ARTICLE
|
doi:10.20944/preprints202002.0438.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Simeprevir; Protease inhibitor; Virtual screening; Docking
Online: 28 February 2020 (13:14:38 CET)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0334.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
SARS-COV-2; folding/unfolding; antiparasitic; molecular docking; molecular dynamics; COVID-19; Ivermectin
Online: 19 April 2020 (06:56:09 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0079.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Nigella Sativa; 6LU7; 2GTB; molecular docking; MOE software
Online: 7 April 2020 (08:58:42 CEST)
ARTICLE
|
doi:10.20944/preprints201708.0057.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
[18F]PSMA-1007; fluorine-18; PSMA; automation; prostate cancer; PET
Online: 17 August 2017 (06:10:57 CEST)
ARTICLE
|
doi:10.20944/preprints202006.0326.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
2019-nCoV; 3CLpro protein; Cat's Claw; Uncaria tomentosa; Molecular Modeling
Online: 28 June 2020 (09:05:54 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0372.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; SARS-CoV-2; Marine natural product; Virtual screening; Docking
Online: 25 March 2020 (08:23:57 CET)
ARTICLE
|
doi:10.20944/preprints201608.0013.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
α-mangostin; antibacterial; antifungal; food packaging; semi-synthetic modification
Online: 2 August 2016 (09:02:09 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0119.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
thiazoles; thiadiazoles; hydrazonoyl chlorides; anticancer activity; structure activity relationship
Online: 11 August 2016 (11:05:21 CEST)
REVIEW
|
doi:10.20944/preprints201705.0115.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Palladium; Suzuki cross coupling; natural product; non-natural product
Online: 15 May 2017 (18:30:52 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0152.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chlorophyll; carotenoids; methanol; photo-protection; phytoextraction; Portulaca oleracea
Online: 15 September 2019 (15:04:55 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0086.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Acid hydrolysis; Degradation product; Saikosaponin a
Online: 9 August 2016 (11:32:29 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0122.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cancer; FGFR; Inhibitor; 4‐Substituted‐1H‐indazole
Online: 29 September 2016 (15:42:08 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0071.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
diabetes mellitus; metformin; glibenclamide and lipid profile
Online: 14 November 2016 (07:14:00 CET)
CASE REPORT
|
doi:10.20944/preprints201611.0134.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
GINKGO; hyperlipideamia; lipid profile
Online: 27 November 2016 (04:43:15 CET)
ARTICLE
|
doi:10.20944/preprints201703.0053.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,4-Thiadiazole; 1,2,4-Triazole; synthesis; MTT assay; Cytotoxicity of Schiff base
Online: 10 March 2017 (10:11:56 CET)
ARTICLE
|
doi:10.20944/preprints201608.0145.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
methyl 3,4-dihydroxybenzoate; oxidative stress; apoptosis; neuroprotection; nuclear factor erythroid 2-related factor 2
Online: 15 August 2016 (10:42:05 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0084.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
in silico repositioning; dual inhibitor; Covid-19; 3CLpro; PLpro; remdesivir
Online: 7 April 2020 (10:44:11 CEST)
ARTICLE
|
doi:10.20944/preprints201612.0082.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
transdermal physical penetration technology; Fu’s Cupping Therapy; pharmacokinetics; SEM; TEM; stratum corneum; mechanism
Online: 15 December 2016 (10:57:46 CET)
ARTICLE
|
doi:10.20944/preprints201611.0043.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chalcone; cytotoxic activity; pharmacophore model
Online: 7 November 2016 (08:30:12 CET)
ARTICLE
|
doi:10.20944/preprints201610.0137.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
glibenclamide therapies; glycemic; Glucose-6-phosphatase
Online: 31 October 2016 (08:35:41 CET)
REVIEW
|
doi:10.20944/preprints201703.0118.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
dengue; chikungunya; virus enzymes; antiviral; natural products
Online: 16 March 2017 (09:42:52 CET)
ARTICLE
|
doi:10.20944/preprints201611.0072.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aporphine derivatives; antiarrhythmia; 10,11-dibromocrebanine; 3-bromocrebanine; crebanine; stephanine
Online: 14 November 2016 (07:24:04 CET)
ARTICLE
|
doi:10.20944/preprints202006.0358.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Enzyme inhibition; Secondary Metabolites; In-silico Analysis; Molecular docking; Drug candidates
Online: 30 June 2020 (08:11:28 CEST)
ARTICLE
|
doi:10.20944/preprints201703.0037.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hypertension; 4-hydroxy-2-nonenal (4HNE); reactive oxygen species(ROS)
Online: 7 March 2017 (07:00:16 CET)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
ARTICLE
|
doi:10.20944/preprints201902.0064.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Dopamine receptors, Molecular Docking, Molecular Dynamics, Receptor-Ligand Interactions
Online: 6 February 2019 (13:54:13 CET)
REVIEW
|
doi:10.20944/preprints201906.0219.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
phytochemistry; biological activities; Apocynaceae family
Online: 21 June 2019 (18:28:55 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0194.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Africa; Terminalia brownii; antifungal extracts; Aspergillus, Nattrassia, Fusarium; triterpenoids; flavonoids; ellagitannins; stilbenes
Online: 31 October 2017 (09:54:35 CET)
ARTICLE
|
doi:10.20944/preprints201706.0132.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
arylamine N-acetyltransferases; cancer; tuberculosis; drug discovery; traditional Chinese medicine; virtual screening; molecular dynamics simulation; MM-PBSA
Online: 30 June 2017 (11:36:22 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0292.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
African medicinal plants; Leishmaniasis; natural products; protozoal diseases; Schistosomiasis; Trypanosomiasis
Online: 31 January 2018 (05:28:15 CET)
ARTICLE
|
doi:10.20944/preprints201710.0196.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
osteoporosis; herbal medicine; Kukoamine B; osteoblast; osteoclast; bone mineral density; ovariectomized mice
Online: 31 October 2017 (15:35:04 CET)
COMMUNICATION
|
doi:10.20944/preprints201706.0074.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
deep-sea; actinomycete; Microbacterium sp.; indole
Online: 16 June 2017 (04:40:54 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0128.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
steroidal dimer; steroidal N-heterocycles; antiproliferative activity; esophageal cancer cells
Online: 30 June 2017 (07:43:06 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0142.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
reactive selenium species; arylmethyl selenocyanate; cellular thiolstat; antimicrobial; anticancer; ESKAPE; multidrug resistance
Online: 22 February 2018 (11:34:22 CET)
ARTICLE
|
doi:10.20944/preprints201801.0079.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Diabetes; GPR40; AKRB1; PPARγ; GLUT-4
Online: 9 January 2018 (08:54:18 CET)
ARTICLE
|
doi:10.20944/preprints201712.0066.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cancer; cell line; urea derivatives; synthesis; antiproliferative activity
Online: 11 December 2017 (15:10:36 CET)
ARTICLE
|
doi:10.20944/preprints201801.0214.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antitumour; cancer; chalcone; DMPK; in silico; in vivo
Online: 23 January 2018 (09:46:42 CET)
ARTICLE
|
doi:10.20944/preprints201803.0142.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chitosan; thermoresponsive hydrogel; nitric oxide; s-nitrosothiols; biocompatibility; antimicrobial; Pseudomonas aeruginosa; pluronic F127
Online: 19 March 2018 (07:25:27 CET)
REVIEW
|
doi:10.20944/preprints201707.0019.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
affective disorders; alzheimer’s disease; l-Deprenyl (Selegiline); donepezil; galantamine; value; inhibitor constant; mechanism-based inhibition; multitarget-directed ligand (MTDL); rasagiline; rivastigmine
Online: 11 July 2017 (05:58:53 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0253.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
halogen bonding; fluorine; iodine; pentafluorosulfanyl; titration; ab initio calculation; NMR study; drug design
Online: 25 August 2019 (15:41:59 CEST)
REVIEW
|
doi:10.20944/preprints201811.0409.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
G quadruplex, Oncogene, ligand, cancer
Online: 16 November 2018 (11:34:24 CET)
ARTICLE
|
doi:10.20944/preprints201803.0050.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
carboxamide; carbohydrazine; antibacterial; antifungal; molecular docking; Schiff base; NMR; IR
Online: 7 March 2018 (05:11:10 CET)
ARTICLE
|
doi:10.20944/preprints201710.0088.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Caesalpinia sappan; cassane diterpenes; N bridge; antimalarial activity
Online: 13 October 2017 (06:30:04 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0307.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
molecular docking; fluoroquinolones; antimicrobial activity
Online: 30 January 2019 (09:31:52 CET)
ARTICLE
|
doi:10.20944/preprints201802.0021.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Keywords: one-pot synthesis; single crystal x-ray crystallography; oxovanadium(IV); zinc(II); spectroscopic studies; in vitro antibacterial studies.
Online: 2 February 2018 (16:00:10 CET)
REVIEW
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Simaroubaceae; Picrasma javanica; quassionoids; phytochemicals; pharmacological properties
Online: 19 March 2019 (10:49:34 CET)
ARTICLE
|
doi:10.20944/preprints201809.0048.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
pretargeting; Fusarinine C; rituximab; click chemistry; multimerization; PET; gallium-68
Online: 3 September 2018 (15:55:44 CEST)
REVIEW
|
doi:10.20944/preprints202308.1912.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
3D printing; polymers for maxillofacial prostheses; adhesives; osseointegrated implants; nasal; auricle and ocular prostheses
Online: 29 August 2023 (03:30:06 CEST)
REVIEW
|
doi:10.20944/preprints201808.0032.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
caffeine; methylxanthine; chlorogenic acid; caffeic acid; inflammation; antimutagen; anticancer; antioxidant
Online: 2 August 2018 (05:14:02 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0091.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
asymmetrical mono-carbonyl analogs of curcumin (AMACs); synthesis; cytotoxicity, Vero; HeLa; MCF7; cell lines
Online: 4 June 2018 (08:19:03 CEST)
ARTICLE
|
doi:10.20944/preprints201903.0166.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Structure-based design; glycogen phosphorylase inhibitor; glycogen metabolism; type 2 diabetes; X-ray crystallography; N-acyl-β-D-glucopyranosylamine
Online: 15 March 2019 (14:06:06 CET)
ARTICLE
|
doi:10.20944/preprints201909.0024.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
JBIR-99; high-speed counter-current chromatography; polyketide; NMR spectroscopy; mass spectroscopy; X-ray crystallography; Meyerozyma guilliermondii
Online: 2 September 2019 (11:20:28 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0012.v3
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chitosan; self-assembled; polyelectrolyte complex; nanoparticle; drug delivery
Online: 21 February 2018 (16:00:38 CET)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)
ARTICLE
|
doi:10.20944/preprints201803.0003.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
derivatives of N-phenylanthranilic acids; anti-inflammatory activity; flexible molecular docking; microsomal prostaglandin E synthase-1
Online: 1 March 2018 (04:58:58 CET)
ARTICLE
|
doi:10.20944/preprints201908.0127.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Cucurbitaceae; cucurbitacines; triterpenic saponines; cell cancer lines; antiproliferative activities
Online: 11 August 2019 (08:50:51 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Keywords: methotrexate, cubic phase, magnetocubosomes, monoolein, liquid crystalline phase, drug delivery system, alternating magnetic field
Online: 4 January 2019 (14:32:38 CET)
ARTICLE
|
doi:10.20944/preprints201805.0133.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antioxidant potential; molecular docking; molecular descriptors; binding free energy; free radicals; oxidative stress
Online: 8 May 2018 (15:38:38 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0223.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
LSD1; molecular inhibitors; thieno[3,2-b]pyrrole-5-carboxamide derivatives; Molecular docking; 3D-QSAR; Molecular dynamics simulations
Online: 21 August 2019 (09:54:43 CEST)
ARTICLE
|
doi:10.20944/preprints201910.0174.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
AQP3 protein; molecular docking; molecular dynamics; MM-GBSA analysis; pharmacophore-based filter
Online: 16 October 2019 (04:37:31 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0251.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
docking; epigenetics; epi-informatics; molecular interactions; molecular dynamics; natural products; flavonoids
Online: 14 July 2018 (17:45:16 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0177.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochroman-4-ones; acyl hydrazone; cytotoxicity
Online: 2 January 2018 (10:11:55 CET)
ARTICLE
|
doi:10.20944/preprints201710.0200.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Thiazolidinones; ORAC assay; Metalloproteinase-9; Docking study; Keratinocytes cultures; Nuclear factor -kB.
Online: 31 October 2017 (16:36:16 CET)
SHORT NOTE
|
doi:10.20944/preprints201801.0087.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
redox-sensitive; disulfide linker; gemini amphiphiles; gene therapy
Online: 10 January 2018 (09:12:03 CET)
ARTICLE
|
doi:10.20944/preprints201805.0085.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
7-acetamido-2-aryl-5-bromoindoles; trifluoroacetylation; cytotoxicity; apoptosis; tubulin polymerization; molecular docking
Online: 4 May 2018 (07:47:06 CEST)
REVIEW
|
doi:10.20944/preprints201807.0226.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
galvanic replacement; photothermal therapy; drug delivery; nanoparticles; cancer treatment
Online: 13 July 2018 (05:11:21 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0419.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
doxorubicin; heterobifunctional; linker
Online: 29 May 2018 (08:54:56 CEST)
REVIEW
|
doi:10.20944/preprints201905.0066.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chitin; chitosan; cosmetics; biodegradability; biomaterials; polysaccharides; green technology; marine cosmetic ingredients; marine green source; marine resources
Online: 6 May 2019 (12:37:44 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0189.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
G-quadruplex DNA; interactions; berberine and palmatine analogues; chemotherapy; NMR; FRET and MST assays
Online: 14 May 2018 (11:44:10 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201807.0039.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
xanthohumol; biotinylated chalcones; anticancer activity; antioxidants
Online: 3 July 2018 (11:42:41 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0558.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; protein protein interactions; virtual screening; docking; molecular dynamics; zinc
Online: 2 September 2020 (09:48:48 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0371.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
biosynthesis; nanoparticles; plant extracts; Citrus reticulata
Online: 16 November 2018 (04:33:22 CET)
ARTICLE
|
doi:10.20944/preprints201808.0011.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chitosan; aldehydes; chalcone; MIC; anti-cancer activity
Online: 1 August 2018 (09:38:35 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0561.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
cheminformatics, drugs, drug-likeness, drug discovery, natural products
Online: 23 November 2018 (13:56:32 CET)
ARTICLE
|
doi:10.20944/preprints201909.0130.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Synthesis; triazinoindole; thiosemicarbazide; alpha-glucosidase; molecular docking study; SAR
Online: 13 September 2019 (10:54:30 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminopeptidases; inhibitors; aminophosphonate; phenylglycine analogues; fluorine substituted; molecular modeling
Online: 6 May 2019 (10:16:45 CEST)
HYPOTHESIS
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
SARS-CoV-2; zinc; zn; zinc-deficiency; cytokine storm
Online: 8 September 2020 (10:09:19 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0110.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
G-quadruplex; oxadiazole/pyridine polyheteroaryls; G4-ligands; FRET-melting; G4-FID; circular dichroism
Online: 6 July 2018 (08:28:22 CEST)
ARTICLE
|
doi:10.20944/preprints201904.0262.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
total synthesis; antitumor activity; structure-activity relationship
Online: 24 April 2019 (05:29:48 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0106.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ecdysterone; metabolites; excretion profile; urinary pharmacokinetics
Online: 6 May 2021 (15:20:04 CEST)
REVIEW
|
doi:10.20944/preprints201804.0071.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Sulfenic acids; Sulfoxides; Sulfones; Disulfides; Alliin derivatives; Glycoconjugates; Pyrimidine derivatives.
Online: 5 April 2018 (16:30:18 CEST)
ARTICLE
|
doi:10.20944/preprints201902.0248.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
10-methoxycanthin-6-one; quaternization; antibacterial; SARs
Online: 27 February 2019 (05:08:02 CET)
ARTICLE
|
doi:10.20944/preprints201805.0437.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Jatropha pelargoniifolia; alkaloids; flavonoids; coumarinolignans; diterpenes; anti-inflammatory; antinociceptive; antipyretic; free radical scavenging
Online: 30 May 2018 (06:15:42 CEST)
REVIEW
|
doi:10.20944/preprints201806.0093.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
marine organisms; carbohydrate; glycoside; antioxidant; anticoagulant; anti-inflammatory; antitumor; antimicrobial
Online: 6 June 2018 (12:32:12 CEST)
ARTICLE
|
doi:10.20944/preprints201907.0215.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Platinum, N-heterocyclic carbene ligand, anticancer activity, DNA interaction, optical tweezers technique, liquid phase AFM microscop
Online: 18 July 2019 (10:17:27 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0355.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
assay; diarrhea; isolate; hydrolysis; proteins; inhibition zone
Online: 16 October 2018 (11:26:59 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0448.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
acetyleugenol; Acacia nilotica; anti-tuberculosis; Serine/Threonine kinases; multi-drug resistant TB
Online: 24 April 2020 (14:12:33 CEST)
ARTICLE
|
doi:10.20944/preprints202010.0576.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Antimalarial; Erythrina fusca; Phaseolin; Molecular docking; Phytochemical analysis
Online: 21 October 2021 (12:08:52 CEST)
REVIEW
|
doi:10.20944/preprints201911.0392.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
fungal pathogens; antifungal agents; natural products
Online: 30 November 2019 (11:30:19 CET)
ARTICLE
|
doi:10.20944/preprints202211.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Antivirals; coronavirus; COVID-19; covalent drugs; dynamic light scattering; inhibitors; main protease; natural products
Online: 28 November 2022 (13:40:01 CET)
ARTICLE
|
doi:10.20944/preprints202007.0495.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
In silico target prediction; dihydrochalcones; SEA; SwissTargetPrediction; SuperPred; polyphamracology; virtual screening
Online: 21 July 2020 (13:43:40 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0359.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1, 2, 4-Triazine; Lanosterol 14a-demethylase (CYP51); Drug Resistance; Molecular Docking; Molecular Dynamic Simulation.
Online: 17 August 2021 (12:27:02 CEST)
ARTICLE
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Astragalus aitosensis; flavonoid; glycoside
Online: 29 March 2019 (09:13:02 CET)
ARTICLE
|
doi:10.20944/preprints201812.0027.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Rumex tunetanus; Phenolic compounds; Metabolic profiling; Antioxidant activity; RP-UHPLC-ESI-QTOF-MS
Online: 3 December 2018 (13:58:52 CET)
ARTICLE
|
doi:10.20944/preprints201911.0375.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
synthesis; 2-mercaptabezimidazole; sulfonamide; molecular docking study; α-amylase; sa
Online: 29 November 2019 (10:28:22 CET)
ARTICLE
|
doi:10.20944/preprints201804.0282.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminosteroid; aminocycloartane; alkaloid; 3D-QSAR; CoMFA; antitrypanosomal activity; cytotoxicity
Online: 23 April 2018 (11:02:16 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0063.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
FABP4; A-FABP; aP2; antidiabetes; antiobesity; antiatherosclerosis; anticancer; computational tools; computer-aided drug discovery
Online: 5 September 2019 (15:39:58 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0574.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
activity cliff; activity landscape plotter; epigenetics; docking; drug discovery; D-tools; molecular dynamics; Epi-polypharmacology; SmART; structure-activity relationships
Online: 26 November 2018 (07:14:05 CET)