ARTICLE
|
doi:10.20944/preprints201801.0214.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antitumour; cancer; chalcone; DMPK; in silico; in vivo
Online: 23 January 2018 (09:46:42 CET)
SHORT NOTE
|
doi:10.20944/preprints201801.0087.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
redox-sensitive; disulfide linker; gemini amphiphiles; gene therapy
Online: 10 January 2018 (09:12:03 CET)
ARTICLE
|
doi:10.20944/preprints201801.0079.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Diabetes; GPR40; AKRB1; PPARγ; GLUT-4
Online: 9 January 2018 (08:54:18 CET)
ARTICLE
|
doi:10.20944/preprints201711.0177.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochroman-4-ones; acyl hydrazone; cytotoxicity
Online: 2 January 2018 (10:11:55 CET)
ARTICLE
|
doi:10.20944/preprints201712.0066.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cancer; cell line; urea derivatives; synthesis; antiproliferative activity
Online: 11 December 2017 (15:10:36 CET)
ARTICLE
|
doi:10.20944/preprints201710.0200.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Thiazolidinones; ORAC assay; Metalloproteinase-9; Docking study; Keratinocytes cultures; Nuclear factor -kB.
Online: 31 October 2017 (16:36:16 CET)
ARTICLE
|
doi:10.20944/preprints201710.0196.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
osteoporosis; herbal medicine; Kukoamine B; osteoblast; osteoclast; bone mineral density; ovariectomized mice
Online: 31 October 2017 (15:35:04 CET)
ARTICLE
|
doi:10.20944/preprints201710.0194.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Africa; Terminalia brownii; antifungal extracts; Aspergillus, Nattrassia, Fusarium; triterpenoids; flavonoids; ellagitannins; stilbenes
Online: 31 October 2017 (09:54:35 CET)
ARTICLE
|
doi:10.20944/preprints201710.0088.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Caesalpinia sappan; cassane diterpenes; N bridge; antimalarial activity
Online: 13 October 2017 (06:30:04 CEST)
ARTICLE
|
doi:10.20944/preprints201708.0057.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
[18F]PSMA-1007; fluorine-18; PSMA; automation; prostate cancer; PET
Online: 17 August 2017 (06:10:57 CEST)
REVIEW
|
doi:10.20944/preprints201707.0019.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
affective disorders; alzheimer’s disease; l-Deprenyl (Selegiline); donepezil; galantamine; value; inhibitor constant; mechanism-based inhibition; multitarget-directed ligand (MTDL); rasagiline; rivastigmine
Online: 11 July 2017 (05:58:53 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0132.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
arylamine N-acetyltransferases; cancer; tuberculosis; drug discovery; traditional Chinese medicine; virtual screening; molecular dynamics simulation; MM-PBSA
Online: 30 June 2017 (11:36:22 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0128.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
steroidal dimer; steroidal N-heterocycles; antiproliferative activity; esophageal cancer cells
Online: 30 June 2017 (07:43:06 CEST)
COMMUNICATION
|
doi:10.20944/preprints201706.0074.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
deep-sea; actinomycete; Microbacterium sp.; indole
Online: 16 June 2017 (04:40:54 CEST)
REVIEW
|
doi:10.20944/preprints201705.0115.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Palladium; Suzuki cross coupling; natural product; non-natural product
Online: 15 May 2017 (18:30:52 CEST)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
REVIEW
|
doi:10.20944/preprints201703.0118.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
dengue; chikungunya; virus enzymes; antiviral; natural products
Online: 16 March 2017 (09:42:52 CET)
ARTICLE
|
doi:10.20944/preprints201703.0053.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,4-Thiadiazole; 1,2,4-Triazole; synthesis; MTT assay; Cytotoxicity of Schiff base
Online: 10 March 2017 (10:11:56 CET)
ARTICLE
|
doi:10.20944/preprints201703.0037.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hypertension; 4-hydroxy-2-nonenal (4HNE); reactive oxygen species(ROS)
Online: 7 March 2017 (07:00:16 CET)
ARTICLE
|
doi:10.20944/preprints201612.0082.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
transdermal physical penetration technology; Fu’s Cupping Therapy; pharmacokinetics; SEM; TEM; stratum corneum; mechanism
Online: 15 December 2016 (10:57:46 CET)
CASE REPORT
|
doi:10.20944/preprints201611.0134.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
GINKGO; hyperlipideamia; lipid profile
Online: 27 November 2016 (04:43:15 CET)
ARTICLE
|
doi:10.20944/preprints201611.0072.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aporphine derivatives; antiarrhythmia; 10,11-dibromocrebanine; 3-bromocrebanine; crebanine; stephanine
Online: 14 November 2016 (07:24:04 CET)
ARTICLE
|
doi:10.20944/preprints201611.0071.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
diabetes mellitus; metformin; glibenclamide and lipid profile
Online: 14 November 2016 (07:14:00 CET)
ARTICLE
|
doi:10.20944/preprints201611.0043.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chalcone; cytotoxic activity; pharmacophore model
Online: 7 November 2016 (08:30:12 CET)
ARTICLE
|
doi:10.20944/preprints201610.0137.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
glibenclamide therapies; glycemic; Glucose-6-phosphatase
Online: 31 October 2016 (08:35:41 CET)
ARTICLE
|
doi:10.20944/preprints201609.0122.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cancer; FGFR; Inhibitor; 4‐Substituted‐1H‐indazole
Online: 29 September 2016 (15:42:08 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0145.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
methyl 3,4-dihydroxybenzoate; oxidative stress; apoptosis; neuroprotection; nuclear factor erythroid 2-related factor 2
Online: 15 August 2016 (10:42:05 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0119.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
thiazoles; thiadiazoles; hydrazonoyl chlorides; anticancer activity; structure activity relationship
Online: 11 August 2016 (11:05:21 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0086.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Acid hydrolysis; Degradation product; Saikosaponin a
Online: 9 August 2016 (11:32:29 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0013.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
α-mangostin; antibacterial; antifungal; food packaging; semi-synthetic modification
Online: 2 August 2016 (09:02:09 CEST)