REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1288.v2
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
SGLT2 Inhibitors; Empagliflozin; Renal fibrosis; Connective tissue growth factor; Epithelial-mesenchymal transition
Online: 23 February 2024 (13:25:01 CET)
ARTICLE
|
doi:10.20944/preprints201611.0023.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
anti-yeast; enzyme inhibitors; Terminalia mantaly; Combretaceae
Online: 3 November 2016 (09:35:17 CET)
REVIEW
|
doi:10.20944/preprints202402.1496.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Proton-pump inhibitors; eosinophilic esophagitis; pharmacogenetics; CYP219 gene; STAT6 gene.
Online: 26 February 2024 (23:53:49 CET)
REVIEW
|
doi:10.20944/preprints202402.1593.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
type 2 diabetes; therapeutic inertia; clinical guidelines; sodium-glucose cotransporter-2 inhibitors; glucagon-like peptide-1 receptor agonists; primary health care
Online: 28 February 2024 (10:53:42 CET)
REVIEW
|
doi:10.20944/preprints202403.1203.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
rectal cancer; total neoadjuvant treatment; immunocheckpoint inhibitors; nonoperative management; ctDNA.
Online: 20 March 2024 (16:08:21 CET)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
CASE REPORT
|
doi:10.20944/preprints202402.0658.v3
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pharmacokinetic-pharmacodynamic interactions; low-dose methotrexate; proton pump inhibitors; analgesics; pancytopenia; hepatotoxicity
Online: 1 April 2024 (11:53:15 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
REVIEW
|
doi:10.20944/preprints201905.0358.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
alloimmune response; immunosuppressants; calcineurin inhibitors; corticosteroids; mTOR inhibitors; neurotoxicity; neuroprotective effects
Online: 29 May 2019 (16:37:44 CEST)
REVIEW
|
doi:10.20944/preprints202306.0041.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
APE1; inhibitors; cancer.
Online: 1 June 2023 (07:05:48 CEST)
REVIEW
|
doi:10.20944/preprints202309.0120.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Melanoma; BRAF mutations; BRAF inhibitors; MEK inhibitors; Immunotherapy
Online: 4 September 2023 (15:46:20 CEST)
REVIEW
|
doi:10.20944/preprints201903.0288.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Enhancers; BET inhibitors; CDK7 inhibitors; HDAC inhibitors; Transcription factors; eRNAs; cancer
Online: 30 March 2019 (08:33:07 CET)
ARTICLE
|
doi:10.20944/preprints202403.0239.v1
Subject:
Clinical Medicine,
Medicine And Pharmacology
Keywords:
JAK inhibitors; Psoriasis; Psoriatic arthitis
Online: 5 March 2024 (06:02:35 CET)
REVIEW
|
doi:10.20944/preprints202307.0539.v3
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Hepatocellular carcinoma; tyrosine kinase inhibitors; immune checkpoint inhibitors; biomarkers
Online: 17 July 2023 (13:22:33 CEST)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1058.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Heart Failure; Therapy; type-2 sodium-glucose cotransporters inhibitors; angiotensin receptor neprylisin inhibitors
Online: 17 July 2023 (15:07:48 CEST)
REVIEW
|
doi:10.20944/preprints201903.0256.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immunocheckpoint inhibitors; chemotherapy; tirosin kinase inhibitors; angiogenesis
Online: 28 March 2019 (06:48:37 CET)
REVIEW
|
doi:10.20944/preprints202003.0251.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
gastric acid suppressant; chemotherapy; tyrosine kinase inhibitors; proton pump inhibitors
Online: 31 March 2020 (03:40:46 CEST)
REVIEW
|
doi:10.20944/preprints202307.0043.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Gliomas; Tumour Microenvironment; Immunotherapy; Immune Checkpoint Inhibitors; Vaccines
Online: 4 July 2023 (02:39:07 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1065.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
psoriasis; plasma cytokines; TNFα inhibitors; etanercept; infliximab; adalimumab
Online: 18 September 2023 (02:32:17 CEST)
REVIEW
|
doi:10.20944/preprints202401.1747.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
chronic lymphocytic leukemia; BTK inhibitors; BCL-2 inhibitors; prognostic scores; predictive factors; TP53 abnormalities; IGHV; complex karyotype
Online: 24 January 2024 (13:39:51 CET)
ARTICLE
|
doi:10.20944/preprints202306.2038.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Neurodegenerative diseases; cholinesterase inhibitors; monoaminoxidase inhibitors; photo-pharmacology
Online: 29 June 2023 (02:47:23 CEST)
REVIEW
|
doi:10.20944/preprints202402.1417.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
heart failure; type 1 diabetes; diabetic cardiomyopathy; hospitalization; HFpEF; HFrEF; SGLT2-i; sodium-glucose cotransporter-2 inhibitors; diabetic ketoacidosis; epidemiologic studies; patient education; continuous monitoring of ketone levels; ketonemia
Online: 26 February 2024 (11:54:41 CET)
REVIEW
|
doi:10.20944/preprints202401.0800.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
psoriasis; oral therapies; topical therapies; biologics; Jak inhibitors; PDE4 inhibitors; systemic treatment; IL-17 inhibitors; IL-23 inhibitors; tapinarof; roflumilast
Online: 10 January 2024 (08:49:06 CET)
COMMUNICATION
|
doi:10.20944/preprints202012.0365.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
corrosion; amino acids; inhibitors; steel; iron; Monte Carlo simulation
Online: 15 December 2020 (10:09:29 CET)
REVIEW
|
doi:10.20944/preprints202307.0013.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
prostate cancer; PARP inhibitors; DDR gene; CRPC
Online: 3 July 2023 (08:22:22 CEST)
REVIEW
|
doi:10.20944/preprints202111.0087.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virome; microbiota; cancer; bacteriophages; fecal microbiota transplantation; checkpoint inhibitors; immunotherapy
Online: 3 November 2021 (14:30:14 CET)
REVIEW
|
doi:10.20944/preprints202104.0679.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Sildenafil; phosphodiesterase 5 inhibitors; drug repurposing; cancer; chemoadjuvant
Online: 26 April 2021 (15:02:08 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
REVIEW
|
doi:10.20944/preprints202306.0609.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Kinases; human diseases; macrocyclic inhibitors; drug discovery
Online: 8 June 2023 (08:54:08 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0027.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
microginins; cyanobacteria; Microcystis; aminopeptidase M inhibitors
Online: 5 January 2018 (04:16:23 CET)
ARTICLE
|
doi:10.20944/preprints202109.0520.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Phytoene, Dunaliella salina, mitosis inhibitors, herbicides, red light
Online: 30 September 2021 (14:18:55 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1422.v1
Subject:
Gastroenterology And Hepatology,
Medicine And Pharmacology
Keywords:
eosinophilic esophagitis; esophagus; proton pump inhibitors
Online: 22 May 2024 (07:54:48 CEST)
REVIEW
|
doi:10.20944/preprints202208.0008.v3
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adamantanes; antivirals; cap-dependent endonuclease inhibitors; influenza; neuraminidase inhibitors; umifenovir
Online: 19 September 2023 (04:16:16 CEST)
REVIEW
|
doi:10.20944/preprints201809.0291.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
CCR6, CCL20, Inhibitors, TH17, Treg, Inflammatory diseases, Cancer
Online: 17 September 2018 (09:31:43 CEST)
REVIEW
|
doi:10.20944/preprints202304.0843.v2
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
CLL, Zanubrutinib, BTK inhibitors, efficacy, safety, chronic lymphocytic leukemia
Online: 22 May 2023 (16:15:16 CEST)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
ARTICLE
|
doi:10.20944/preprints202311.1799.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
usnic acid derivatives; TDP1 inhibitors; anticancer therapy; topotecan
Online: 28 November 2023 (10:06:47 CET)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
REVIEW
|
doi:10.20944/preprints202004.0160.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; ACE; ACE2; Angiotensin II; Bradykinin; RAS inhibitors; ACE inhibitors; AT1 receptor blockers; Losartan; Bradykinin Antagonists; Ang II loading; Giapreza; Icatibant.
Online: 14 April 2020 (14:34:43 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0540.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
3-hydroxy-3-methylglutaryl-coenzyme-A inhibitors; Sepsis
Online: 27 July 2018 (13:07:17 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0483.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
MRONJ; CDK4/6 inhibitors; metastatic breast cancer; oral epidemiology
Online: 8 November 2023 (08:42:55 CET)
REVIEW
|
doi:10.20944/preprints202306.0143.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Systemic sclerosis; treatment; Janus kinase inhibitors; fibrosis; anti-cytokine treatment
Online: 2 June 2023 (07:07:00 CEST)
REVIEW
|
doi:10.20944/preprints202401.0541.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
NSCLC; ALK inhibitors; lung cancer; targeted therapy; precision medicine
Online: 8 January 2024 (11:27:23 CET)
CASE REPORT
|
doi:10.20944/preprints202312.1085.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
Antiphospholipid syndrome; TNF-α Inhibitors; Dangerous pregnancy; gestational weeks
Online: 14 December 2023 (12:15:47 CET)
REVIEW
|
doi:10.20944/preprints202401.0407.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
prostatic neoplasm; biochemical recurrence; androgen receptor signaling inhibitors; androgen deprivation therapy
Online: 4 January 2024 (11:22:30 CET)
ARTICLE
|
doi:10.20944/preprints201911.0010.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
aromatase inhibitors; anastrozole; levonorgestrel-iud; endometriosis; endometriomas; clinical trial
Online: 1 November 2019 (12:47:34 CET)
ARTICLE
|
doi:10.20944/preprints202309.1391.v1
Online: 21 September 2023 (03:32:12 CEST)
ARTICLE
|
doi:10.20944/preprints202310.0713.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
colon cancer; cathepsin B; radiotherapy; radioresistance; cathepsin inhibitors; CA074
Online: 11 October 2023 (10:48:48 CEST)
ARTICLE
|
doi:10.20944/preprints202102.0525.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
HIV-RT; ribonuclease H; dual inhibitors; docking; putative binding
Online: 23 February 2021 (15:51:40 CET)
REVIEW
|
doi:10.20944/preprints202108.0364.v1
Subject:
Medicine And Pharmacology,
Tropical Medicine
Keywords:
dengue virus; antiviral targets; NS5; flavivirus; polymerase; nucleoside inhibitors; non-nucleoside inhibitors
Online: 17 August 2021 (14:07:29 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0016.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; elderly; proton pump inhibitors; antipsychotics; metformin; oral antidiabetics
Online: 2 May 2020 (15:48:33 CEST)
REVIEW
|
doi:10.20944/preprints202108.0037.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ovarian cancer; checkpoint inhibitors; ICIs; immunotherapy; PARP; avelumab; pembrolizumab; nivolumab; bevacizumab; platinum
Online: 2 August 2021 (13:01:35 CEST)
REVIEW
|
doi:10.20944/preprints202311.1805.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
HDAC6; histone deacetylases inhibitors; colorectal cancer
Online: 28 November 2023 (10:13:23 CET)
ARTICLE
|
doi:10.20944/preprints202307.1694.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
Idiopathic Pulmonary Fibrosis; Lung Neoplasms; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Database
Online: 25 July 2023 (10:01:14 CEST)
REVIEW
|
doi:10.20944/preprints202305.1789.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PTK6; Colorectal cancer; Tyrosine Kinase Inhibitors
Online: 25 May 2023 (09:52:24 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0103.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Nipah Virus, outbreak, inhibitors, QSAR, database, prediction algorithm
Online: 5 October 2018 (15:04:23 CEST)
REVIEW
|
doi:10.20944/preprints201809.0435.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Acute Myeloid Leukemia; FLT3; Tyrosine kinase inhibitors; resistance
Online: 21 September 2018 (10:28:34 CEST)
ARTICLE
|
doi:10.20944/preprints202110.0171.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
chronic myeloid leukemia; dasatinib; ponatinib; pimozide; STAT inhibitors; K562
Online: 11 October 2021 (16:17:32 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1726.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
dacomitinib; EGFR inhibitor; overall survival; pharmacokinetics; progression-free survival; proton pump inhibitors
Online: 27 October 2023 (07:06:07 CEST)
REVIEW
|
doi:10.20944/preprints202304.0564.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
serotonin antagonist/reuptake inhibitors; comorbidity; psychiatric disorders; trazodone; neurobiology; emotion
Online: 19 April 2023 (07:52:17 CEST)
REVIEW
|
doi:10.20944/preprints201907.0286.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 Gag; Gag inhibitors; Protease; Protease inhibitors; drug resistance mutations; drug design
Online: 25 July 2019 (10:05:03 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0279.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
NS3 inhibitors; allosteric inhibitors; NS4A; peptidomimetics; imidazole; hepatitis C virus; molecular dynamics; Flaviviridae; DSLS; binding assay
Online: 24 January 2020 (11:11:46 CET)
REVIEW
|
doi:10.20944/preprints202302.0205.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast cancer; ovarian cancer; PARP inhibitors; Alu repeats; protein-protein interactions
Online: 13 February 2023 (07:54:35 CET)
REVIEW
|
doi:10.20944/preprints201805.0129.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
BET inhibitors; HDAC inhibitors; pancreatic cancer; aberrant transcription; enhancers; transcription factors; distal regulatory elements; MYC; FOXA1; BRD4
Online: 8 May 2018 (10:47:27 CEST)
ARTICLE
|
doi:10.20944/preprints201911.0094.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
hPSCs; ROCK inhibitors; fasudil; cell survival; metabolism; differentiation
Online: 8 November 2019 (10:41:13 CET)
ARTICLE
|
doi:10.20944/preprints202307.1626.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Proton pump inhibitors; Clopidogrel; Stroke; Myocardial infarction
Online: 25 July 2023 (07:26:31 CEST)
REVIEW
|
doi:10.20944/preprints202405.0212.v1
Subject:
Oncology And Oncogenics,
Medicine And Pharmacology
Keywords:
Hepatocellular carcinoma (HCC); systemic therapies; bridging; liver transplantation (LT); Tyrosine Kinase Inhibitors (TKIs); Immune Checkpoint Inhibitors (ICIs)
Online: 6 May 2024 (04:52:05 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0503.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
HNSCC; PI3K inhibitors; ErbB inhibitor; targeted therapy
Online: 8 February 2024 (14:11:24 CET)
ARTICLE
|
doi:10.20944/preprints201706.0022.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
HPPD inhibitors; pharmacophore model; molecule docking; HipHop model; virtual screening; ChemDiv
Online: 5 June 2017 (05:16:39 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0542.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
safety analysis; targeted therapy; monoclonal antibody therapy; immune checkpoint inhibibitors; tyrosine kinase inhibitors; breast cancer; gynecological cancer; Helixor; Viscum album L.; PARP inhibitors; CDK 4/6 inhibitors
Online: 30 December 2022 (12:00:35 CET)
REVIEW
|
doi:10.20944/preprints202304.1236.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
FLT3 mutations; resistant/relapsed acute myeloid leukemia; tyrosine kinase inhibitors; gilteritinib
Online: 29 April 2023 (10:55:21 CEST)
REVIEW
|
doi:10.20944/preprints202306.1269.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
tumor microenvironment; extracellular matrix; proteoglycans; tumor-associated fibroblasts; tumor immunity; immune checkpoint inhibitors; tumor stroma; angiogenesis
Online: 19 June 2023 (03:16:16 CEST)
REVIEW
|
doi:10.20944/preprints202309.1061.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
prodrugs; HIV; AIDS; Nucleoside Reverse Transcriptase Inhibitors (NRTI); co-drugs; new drugs; medicinal chemistry
Online: 18 September 2023 (05:47:07 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0063.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Cx43; gap junctions; conductance; inhibitors; docking; IC50
Online: 5 April 2023 (12:30:58 CEST)
REVIEW
|
doi:10.20944/preprints202105.0140.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Adsorption; Scale Inhibitors; Fine sands; Colloids; Reservoir
Online: 7 May 2021 (10:42:36 CEST)
REVIEW
|
doi:10.20944/preprints202003.0378.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
China's COVID-19 Guide; Remdesivir; Xuebijing; Hydroxychloroquine; IL6 inhibitors; COVID-19
Online: 26 March 2020 (01:48:42 CET)
REVIEW
|
doi:10.20944/preprints202306.0128.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PD-L1; CTCs; immunotherapy; immune checkpoint inhibitors
Online: 2 June 2023 (04:28:01 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0449.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
herpes zoster; immune checkpoint inhibitors; standardized incidence ratio; cancer patients
Online: 7 February 2024 (14:34:28 CET)
ARTICLE
|
doi:10.20944/preprints202310.0751.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Drosophila; male meiosis; cyclin B; Cyclin-dependent kinase 1; Cyclin-dependent kinase inhibitors
Online: 12 October 2023 (05:32:28 CEST)
REVIEW
|
doi:10.20944/preprints202302.0380.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
serotonin antagonist/reuptake inhibitors; comorbidity; psychiatric disorders; neurological disorders; dementia; primary care
Online: 22 February 2023 (08:42:51 CET)
REVIEW
|
doi:10.20944/preprints202212.0026.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Advanced Hepatocellular carcinoma; Immune checkpoint inhibitors; Low middle-income countries; Financial Toxicity
Online: 1 December 2022 (10:33:14 CET)
REVIEW
|
doi:10.20944/preprints202310.2105.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
radiotherapy; CD8+ T cells; immune checkpoint inhibitors
Online: 31 October 2023 (17:22:30 CET)
ARTICLE
|
doi:10.20944/preprints201810.0133.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
aging; angiotensin-converting enzyme inhibitors; nutrient metabolism; genetic background; nutritional stress
Online: 29 October 2018 (10:33:59 CET)
REVIEW
|
doi:10.20944/preprints202311.0529.v1
Subject:
Public Health And Healthcare,
Primary Health Care
Keywords:
SARS-CoV-2; Papain-like protease; COVID-19; Molecular modelling; Molecular dynamics simulations; Drug discovery; Antiviral drugs; Inhibitors; Therapeutic agents; therapeutic targets; Irreversible inhibitors; Repurposing drugs
Online: 8 November 2023 (16:11:55 CET)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0638.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 26 May 2021 (13:14:06 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 25 January 2021 (15:01:17 CET)
REVIEW
|
doi:10.20944/preprints202110.0298.v1
Subject:
Medicine And Pharmacology,
Orthopedics And Sports Medicine
Keywords:
Osteoarthritis; LithoLexal; Lithothamnion; Disease-modifying adjunctive therapy; Anti-inflammatory agents; Cytokine inhibitors
Online: 20 October 2021 (22:49:47 CEST)
REVIEW
|
doi:10.20944/preprints202312.1388.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Rheb1; Rheb2; Cancer; mTOR; Hallmarks; Neurons; Rheb1 inhibitors
Online: 19 December 2023 (05:58:46 CET)
ARTICLE
|
doi:10.20944/preprints202308.0880.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
tyrosyl-DNA phosphodiesterase 1 (Tdp1); tyrosyl-DNA phosphodiesterase 2 (Tdp2); usnic acid; Tdp2 inhibitors; Tdp1 inhibitors
Online: 11 August 2023 (08:18:31 CEST)
REVIEW
|
doi:10.20944/preprints202011.0005.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminoacyl-tRNA synthetase, small molecule inhibitors, human diseases
Online: 2 November 2020 (09:09:37 CET)
ARTICLE
|
doi:10.20944/preprints201807.0199.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
ALS-inhibitors; horseweed; multiple-resistance; alternative chemical control
Online: 11 July 2018 (11:56:59 CEST)
REVIEW
|
doi:10.20944/preprints202307.2046.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CADD; SBDD; LBDD; kinase; small molecule kinase inhibitors
Online: 31 July 2023 (03:05:42 CEST)