Innovation
Online: 12 May 2023 (12:18:59 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0109.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
triple negative breast cancer; MCAK/KIF2C; aneuploidy; chromosomal instability; drug discovery
Online: 1 June 2023 (15:47:29 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1350.v1
Subject:
Computer Science And Mathematics,
Computer Networks And Communications
Keywords:
echo chamber; filter bubble; digital social networks; social network analysis; polarization; diversity; community discovery
Online: 20 September 2023 (04:51:16 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0907.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
cancer; protein degradation; degraders; drug discovery; PROTAC; CDK9
Online: 11 January 2024 (10:20:13 CET)
ARTICLE
|
doi:10.20944/preprints202305.0908.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Deep Learning; Topic Discovery; Latent Dirichlet Allocation; Latent Semantic Analysis; Probabilistic Latent Semantic Analysis
Online: 12 May 2023 (08:52:57 CEST)
ARTICLE
|
doi:10.20944/preprints202307.2034.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bcl-2; Anti-apoptotic protein; Indole; Cancer drug discovery
Online: 28 July 2023 (14:36:37 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202310.1222.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Supercomputers; Pandemic; Drug Discovery; Public Health Preparedness
Online: 19 October 2023 (05:19:13 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0766.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 13 November 2023 (08:41:42 CET)
REVIEW
|
doi:10.20944/preprints202312.1443.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
marine Streptomyces; alkaloid; secondary metabolite; discovery; development
Online: 19 December 2023 (16:05:45 CET)
ARTICLE
|
doi:10.20944/preprints202402.0943.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
degradation monitoring; health monitoring; causal discovery; jaccard distance, inter- 14 pretability; causal interpretability
Online: 19 February 2024 (10:09:53 CET)
REVIEW
|
doi:10.20944/preprints202312.0982.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
HER2; HER2 discovery; HER2 role in cancers; HER 2 low; HER2DX; prognostic; predictive; biomarker; anti-HER therapies; HER2 landmark trials
Online: 13 December 2023 (11:35:40 CET)
ARTICLE
|
doi:10.20944/preprints202306.1818.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Alternative Splicing; two-colour (GFP/RFP) Fluorescent Reporter; MAPT; Exon-Skipping; FTDP-17; High Content Screening; siRNA; Nucleic Acids Therapeutics; Drug discovery
Online: 26 June 2023 (13:55:26 CEST)
REVIEW
|
doi:10.20944/preprints202404.0437.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
neurodegenerative diseases; Parkinson’ s disease; Alzheimer’ s disease; drug discovery; disease-modifying drugs
Online: 5 April 2024 (12:39:57 CEST)
REVIEW
|
doi:10.20944/preprints202311.1221.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
oxidative stress; atrial fibrillation; mitochondrial dysfunction; inflammation; antioxidant drug discovery
Online: 20 November 2023 (05:08:48 CET)
REVIEW
|
doi:10.20944/preprints202312.0548.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
brain cancers; gangliosides; mass spectrometry; biomarker discovery; screening; structural analysis
Online: 7 December 2023 (19:55:09 CET)
ARTICLE
|
doi:10.20944/preprints202308.1966.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Drug discovery; computational chemistry; conceptual DFT; marine cyclopeptides; chemical reactivity properties; bioavailability scores
Online: 29 August 2023 (09:36:49 CEST)
ARTICLE
|
doi:10.20944/preprints202401.2140.v1
Subject:
Environmental And Earth Sciences,
Soil Science
Keywords:
causal machine learning; soil analysis; causal discovery; crop fertilization; flood; agriculture; deposition; climate change
Online: 31 January 2024 (02:55:42 CET)
ARTICLE
|
doi:10.20944/preprints202403.1775.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Hepatitis B virus; Antivirals; Flavonoid; Drug discovery; Pharmacophore; Quantitative structure-activity relationship
Online: 28 March 2024 (13:31:24 CET)
ARTICLE
|
doi:10.20944/preprints202306.2033.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Process Mining; Process Model Discovery; Mining action+state evolution
Online: 28 June 2023 (16:19:00 CEST)
REVIEW
|
doi:10.20944/preprints202404.0055.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Lead optimization; drug discovery; artificial intelligence; machine learning; deep neural networks; cheminformatics; chemical modifications; drug development
Online: 1 April 2024 (13:35:22 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1460.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Onchocerciasis; drug discovery; anthelmintics; O. gutturosa; motility and MTT inhibition; FDA approved drugs
Online: 23 November 2023 (09:31:11 CET)
ARTICLE
|
doi:10.20944/preprints202309.0699.v1
Subject:
Computer Science And Mathematics,
Computer Networks And Communications
Keywords:
wireless sensor networks; energy harvesting; neighbor discovery; data fusion
Online: 12 September 2023 (04:10:25 CEST)
ARTICLE
|
doi:10.20944/preprints202312.2030.v1
Subject:
Biology And Life Sciences,
Aquatic Science
Keywords:
Myzostomida; symbiotic polychaetes; crinoids; Hainan Island; marine biodiversity; echinoderm symbionts; SCUBA; Sanya; new species discovery
Online: 27 December 2023 (10:08:27 CET)
Subject:
Environmental And Earth Sciences,
Paleontology
Keywords:
Pyrenees; paleoecology; hypothesis testing; discovery; serendipity; Quaternary; Lateglacial; Holocene; last millennia
Online: 10 May 2023 (08:24:15 CEST)
REVIEW
|
doi:10.20944/preprints202312.1256.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Biobanking; human biospecimens; drug discovery; health research
Online: 18 December 2023 (10:33:49 CET)
REVIEW
|
doi:10.20944/preprints202404.1013.v3
Subject:
Pharmacy,
Medicine And Pharmacology
Keywords:
computational pharmaceutics; AI; multi-scale modeling; quantum computing; drug discovery; blockchain frameworks
Online: 22 April 2024 (18:38:54 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2118.v1
Subject:
Engineering,
Other
Keywords:
Behaviour analysis; domestic environments; activities of daily living; knowledge discovery in databases
Online: 31 August 2023 (09:30:42 CEST)
REVIEW
|
doi:10.20944/preprints202405.0601.v1
Subject:
Life Sciences,
Biology And Life Sciences
Keywords:
Data science; Big data; Data mining; Bioinformatics; Chemometric; Medicinal chemistry; Targets; Knowledge discovery; Artificial intelligence, Machine learning, Deep learning; Data integration; Metadata, Database; QSAR; Collaborative drug discovery; Structure-based drug design; Ligand-based drug discovery; Clinical trials; Product development.
Online: 10 May 2024 (10:15:20 CEST)
CASE REPORT
|
doi:10.20944/preprints202405.0748.v1
Subject:
Library And Information Sciences,
Social Sciences
Keywords:
FAIR Principles; Open Science; Social Sciences and Humanities (SSH); Information and Data Management Systems; Discovery Platforms for SSH Research; OPERAS Services
Online: 13 May 2024 (08:04:58 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1701.v1
Subject:
Computer Networks And Communications,
Computer Science And Mathematics
Keywords:
Cryptographic; Private Set Intersection; Cuckoo Filter; Cloud Assistance; Private Contact Discovery)
Online: 26 April 2024 (00:14:06 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0971.v1
Subject:
Virology,
Biology And Life Sciences
Keywords:
virus detection; next-generation sequencing; bioinformatics analysis; SNP discovery; viral genomics; AI-assisted genomics
Online: 14 May 2024 (13:26:57 CEST)