@article{202305.1103, doi = {10.20944/preprints202305.1103.v1}, url = {https://doi.org/10.20944/preprints202305.1103.v1}, year = 2023, month = {May}, publisher = {Preprints}, author = {Maria Francesca Armentano and Paolo Lupattelli and Faustino Bisaccia and Rosarita D’Orsi and Rocchina Miglionico and Ilaria Nigro and Alessandro Santarsiere and Federico Berti and Maria Funicello and Lucia Chiummiento}, title = {Novel Wild Type and Mutate HIV-1 Protease Inhibitors Containing Heteroaryl Carboxamides in P2: Synthesis, Biological and ADME Evaluations}, journal = {Preprints} }