ARTICLE
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doi:10.20944/preprints202308.1882.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
fSP3; drug design; bioavailability; non-systemic drugs; druglikeness; cheminformatics
Online: 29 August 2023 (03:25:53 CEST)
REVIEW
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doi:10.20944/preprints202304.0933.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Spirocycles; three-dimensional; high-Fsp3; spirocyclizations; cyclodehydration; ketalization; intramolecular Claisen condensation; intramolecular alkylation; approved drugs
Online: 26 April 2023 (03:09:08 CEST)